PT2521452E - Tiazolo[5,4-d]pirimidinas e a sua utilização como agroquímicos - Google Patents
Tiazolo[5,4-d]pirimidinas e a sua utilização como agroquímicos Download PDFInfo
- Publication number
- PT2521452E PT2521452E PT117321331T PT11732133T PT2521452E PT 2521452 E PT2521452 E PT 2521452E PT 117321331 T PT117321331 T PT 117321331T PT 11732133 T PT11732133 T PT 11732133T PT 2521452 E PT2521452 E PT 2521452E
- Authority
- PT
- Portugal
- Prior art keywords
- thiazolo
- agrochemicals
- pyrimidines
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US29301410P | 2010-01-07 | 2010-01-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT2521452E true PT2521452E (pt) | 2015-02-24 |
Family
ID=44225056
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT117321331T PT2521452E (pt) | 2010-01-07 | 2011-01-06 | Tiazolo[5,4-d]pirimidinas e a sua utilização como agroquímicos |
Country Status (19)
Country | Link |
---|---|
US (1) | US8921382B2 (pt) |
EP (1) | EP2521452B1 (pt) |
JP (1) | JP5781090B2 (pt) |
KR (1) | KR101814835B1 (pt) |
CN (1) | CN102791135B (pt) |
BR (1) | BR112012016866A2 (pt) |
CA (1) | CA2786250A1 (pt) |
CL (1) | CL2012001851A1 (pt) |
CO (1) | CO6612238A2 (pt) |
ES (1) | ES2529247T3 (pt) |
HK (1) | HK1176236A1 (pt) |
IN (1) | IN2012DN06323A (pt) |
MX (1) | MX2012007954A (pt) |
PL (1) | PL2521452T3 (pt) |
PT (1) | PT2521452E (pt) |
RU (1) | RU2547721C2 (pt) |
UA (1) | UA109780C2 (pt) |
WO (1) | WO2011085084A1 (pt) |
ZA (1) | ZA201204871B (pt) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
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AR077280A1 (es) | 2009-06-29 | 2011-08-17 | Incyte Corp | Pirimidinonas como inhibidores de pi3k, y composiciones farmaceuticas que los comprenden |
AU2012284091B2 (en) | 2011-07-19 | 2015-11-12 | Infinity Pharmaceuticals Inc. | Heterocyclic compounds and uses thereof |
WO2013031694A1 (ja) * | 2011-08-26 | 2013-03-07 | 富山化学工業株式会社 | アミン化合物またはその塩 |
PE20181272A1 (es) | 2011-09-02 | 2018-08-03 | Incyte Holdings Corp | Heterociclilaminas como inhibidores de pi3k |
BR112014018812A8 (pt) | 2012-02-03 | 2017-07-11 | Basf Se | Compostos, processo para preparar os compostos i, composição agroquímica, método para combater fungos nocivos fitopagênicos, uso dos compostos de fórmula i e semente |
WO2013113863A1 (en) | 2012-02-03 | 2013-08-08 | Basf Se | Fungicidal pyrimidine compounds |
WO2013135672A1 (en) | 2012-03-13 | 2013-09-19 | Basf Se | Fungicidal pyrimidine compounds |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
CN103668956B (zh) * | 2012-09-21 | 2015-08-12 | 上海韬鸿化工科技有限公司 | 防螨虫整理剂、织物的防螨虫整理方法及防螨虫织物 |
EP2972299A4 (en) * | 2013-03-15 | 2017-01-25 | The Regents of The University of California | Methods for identifying arthropod repellents and attractants, and compounds and compositions identified by such methods |
US10077277B2 (en) | 2014-06-11 | 2018-09-18 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors |
CN105594748A (zh) * | 2014-10-15 | 2016-05-25 | 浙江新安化工集团股份有限公司 | 一种精准定向、高效的防治鳞翅目害虫的杀虫组合物及其使用方法 |
CN104391070B (zh) * | 2014-12-05 | 2016-06-08 | 山东省城市供排水水质监测中心 | 一种水中烷基汞的检测方法 |
CR20210055A (es) | 2015-02-27 | 2021-04-27 | Incyte Corp | SALES DE IHNIBIDOR DE PI3K Y PROCESOS DE PREPARACIÓN (Divisional 2017-0389) |
EP3270692A4 (en) | 2015-03-18 | 2019-02-13 | The Regents of the University of California | ANTI-ARTHROPOD CHEMICALS |
US9988401B2 (en) | 2015-05-11 | 2018-06-05 | Incyte Corporation | Crystalline forms of a PI3K inhibitor |
CN105606755A (zh) * | 2016-01-30 | 2016-05-25 | 郭庆龙 | 一种胺苯吡唑酮残留量的gc-nci-ms测定方法 |
JP7037507B2 (ja) | 2017-01-26 | 2022-03-16 | 三井化学アグロ株式会社 | ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤 |
EP3611166B1 (en) | 2017-04-10 | 2022-09-21 | Mitsui Chemicals Agro, Inc. | Pyridone compound, and agricultural and horticultural fungicide having this as active component |
CA3059675A1 (en) | 2017-04-10 | 2018-10-18 | Mitsui Chemicals Agro, Inc. | Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients |
US11178870B2 (en) | 2017-04-11 | 2021-11-23 | Mitsui Chemicals Agro, Inc. | Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients |
JP7157738B2 (ja) | 2017-06-08 | 2022-10-20 | 三井化学アグロ株式会社 | ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤 |
TWI828725B (zh) | 2018-07-25 | 2024-01-11 | 日商三井化學植保股份有限公司 | 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑 |
CN112010848B (zh) * | 2020-09-29 | 2021-12-24 | 南通大学 | 含三氟甲基吡啶联芳氧基结构的1,3,4-噁二唑类化合物的制备方法和应用 |
Family Cites Families (29)
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US3309359A (en) | 1965-10-22 | 1967-03-14 | Hoffmann La Roche | N-mono-acyl-5-fluorocytosine derivatives and process |
US3368938A (en) | 1966-01-13 | 1968-02-13 | Hoffmann La Roche | Controlling fungi with 5-fluorocytosine |
US3868373A (en) | 1970-01-27 | 1975-02-25 | Hoffmann La Roche | 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines |
CH579057A5 (pt) | 1973-09-07 | 1976-08-31 | Hoffmann La Roche | |
FR2530636A1 (fr) * | 1982-07-23 | 1984-01-27 | Rhone Poulenc Agrochimie | Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides |
GR80171B (en) | 1983-08-29 | 1985-01-02 | Ciba Geigy Ag | N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use |
US4845081A (en) | 1984-10-18 | 1989-07-04 | University Of Florida | Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes |
ATE109776T1 (de) | 1988-03-09 | 1994-08-15 | Ciba Geigy Ag | Mittel zum schutz von pflanzen gegen krankheiten. |
DE3821711A1 (de) | 1988-06-28 | 1990-02-08 | Bayer Ag | Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
US5034393A (en) | 1989-07-27 | 1991-07-23 | Dowelanco | Fungicidal use of pyridopyrimidine, pteridine, pyrimidopyrimidine, pyrimidopyridazine, and pyrimido-1,2,4-triazine derivatives |
JP3109012B2 (ja) | 1992-06-18 | 2000-11-13 | クミアイ化学工業株式会社 | チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤 |
JP3217191B2 (ja) * | 1992-07-16 | 2001-10-09 | ビーエーエスエフ アクチェンゲゼルシャフト | ヘテロ芳香族化合物およびこれを含有する植物保護剤 |
US5326766A (en) | 1992-08-19 | 1994-07-05 | Dreikorn Barry A | 4-(2-(4-(2-pyridinyloxy)phenyl)ethoxy)quinazoline and analogues thereof |
AU6478396A (en) | 1995-07-05 | 1997-02-05 | E.I. Du Pont De Nemours And Company | Fungicidal pyrimidinones |
ATE216999T1 (de) | 1996-03-11 | 2002-05-15 | Syngenta Participations Ag | Pyrimidin-4-on derivate als pestizidesmittel |
HRP970239B1 (en) | 1997-05-09 | 2004-04-30 | Inst Ru Er Bouekovic | Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity |
GT199900185A (es) | 1998-11-06 | 2001-04-18 | Novedosa pirimidin-4-enamina como fungicida. | |
US6448262B1 (en) * | 1998-11-16 | 2002-09-10 | American Cyanamid Company | Pesticidal and parasiticidal use of 2-(substituted thio) thiazolo-[4,5-b]pyridine compounds |
CN1243474C (zh) * | 2001-01-31 | 2006-03-01 | 拜尔作物科学有限公司 | 基于异噁唑啉羧酸酯安全剂的除草剂-安全剂组合物 |
WO2003018051A1 (en) | 2001-08-27 | 2003-03-06 | Vic Jira | Anti-fungal composition |
EP1427287B1 (en) * | 2001-09-10 | 2007-06-06 | Basf Aktiengesellschaft | Pesticidal and parasitical di-and trifluorosubstituted alkene compounds |
EP1731523A4 (en) * | 2004-04-01 | 2009-08-12 | Takeda Pharmaceutical | THIAZOLOPYRIMIDINE DERIVATIVE |
WO2007046809A1 (en) | 2005-10-21 | 2007-04-26 | Dow Agrosciences Llc | Thieno-pyrimidine compounds having fungicidal activity |
US20080004253A1 (en) * | 2006-06-30 | 2008-01-03 | Bryan James Branstetter | Thiazolopyrimidine modulators of TRPV1 |
PL2562162T3 (pl) | 2008-01-22 | 2016-01-29 | Dow Agrosciences Llc | Pochodne N-cyjano-4-amino-5-fluoropirymidyny jako fungicydy |
CN104521977A (zh) | 2008-08-01 | 2015-04-22 | 陶氏益农公司 | 5-氟胞嘧啶作为杀真菌剂的用途 |
PL2389375T3 (pl) | 2009-01-23 | 2015-11-30 | Euro Celtique Sa | Pochodne kwasu hydroksamowego |
CN101613362B (zh) * | 2009-07-31 | 2011-11-16 | 南京工业大学 | 3-羰基-6-乙氧甲酰基-噻唑并嘧啶类化合物及其合成方法和用途 |
KR101743791B1 (ko) | 2009-08-07 | 2017-06-05 | 다우 아그로사이언시즈 엘엘씨 | N1-술포닐-5-플루오로피리미디논 유도체 |
-
2011
- 2011-01-06 UA UAA201209585A patent/UA109780C2/uk unknown
- 2011-01-06 ES ES11732133.1T patent/ES2529247T3/es active Active
- 2011-01-06 MX MX2012007954A patent/MX2012007954A/es active IP Right Grant
- 2011-01-06 IN IN6323DEN2012 patent/IN2012DN06323A/en unknown
- 2011-01-06 EP EP11732133.1A patent/EP2521452B1/en active Active
- 2011-01-06 CA CA2786250A patent/CA2786250A1/en not_active Abandoned
- 2011-01-06 BR BRBR112012016866-5A patent/BR112012016866A2/pt not_active Application Discontinuation
- 2011-01-06 PL PL11732133T patent/PL2521452T3/pl unknown
- 2011-01-06 PT PT117321331T patent/PT2521452E/pt unknown
- 2011-01-06 WO PCT/US2011/020351 patent/WO2011085084A1/en active Application Filing
- 2011-01-06 US US12/985,772 patent/US8921382B2/en not_active Expired - Fee Related
- 2011-01-06 CN CN201180012818.XA patent/CN102791135B/zh not_active Expired - Fee Related
- 2011-01-06 RU RU2012133570/13A patent/RU2547721C2/ru not_active IP Right Cessation
- 2011-01-06 KR KR1020127020594A patent/KR101814835B1/ko active IP Right Grant
- 2011-01-06 JP JP2012548116A patent/JP5781090B2/ja not_active Expired - Fee Related
-
2012
- 2012-06-29 ZA ZA2012/04871A patent/ZA201204871B/en unknown
- 2012-07-06 CL CL2012001851A patent/CL2012001851A1/es unknown
- 2012-08-03 CO CO12131428A patent/CO6612238A2/es active IP Right Grant
-
2013
- 2013-03-26 HK HK13103749.3A patent/HK1176236A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EP2521452B1 (en) | 2014-12-24 |
BR112012016866A2 (pt) | 2015-09-01 |
US20110166164A1 (en) | 2011-07-07 |
CA2786250A1 (en) | 2011-07-14 |
RU2547721C2 (ru) | 2015-04-10 |
CL2012001851A1 (es) | 2012-12-14 |
KR101814835B1 (ko) | 2018-01-04 |
JP5781090B2 (ja) | 2015-09-16 |
PL2521452T3 (pl) | 2015-05-29 |
CN102791135A (zh) | 2012-11-21 |
ES2529247T3 (es) | 2015-02-18 |
CO6612238A2 (es) | 2013-02-01 |
UA109780C2 (uk) | 2015-10-12 |
MX2012007954A (es) | 2012-08-03 |
ZA201204871B (en) | 2013-09-25 |
WO2011085084A1 (en) | 2011-07-14 |
EP2521452A4 (en) | 2013-07-03 |
JP2013516476A (ja) | 2013-05-13 |
RU2012133570A (ru) | 2014-02-20 |
CN102791135B (zh) | 2015-05-20 |
IN2012DN06323A (pt) | 2015-10-02 |
US8921382B2 (en) | 2014-12-30 |
KR20120115538A (ko) | 2012-10-18 |
EP2521452A1 (en) | 2012-11-14 |
HK1176236A1 (en) | 2013-07-26 |
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