PL2521452T3 - Tiazolo[5,4-d]pirymidyny i ich zastosowanie jako agrochemikaliów - Google Patents

Tiazolo[5,4-d]pirymidyny i ich zastosowanie jako agrochemikaliów

Info

Publication number
PL2521452T3
PL2521452T3 PL11732133T PL11732133T PL2521452T3 PL 2521452 T3 PL2521452 T3 PL 2521452T3 PL 11732133 T PL11732133 T PL 11732133T PL 11732133 T PL11732133 T PL 11732133T PL 2521452 T3 PL2521452 T3 PL 2521452T3
Authority
PL
Poland
Prior art keywords
thiazolo
agrochemicals
pyrimidines
Prior art date
Application number
PL11732133T
Other languages
English (en)
Polish (pl)
Inventor
William Brewster
Carla Klittich
Brent Rieder
Thomas Siddall
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PL2521452T3 publication Critical patent/PL2521452T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
PL11732133T 2010-01-07 2011-01-06 Tiazolo[5,4-d]pirymidyny i ich zastosowanie jako agrochemikaliów PL2521452T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29301410P 2010-01-07 2010-01-07
EP11732133.1A EP2521452B1 (en) 2010-01-07 2011-01-06 THIAZOLO[5,4-d]PYRIMIDINES AND THEIR USE AS AGROCHEMICALS
PCT/US2011/020351 WO2011085084A1 (en) 2010-01-07 2011-01-06 THIAZOLO[5,4-d] PYRIMIDINES AND THEIR USE AS AGROCHEMICALS

Publications (1)

Publication Number Publication Date
PL2521452T3 true PL2521452T3 (pl) 2015-05-29

Family

ID=44225056

Family Applications (1)

Application Number Title Priority Date Filing Date
PL11732133T PL2521452T3 (pl) 2010-01-07 2011-01-06 Tiazolo[5,4-d]pirymidyny i ich zastosowanie jako agrochemikaliów

Country Status (18)

Country Link
US (1) US8921382B2 (enExample)
EP (1) EP2521452B1 (enExample)
JP (1) JP5781090B2 (enExample)
KR (1) KR101814835B1 (enExample)
CN (1) CN102791135B (enExample)
BR (1) BR112012016866A2 (enExample)
CA (1) CA2786250A1 (enExample)
CL (1) CL2012001851A1 (enExample)
CO (1) CO6612238A2 (enExample)
ES (1) ES2529247T3 (enExample)
IN (1) IN2012DN06323A (enExample)
MX (1) MX2012007954A (enExample)
PL (1) PL2521452T3 (enExample)
PT (1) PT2521452E (enExample)
RU (1) RU2547721C2 (enExample)
UA (1) UA109780C2 (enExample)
WO (1) WO2011085084A1 (enExample)
ZA (1) ZA201204871B (enExample)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG177384A1 (en) 2009-06-29 2012-02-28 Incyte Corp Pyrimidinones as pi3k inhibitors
CA2842190A1 (en) 2011-07-19 2013-01-24 Infinity Pharmaceuticals Inc. Heterocyclic compounds and uses thereof
WO2013031694A1 (ja) * 2011-08-26 2013-03-07 富山化学工業株式会社 アミン化合物またはその塩
PL3196202T3 (pl) 2011-09-02 2019-09-30 Incyte Holdings Corporation Heterocykloaminy jako inhibitory pi3k
CN104220428A (zh) 2012-02-03 2014-12-17 巴斯夫欧洲公司 杀真菌嘧啶化合物
EP2809658B1 (en) 2012-02-03 2015-09-30 Basf Se Fungicidal pyrimidine compounds
WO2013135672A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
CN103668956B (zh) * 2012-09-21 2015-08-12 上海韬鸿化工科技有限公司 防螨虫整理剂、织物的防螨虫整理方法及防螨虫织物
EP2972299A4 (en) * 2013-03-15 2017-01-25 The Regents of The University of California Methods for identifying arthropod repellents and attractants, and compounds and compositions identified by such methods
WO2015191677A1 (en) 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
CN105594748A (zh) * 2014-10-15 2016-05-25 浙江新安化工集团股份有限公司 一种精准定向、高效的防治鳞翅目害虫的杀虫组合物及其使用方法
CN104391070B (zh) * 2014-12-05 2016-06-08 山东省城市供排水水质监测中心 一种水中烷基汞的检测方法
MD3831833T2 (ro) 2015-02-27 2023-04-30 Incyte Holdings Corp Procedee pentru prepararea unui inhibitor PI3K
WO2016149567A1 (en) 2015-03-18 2016-09-22 The Regents Of The University Of California Anthropod repellent chemicals
WO2016183063A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Crystalline forms of a pi3k inhibitor
CN105606755A (zh) * 2016-01-30 2016-05-25 郭庆龙 一种胺苯吡唑酮残留量的gc-nci-ms测定方法
JP7037507B2 (ja) 2017-01-26 2022-03-16 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
WO2018190351A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
CA3059675A1 (en) 2017-04-10 2018-10-18 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients
EP3611165B1 (en) 2017-04-11 2023-08-16 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compound, and agricultural and horticultural fungicide having this as active component
WO2018225829A1 (ja) 2017-06-08 2018-12-13 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
CA3101323A1 (en) 2018-06-01 2019-12-05 Incyte Corporation Dosing regimen for the treatment of pi3k related disorders
TWI828725B (zh) 2018-07-25 2024-01-11 日商三井化學植保股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
UA129572C2 (uk) 2020-02-11 2025-06-04 Сінгента Кроп Протекшн Аг Спосіб контролю грибів
CN112010848B (zh) * 2020-09-29 2021-12-24 南通大学 含三氟甲基吡啶联芳氧基结构的1,3,4-噁二唑类化合物的制备方法和应用
CN116250525B (zh) * 2023-03-08 2024-12-24 内蒙古民族大学 一种小型哺乳类剥制标本安全防腐剂及其制备方法

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) * 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
DE58908159D1 (de) 1988-03-09 1994-09-15 Ciba Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
US5034393A (en) 1989-07-27 1991-07-23 Dowelanco Fungicidal use of pyridopyrimidine, pteridine, pyrimidopyrimidine, pyrimidopyridazine, and pyrimido-1,2,4-triazine derivatives
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
US5326766A (en) 1992-08-19 1994-07-05 Dreikorn Barry A 4-(2-(4-(2-pyridinyloxy)phenyl)ethoxy)quinazoline and analogues thereof
ES2167586T3 (es) 1995-07-05 2002-05-16 Du Pont Pirimidinonas fungicidas.
CZ288498A3 (cs) 1996-03-11 1998-12-16 Novartis Ag Deriváty pyrimidin-4-onu jako pesticidní látky, způsob jejich přípravy a agrochemické prostředky, které je obsahují
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US6448262B1 (en) 1998-11-16 2002-09-10 American Cyanamid Company Pesticidal and parasiticidal use of 2-(substituted thio) thiazolo-[4,5-b]pyridine compounds
UA77407C2 (en) * 2001-01-31 2006-12-15 Bayer Cropscience Gmbh Herbicide-safener composition based on isoxosoline carboxylate safener, a method to control weeds and a method to lower the phytotoxicity of a herbicide
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
ATE363829T1 (de) 2001-09-10 2007-06-15 Basf Ag Pestizide und parasitizide di- und trifluorsubstituierte alkenverbindungen
EP1731523A4 (en) 2004-04-01 2009-08-12 Takeda Pharmaceutical THIAZOLOPYRIMIDINDERIVAT
JP5243960B2 (ja) 2005-10-21 2013-07-24 ダウ アグロサイエンシィズ エルエルシー 殺菌活性を有するチエノ−ピリミジン化合物
EP2044086A2 (en) 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
PT2562166E (pt) 2008-01-22 2015-10-28 Dow Agrosciences Llc Derivados de 5-fluoro-pirimidina como fungicidas
PL2317851T3 (pl) 2008-08-01 2014-06-30 Dow Agrosciences Llc Zastosowanie 5-fluorocytozyny jako fungicydu
US8609864B2 (en) 2009-01-23 2013-12-17 Purdue Pharmaceutical Products, L.P. Hydroxamic acid derivatives
CN101613362B (zh) * 2009-07-31 2011-11-16 南京工业大学 3-羰基-6-乙氧甲酰基-噻唑并嘧啶类化合物及其合成方法和用途
MX2012001622A (es) 2009-08-07 2012-04-11 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona.

Also Published As

Publication number Publication date
ES2529247T3 (es) 2015-02-18
WO2011085084A1 (en) 2011-07-14
JP2013516476A (ja) 2013-05-13
BR112012016866A2 (pt) 2015-09-01
JP5781090B2 (ja) 2015-09-16
RU2547721C2 (ru) 2015-04-10
US8921382B2 (en) 2014-12-30
RU2012133570A (ru) 2014-02-20
CA2786250A1 (en) 2011-07-14
CN102791135B (zh) 2015-05-20
US20110166164A1 (en) 2011-07-07
IN2012DN06323A (enExample) 2015-10-02
EP2521452B1 (en) 2014-12-24
UA109780C2 (uk) 2015-10-12
KR20120115538A (ko) 2012-10-18
CL2012001851A1 (es) 2012-12-14
HK1176236A1 (en) 2013-07-26
EP2521452A4 (en) 2013-07-03
MX2012007954A (es) 2012-08-03
KR101814835B1 (ko) 2018-01-04
EP2521452A1 (en) 2012-11-14
CN102791135A (zh) 2012-11-21
CO6612238A2 (es) 2013-02-01
ZA201204871B (en) 2013-09-25
PT2521452E (pt) 2015-02-24

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