PH25532A - Novel n-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives, pharm,aceutical composition containing said compound, method of use thereof - Google Patents

Novel n-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives, pharm,aceutical composition containing said compound, method of use thereof

Info

Publication number
PH25532A
PH25532A PH37085A PH37085A PH25532A PH 25532 A PH25532 A PH 25532A PH 37085 A PH37085 A PH 37085A PH 37085 A PH37085 A PH 37085A PH 25532 A PH25532 A PH 25532A
Authority
PH
Philippines
Prior art keywords
alk
piperidinyl
novel
pharm
compound
Prior art date
Application number
PH37085A
Other languages
English (en)
Inventor
Frans Eduard Janssens
Joseph Leo Ghislanus Torremans
Gaston Stanislas Mercell Diels
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PH25532A publication Critical patent/PH25532A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Lubricants (AREA)
PH37085A 1987-06-19 1988-06-17 Novel n-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives, pharm,aceutical composition containing said compound, method of use thereof PH25532A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6389987A 1987-06-19 1987-06-19

Publications (1)

Publication Number Publication Date
PH25532A true PH25532A (en) 1991-07-24

Family

ID=22052235

Family Applications (1)

Application Number Title Priority Date Filing Date
PH37085A PH25532A (en) 1987-06-19 1988-06-17 Novel n-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives, pharm,aceutical composition containing said compound, method of use thereof

Country Status (22)

Country Link
US (1) US4897401A (cs)
EP (1) EP0295742B1 (cs)
JP (1) JP2609464B2 (cs)
KR (1) KR970001158B1 (cs)
CN (1) CN1029964C (cs)
AT (1) ATE79878T1 (cs)
AU (1) AU600144B2 (cs)
CA (1) CA1324133C (cs)
DE (1) DE3874013T2 (cs)
DK (1) DK169761B1 (cs)
ES (1) ES2045083T3 (cs)
FI (1) FI90233C (cs)
GR (1) GR3006205T3 (cs)
HU (1) HU201755B (cs)
IE (1) IE61728B1 (cs)
IL (1) IL86788A (cs)
NO (1) NO167803C (cs)
NZ (1) NZ224928A (cs)
PH (1) PH25532A (cs)
PT (1) PT87742B (cs)
SU (1) SU1644717A3 (cs)
ZA (1) ZA884346B (cs)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8716313D0 (en) * 1987-07-10 1987-08-19 Janssen Pharmaceutica Nv 2-(heterocyclylalkyl)imidazopyridines
GB8900380D0 (en) * 1989-01-09 1989-03-08 Janssen Pharmaceutica Nv 2-aminopyrimidinone derivatives
PH30434A (en) * 1989-04-07 1997-05-09 Janssen Pharmaceutica Nv Hydroxyalkylfuranyl derivatives
US5272150A (en) * 1989-04-07 1993-12-21 Janssen Pharmaceutica N.V. Hydroxyalkylfuranyl derivatives
US5217980A (en) * 1990-07-19 1993-06-08 Janssen Pharmaceutica N.V. Oxazolyl and piperidinyl substituted benimidazolyl compounds
NZ238863A (en) * 1990-07-19 1993-03-26 Janssen Pharmaceutica Nv Substituted thiazolyl and pyridinyl derivatives
KR100190299B1 (ko) * 1990-07-19 1999-06-01 디르크 반테 신규한 옥사졸릴 유도체
US5478858A (en) * 1993-12-17 1995-12-26 The Procter & Gamble Company 5-(2-imidazolinylamino) benzimidazole compounds useful as alpha-2 adrenoceptor agonists
FR2725986B1 (fr) * 1994-10-21 1996-11-29 Adir Nouveaux derives de piperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
KR100731271B1 (ko) 1999-06-28 2007-06-21 얀센 파마슈티카 엔.브이. 호흡기 신시티움 바이러스 복제 억제제
HK1046141B (zh) 1999-06-28 2006-09-22 詹森药业有限公司 呼吸系统的合胞体病毒复制抑制剂
DE60008382T2 (de) 1999-06-28 2004-12-02 Janssen Pharmaceutica N.V. Respiratorisches syncytialvirus replikation inhibitoren
BR0207297A (pt) 2001-02-15 2005-04-19 King Pharmaceuticals Inc Composição farmacêutica em forma sólida e método de preparar uma forma de dosagem sólida de um ingrediente farmaceuticamente ativo
US7101569B2 (en) 2001-08-14 2006-09-05 Franz G Andrew Methods of administering levothyroxine pharmaceutical compositions
EP1479676A1 (en) * 2003-05-19 2004-11-24 Aventis Pharma Deutschland GmbH Benzimidazole-derivatives as factor xa inhibitors
NZ571898A (en) * 2003-06-24 2010-01-29 Pfizer Prod Inc Reaction of 2-chloro-8-benzyloxyquinoline with 2-nitrophenylamine in the presence of 1,2-bis(diphenylphosphino)ethane (dppe), palladium catalyst and a base

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4219559A (en) * 1979-01-10 1980-08-26 Janssen Pharmaceutica N.V. N-Heterocyclyl-4-piperidinamines
US4556660A (en) * 1982-07-12 1985-12-03 Janssen Pharmaceutica N.V. N-(Bicyclic heterocyclyl)-4-piperidinamines
US4634704A (en) * 1983-10-06 1987-01-06 Janssen Pharmaceutica, N.V. Anti-allergic five membered heterocyclic ring containing N-(bicyclic heterocycyl)-4-piperidinamines
US4695569A (en) * 1983-11-30 1987-09-22 Janssen Pharmaceutica N.V. Bicyclic heterocyclyl containing N-(bicyclic heterocyclyl)-4-piperidinamines
US4588722A (en) * 1984-01-09 1986-05-13 Janssen Pharmaceutica N.V. N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives
CA1327579C (en) * 1986-02-03 1994-03-08 Frans Eduard Janssens Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines
CA1317939C (en) * 1987-07-01 1993-05-18 Janssen Pharmaceutica Naamloze Vennootschap ¬(bicyclic heterocyclyl)methyl and -hetero| substituted hexahydro-1h-azepines and pyrrolidines

Also Published As

Publication number Publication date
IE61728B1 (en) 1994-11-30
AU1810988A (en) 1988-12-22
NO882641L (no) 1988-12-20
IL86788A (en) 1992-08-18
NZ224928A (en) 1990-04-26
CA1324133C (en) 1993-11-09
DE3874013D1 (de) 1992-10-01
GR3006205T3 (cs) 1993-06-21
US4897401A (en) 1990-01-30
HU201755B (en) 1990-12-28
JPS6425776A (en) 1989-01-27
SU1644717A3 (ru) 1991-04-23
DK333288A (da) 1988-12-20
PT87742A (pt) 1988-07-01
EP0295742B1 (en) 1992-08-26
DK333288D0 (da) 1988-06-17
DK169761B1 (da) 1995-02-20
FI90233B (fi) 1993-09-30
ZA884346B (en) 1990-02-28
FI90233C (fi) 1994-01-10
IE881849L (en) 1988-12-19
CN88103784A (zh) 1988-12-28
FI882909A0 (fi) 1988-06-17
IL86788A0 (en) 1988-11-30
HUT48628A (en) 1989-06-28
NO167803C (no) 1991-12-11
KR890000484A (ko) 1989-03-15
AU600144B2 (en) 1990-08-02
KR970001158B1 (ko) 1997-01-29
CN1029964C (zh) 1995-10-11
FI882909A7 (fi) 1988-12-20
ATE79878T1 (de) 1992-09-15
DE3874013T2 (de) 1993-01-07
NO882641D0 (no) 1988-06-15
JP2609464B2 (ja) 1997-05-14
ES2045083T3 (es) 1994-01-16
EP0295742A1 (en) 1988-12-21
PT87742B (pt) 1992-10-30
NO167803B (no) 1991-09-02

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