CN102791135B - 噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 - Google Patents

噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 Download PDF

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Publication number
CN102791135B
CN102791135B CN201180012818.XA CN201180012818A CN102791135B CN 102791135 B CN102791135 B CN 102791135B CN 201180012818 A CN201180012818 A CN 201180012818A CN 102791135 B CN102791135 B CN 102791135B
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China
Prior art keywords
compound
spp
phenyl
ethyl
thiazole
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Expired - Fee Related
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CN201180012818.XA
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English (en)
Chinese (zh)
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CN102791135A (zh
Inventor
W.布鲁斯特
C.克里蒂科
B.里德
T.西德尔
姚成林
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Corteva Agriscience LLC
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Dow AgroSciences LLC
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Zoology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
  • Plural Heterocyclic Compounds (AREA)
CN201180012818.XA 2010-01-07 2011-01-06 噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 Expired - Fee Related CN102791135B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29301410P 2010-01-07 2010-01-07
US61/293,014 2010-01-07
PCT/US2011/020351 WO2011085084A1 (en) 2010-01-07 2011-01-06 THIAZOLO[5,4-d] PYRIMIDINES AND THEIR USE AS AGROCHEMICALS

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Publication Number Publication Date
CN102791135A CN102791135A (zh) 2012-11-21
CN102791135B true CN102791135B (zh) 2015-05-20

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US (1) US8921382B2 (enExample)
EP (1) EP2521452B1 (enExample)
JP (1) JP5781090B2 (enExample)
KR (1) KR101814835B1 (enExample)
CN (1) CN102791135B (enExample)
BR (1) BR112012016866A2 (enExample)
CA (1) CA2786250A1 (enExample)
CL (1) CL2012001851A1 (enExample)
CO (1) CO6612238A2 (enExample)
ES (1) ES2529247T3 (enExample)
IN (1) IN2012DN06323A (enExample)
MX (1) MX2012007954A (enExample)
PL (1) PL2521452T3 (enExample)
PT (1) PT2521452E (enExample)
RU (1) RU2547721C2 (enExample)
UA (1) UA109780C2 (enExample)
WO (1) WO2011085084A1 (enExample)
ZA (1) ZA201204871B (enExample)

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WO2013012918A1 (en) 2011-07-19 2013-01-24 Infinity Pharmaceuticals Inc. Heterocyclic compounds and uses thereof
JPWO2013031694A1 (ja) * 2011-08-26 2015-03-23 富山化学工業株式会社 アミン化合物またはその塩
LT3196202T (lt) 2011-09-02 2019-07-10 Incyte Holdings Corporation Heterociklilaminai, kaip pi3k slopikliai
CA2862346A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
JP2015511940A (ja) 2012-02-03 2015-04-23 ビーエーエスエフ ソシエタス・ヨーロピアBasf Se 殺菌性ピリミジン化合物
WO2013135672A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
CN103668956B (zh) * 2012-09-21 2015-08-12 上海韬鸿化工科技有限公司 防螨虫整理剂、织物的防螨虫整理方法及防螨虫织物
EP3409115A3 (en) * 2013-03-15 2019-02-27 The Regents of The University of California Methods for identifying arthropod repellents, and compounds and compositions identified by such methods
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
CN105594748A (zh) * 2014-10-15 2016-05-25 浙江新安化工集团股份有限公司 一种精准定向、高效的防治鳞翅目害虫的杀虫组合物及其使用方法
CN104391070B (zh) * 2014-12-05 2016-06-08 山东省城市供排水水质监测中心 一种水中烷基汞的检测方法
CN117736209A (zh) 2015-02-27 2024-03-22 因赛特控股公司 Pi3k抑制剂的盐及其制备方法
US20160272612A1 (en) 2015-03-18 2016-09-22 The Regents Of The University Of California Anthropod repellent chemicals
WO2016183063A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Crystalline forms of a pi3k inhibitor
CN105606755A (zh) * 2016-01-30 2016-05-25 郭庆龙 一种胺苯吡唑酮残留量的gc-nci-ms测定方法
EP3575286B1 (en) 2017-01-26 2022-05-11 Mitsui Chemicals Agro, Inc. Pyridone compound and bactericide for agricultural and horticultural use, which uses said compound as active ingredient
WO2018190351A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
CA3059675A1 (en) 2017-04-10 2018-10-18 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients
US11178870B2 (en) 2017-04-11 2021-11-23 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
EP3636636B1 (en) 2017-06-08 2022-07-06 Mitsui Chemicals Agro, Inc. Pyridone compound and agricultural and horticultural fungicide
PE20211208A1 (es) 2018-06-01 2021-07-05 Incyte Corp Regimen de dosificacion para el tratamiento de trastornos relacionados con pi3k
US12114658B2 (en) 2018-07-25 2024-10-15 Mitsui Chemicals Crop & Life Solutions, Inc. Compounds having a nitrogen-containing unsaturated six-membered ring and agricultural and horticultural fungicides containing the same as active ingredients
CN115003160B (zh) 2020-02-11 2024-04-30 先正达农作物保护股份公司 控制真菌的方法
CN112010848B (zh) * 2020-09-29 2021-12-24 南通大学 含三氟甲基吡啶联芳氧基结构的1,3,4-噁二唑类化合物的制备方法和应用
CN116250525B (zh) * 2023-03-08 2024-12-24 内蒙古民族大学 一种小型哺乳类剥制标本安全防腐剂及其制备方法

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PL2521452T3 (pl) 2015-05-29
JP2013516476A (ja) 2013-05-13
EP2521452A1 (en) 2012-11-14
RU2012133570A (ru) 2014-02-20
JP5781090B2 (ja) 2015-09-16
EP2521452A4 (en) 2013-07-03
US20110166164A1 (en) 2011-07-07
IN2012DN06323A (enExample) 2015-10-02
RU2547721C2 (ru) 2015-04-10
US8921382B2 (en) 2014-12-30
EP2521452B1 (en) 2014-12-24
BR112012016866A2 (pt) 2015-09-01
HK1176236A1 (en) 2013-07-26
PT2521452E (pt) 2015-02-24
CA2786250A1 (en) 2011-07-14
CO6612238A2 (es) 2013-02-01
ZA201204871B (en) 2013-09-25
CL2012001851A1 (es) 2012-12-14
KR20120115538A (ko) 2012-10-18
MX2012007954A (es) 2012-08-03
KR101814835B1 (ko) 2018-01-04
UA109780C2 (uk) 2015-10-12
ES2529247T3 (es) 2015-02-18
CN102791135A (zh) 2012-11-21
WO2011085084A1 (en) 2011-07-14

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