PT2521452E - Tiazolo[5,4-d]pirimidinas e a sua utilização como agroquímicos - Google Patents

Tiazolo[5,4-d]pirimidinas e a sua utilização como agroquímicos Download PDF

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Publication number
PT2521452E
PT2521452E PT117321331T PT11732133T PT2521452E PT 2521452 E PT2521452 E PT 2521452E PT 117321331 T PT117321331 T PT 117321331T PT 11732133 T PT11732133 T PT 11732133T PT 2521452 E PT2521452 E PT 2521452E
Authority
PT
Portugal
Prior art keywords
thiazolo
agrochemicals
pyrimidines
Prior art date
Application number
PT117321331T
Other languages
English (en)
Inventor
William Brewster
Carla Klittich
Brent Rieder
Thomas Siddall
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PT2521452E publication Critical patent/PT2521452E/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
PT117321331T 2010-01-07 2011-01-06 Tiazolo[5,4-d]pirimidinas e a sua utilização como agroquímicos PT2521452E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US29301410P 2010-01-07 2010-01-07

Publications (1)

Publication Number Publication Date
PT2521452E true PT2521452E (pt) 2015-02-24

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
PT117321331T PT2521452E (pt) 2010-01-07 2011-01-06 Tiazolo[5,4-d]pirimidinas e a sua utilização como agroquímicos

Country Status (19)

Country Link
US (1) US8921382B2 (pt)
EP (1) EP2521452B1 (pt)
JP (1) JP5781090B2 (pt)
KR (1) KR101814835B1 (pt)
CN (1) CN102791135B (pt)
BR (1) BR112012016866A2 (pt)
CA (1) CA2786250A1 (pt)
CL (1) CL2012001851A1 (pt)
CO (1) CO6612238A2 (pt)
ES (1) ES2529247T3 (pt)
HK (1) HK1176236A1 (pt)
IN (1) IN2012DN06323A (pt)
MX (1) MX2012007954A (pt)
PL (1) PL2521452T3 (pt)
PT (1) PT2521452E (pt)
RU (1) RU2547721C2 (pt)
UA (1) UA109780C2 (pt)
WO (1) WO2011085084A1 (pt)
ZA (1) ZA201204871B (pt)

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AU2012284091B2 (en) 2011-07-19 2015-11-12 Infinity Pharmaceuticals Inc. Heterocyclic compounds and uses thereof
WO2013031694A1 (ja) * 2011-08-26 2013-03-07 富山化学工業株式会社 アミン化合物またはその塩
PE20181272A1 (es) 2011-09-02 2018-08-03 Incyte Holdings Corp Heterociclilaminas como inhibidores de pi3k
BR112014018812A8 (pt) 2012-02-03 2017-07-11 Basf Se Compostos, processo para preparar os compostos i, composição agroquímica, método para combater fungos nocivos fitopagênicos, uso dos compostos de fórmula i e semente
WO2013113863A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
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AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
CN103668956B (zh) * 2012-09-21 2015-08-12 上海韬鸿化工科技有限公司 防螨虫整理剂、织物的防螨虫整理方法及防螨虫织物
EP2972299A4 (en) * 2013-03-15 2017-01-25 The Regents of The University of California Methods for identifying arthropod repellents and attractants, and compounds and compositions identified by such methods
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
CN105594748A (zh) * 2014-10-15 2016-05-25 浙江新安化工集团股份有限公司 一种精准定向、高效的防治鳞翅目害虫的杀虫组合物及其使用方法
CN104391070B (zh) * 2014-12-05 2016-06-08 山东省城市供排水水质监测中心 一种水中烷基汞的检测方法
CR20210055A (es) 2015-02-27 2021-04-27 Incyte Corp SALES DE IHNIBIDOR DE PI3K Y PROCESOS DE PREPARACIÓN (Divisional 2017-0389)
EP3270692A4 (en) 2015-03-18 2019-02-13 The Regents of the University of California ANTI-ARTHROPOD CHEMICALS
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor
CN105606755A (zh) * 2016-01-30 2016-05-25 郭庆龙 一种胺苯吡唑酮残留量的gc-nci-ms测定方法
JP7037507B2 (ja) 2017-01-26 2022-03-16 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
EP3611166B1 (en) 2017-04-10 2022-09-21 Mitsui Chemicals Agro, Inc. Pyridone compound, and agricultural and horticultural fungicide having this as active component
CA3059675A1 (en) 2017-04-10 2018-10-18 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients
US11178870B2 (en) 2017-04-11 2021-11-23 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
JP7157738B2 (ja) 2017-06-08 2022-10-20 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
TWI828725B (zh) 2018-07-25 2024-01-11 日商三井化學植保股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
CN112010848B (zh) * 2020-09-29 2021-12-24 南通大学 含三氟甲基吡啶联芳氧基结构的1,3,4-噁二唑类化合物的制备方法和应用

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Also Published As

Publication number Publication date
EP2521452B1 (en) 2014-12-24
BR112012016866A2 (pt) 2015-09-01
US20110166164A1 (en) 2011-07-07
CA2786250A1 (en) 2011-07-14
RU2547721C2 (ru) 2015-04-10
CL2012001851A1 (es) 2012-12-14
KR101814835B1 (ko) 2018-01-04
JP5781090B2 (ja) 2015-09-16
PL2521452T3 (pl) 2015-05-29
CN102791135A (zh) 2012-11-21
ES2529247T3 (es) 2015-02-18
CO6612238A2 (es) 2013-02-01
UA109780C2 (uk) 2015-10-12
MX2012007954A (es) 2012-08-03
ZA201204871B (en) 2013-09-25
WO2011085084A1 (en) 2011-07-14
EP2521452A4 (en) 2013-07-03
JP2013516476A (ja) 2013-05-13
RU2012133570A (ru) 2014-02-20
CN102791135B (zh) 2015-05-20
IN2012DN06323A (pt) 2015-10-02
US8921382B2 (en) 2014-12-30
KR20120115538A (ko) 2012-10-18
EP2521452A1 (en) 2012-11-14
HK1176236A1 (en) 2013-07-26

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