PH22338A - 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines - Google Patents

1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines

Info

Publication number
PH22338A
PH22338A PH31451A PH31451A PH22338A PH 22338 A PH22338 A PH 22338A PH 31451 A PH31451 A PH 31451A PH 31451 A PH31451 A PH 31451A PH 22338 A PH22338 A PH 22338A
Authority
PH
Philippines
Prior art keywords
imidazo
carbon atoms
group
quinolines
quinolin
Prior art date
Application number
PH31451A
Other languages
English (en)
Inventor
John F Gerster
Original Assignee
Riker Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Riker Laboratories Inc filed Critical Riker Laboratories Inc
Publication of PH22338A publication Critical patent/PH22338A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Physical Water Treatments (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Macromonomer-Based Addition Polymer (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Alarm Systems (AREA)
  • Quinoline Compounds (AREA)
  • Luminescent Compositions (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Lubricants (AREA)
PH31451A 1983-11-18 1984-11-16 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines PH22338A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55315783A 1983-11-18 1983-11-18
US55315883A 1983-11-18 1983-11-18

Publications (1)

Publication Number Publication Date
PH22338A true PH22338A (en) 1988-08-12

Family

ID=27070262

Family Applications (1)

Application Number Title Priority Date Filing Date
PH31451A PH22338A (en) 1983-11-18 1984-11-16 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines

Country Status (15)

Country Link
EP (2) EP0310950B1 (cs)
JP (1) JPS60123488A (cs)
KR (1) KR900005657B1 (cs)
AT (2) ATE84525T1 (cs)
AU (2) AU581190B2 (cs)
CA (1) CA1271477A (cs)
DE (3) DE3486043T2 (cs)
DK (6) DK164280C (cs)
ES (1) ES537677A0 (cs)
IE (1) IE57874B1 (cs)
IL (2) IL84537A (cs)
NL (2) NL980041I2 (cs)
NO (7) NO163819C (cs)
NZ (1) NZ210228A (cs)
PH (1) PH22338A (cs)

Families Citing this family (74)

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CA1335996C (en) * 1988-02-16 1995-06-20 Susumu Takada 2-substituted carbonylimidazo¬4,5-c|quinolines
EP0361489A3 (en) * 1988-09-30 1991-06-12 Chugai Seiyaku Kabushiki Kaisha Novel 3,4-diaminoquinoline and pyridine compounds
EP0385630B1 (en) * 1989-02-27 1996-11-27 Riker Laboratories, Inc. 1H-imidazo(4,5-c)Quinolin-4-amines as antivirals
CA2011504C (en) * 1989-03-07 1998-06-02 Kenji Ohmori Imidazoquinolone derivatives
US4929624A (en) * 1989-03-23 1990-05-29 Minnesota Mining And Manufacturing Company Olefinic 1H-imidazo(4,5-c)quinolin-4-amines
CA2021338C (en) * 1989-07-18 1996-07-16 Fumio Suzuki Imidazoquinolone derivatives
US4988815A (en) * 1989-10-26 1991-01-29 Riker Laboratories, Inc. 3-Amino or 3-nitro quinoline compounds which are intermediates in preparing 1H-imidazo[4,5-c]quinolines
FR2654021B1 (fr) * 1989-11-07 1992-02-28 Simond Jacques Procede de vitrification de cendres volantes et dispositif pour sa mise en óoeuvre.
GB8928281D0 (en) * 1989-12-14 1990-02-21 Smith Kline French Lab Compounds
EP0459505B1 (en) * 1990-06-01 1996-10-02 Kyowa Hakko Kogyo Co., Ltd. Imidazonaphthyridine derivatives
DK0582581T3 (da) * 1991-03-01 1999-11-08 Minnesota Mining & Mfg 1,2-substituerede 1H-imidazo[4,5-c]quinolin-4-aminer
US5266575A (en) * 1991-11-06 1993-11-30 Minnesota Mining And Manufacturing Company 2-ethyl 1H-imidazo[4,5-ciquinolin-4-amines
IL105325A (en) * 1992-04-16 1996-11-14 Minnesota Mining & Mfg Immunogen/vaccine adjuvant composition
US5395937A (en) * 1993-01-29 1995-03-07 Minnesota Mining And Manufacturing Company Process for preparing quinoline amines
US5693811A (en) * 1996-06-21 1997-12-02 Minnesota Mining And Manufacturing Company Process for preparing tetrahdroimidazoquinolinamines
WO1998030562A1 (en) * 1997-01-09 1998-07-16 Terumo Kabushiki Kaisha Novel amide derivatives and intermediates for the synthesis thereof
JPH10298181A (ja) * 1997-04-25 1998-11-10 Sumitomo Pharmaceut Co Ltd タイプ２ヘルパーｔ細胞選択的免疫応答抑制剤
JP2000119271A (ja) 1998-08-12 2000-04-25 Hokuriku Seiyaku Co Ltd １ｈ―イミダゾピリジン誘導体
UA75622C2 (en) * 2000-12-08 2006-05-15 3M Innovative Properties Co Aryl ether substituted imidazoquinolines, pharmaceutical composition based thereon
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JP2006502121A (ja) 2002-07-23 2006-01-19 テバ ジョジセルジャール レースベニュタールシャシャーグ １Ｈ−イミダゾ［４，５−ｃ］キノリン−４−フタルイミド中間体を介する１Ｈ−イミダゾ−［４，５−ｃ］キノリン−４−アミンの調製
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BRPI0413558A (pt) 2003-08-12 2006-10-17 3M Innovative Properties Co compostos contendo imidazo substituìdo por hidroxilamina
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KR101154101B1 (ko) 2003-10-03 2012-06-11 쓰리엠 이노베이티브 프로퍼티즈 컴파니 알콕시 치환된 이미다조퀴놀린
US7544697B2 (en) 2003-10-03 2009-06-09 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and analogs thereof
ITMI20032121A1 (it) * 2003-11-04 2005-05-05 Dinamite Dipharma Spa In Forma Abbr Eviata Dipharm Procedimento per la preparazione di imiquimod e suoi intermedi
AU2004291101A1 (en) 2003-11-14 2005-06-02 3M Innovative Properties Company Oxime substituted imidazo ring compounds
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US7968563B2 (en) 2005-02-11 2011-06-28 3M Innovative Properties Company Oxime and hydroxylamine substituted imidazo[4,5-c] ring compounds and methods
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US20090324551A1 (en) 2005-08-22 2009-12-31 The Regents Of The University Of California Office Of Technology Transfer Tlr agonists
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ES2456964T3 (es) 2007-02-07 2014-04-24 The Regents Of The University Of California Conjugados de agonistas de TLR sintéticos y usos de los mismos
EP2009002A1 (en) * 2007-06-21 2008-12-31 Institut National De La Sante Et De La Recherche Medicale (Inserm) New process for the manufacture of 1H-imidazo [4,5-c]-quinoline ring systems
WO2010088924A1 (en) 2009-02-06 2010-08-12 Telormedix Sa Pharmaceutical compositions comprising imidazoquinolin(amines) and derivatives thereof suitable for local administration
KR20110117705A (ko) 2009-02-11 2011-10-27 더 리전트 오브 더 유니버시티 오브 캘리포니아 톨-유사 수용체 조정제 및 질병의 치료
BR112013003772A2 (pt) * 2010-08-17 2016-08-02 3M Innovative Properties Co composições de compostos modificadores de resposta imunológica lipidadas, formulações e métodos
US8728486B2 (en) 2011-05-18 2014-05-20 University Of Kansas Toll-like receptor-7 and -8 modulatory 1H imidazoquinoline derived compounds
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US3700674A (en) * 1969-04-30 1972-10-24 American Cyanamid Co 4-alkylamino-3-nitroquinolines
IL68495A0 (en) * 1982-05-03 1983-07-31 Lilly Co Eli 2-phenylimidazo(4,5-c)pyridines

Also Published As

Publication number Publication date
DK135791A (da) 1991-07-16
DE3486043T2 (de) 1993-06-03
DE3486043D1 (de) 1993-02-25
AU2991189A (en) 1989-06-15
CA1271477A (en) 1990-07-10
NZ210228A (en) 1989-01-27
DK165921C (da) 1993-06-28
DK136191D0 (da) 1991-07-16
DK164455C (da) 1992-11-16
DK164455B (da) 1992-06-29
NO168705B (no) 1991-12-16
AU581190B2 (en) 1989-02-16
DK136091D0 (da) 1991-07-16
NO890824D0 (no) 1989-02-27
NO890825D0 (no) 1989-02-27
IE57874B1 (en) 1993-05-05
IL84537A0 (en) 1988-04-29
NO890826D0 (no) 1989-02-27
NO165147B (no) 1990-09-24
JPH0586391B2 (cs) 1993-12-10
DK135791D0 (da) 1991-07-16
NO890823D0 (no) 1989-02-27
DK135991D0 (da) 1991-07-16
ATE84525T1 (de) 1993-01-15
IE842952L (en) 1985-05-18
DK135891A (da) 1991-07-16
DK165921B (da) 1993-02-08
DK542684A (da) 1985-05-19
DK164280B (da) 1992-06-01
NO165146B (no) 1990-09-24
IL84537A (en) 1990-12-23
AU611997B2 (en) 1991-06-27
DK542684D0 (da) 1984-11-15
DK164280C (da) 1992-11-30
NO1999015I1 (no) 1999-07-08
NO890825L (no) 1985-05-20
DK135891D0 (da) 1991-07-16
DK136091A (da) 1991-07-16
AU3540284A (en) 1985-05-23
NO890826L (no) 1985-05-20
NL980041I1 (nl) 1999-02-01
NO890822L (no) 1985-05-20
EP0310950B1 (en) 1993-01-13
DK164451C (da) 1992-11-09
NO169437B (no) 1992-03-16
JPS60123488A (ja) 1985-07-02
NO890823L (no) 1985-05-20
DK136191A (da) 1991-07-16
DK169179B1 (da) 1994-09-05
NO165147C (no) 1991-01-02
EP0145340A2 (en) 1985-06-19
NO165145B (no) 1990-09-24
DK164452C (da) 1992-11-09
EP0310950A1 (en) 1989-04-12
NO163819C (no) 1990-08-01
NL980041I2 (nl) 1999-07-01
DE3481124D1 (de) 1990-03-01
NL980043I1 (nl) 1999-02-01
NO890824L (no) 1985-05-20
DE19975027I2 (de) 2000-09-21
NO168705C (no) 1992-03-25
EP0145340A3 (en) 1986-06-11
ES8603477A1 (es) 1985-12-16
KR900005657B1 (ko) 1990-08-03
KR850003890A (ko) 1985-06-29
NO844565L (no) 1985-05-20
DK135991A (da) 1991-07-16
DK164452B (da) 1992-06-29
NO163819B (no) 1990-04-17
NO165145C (no) 1991-01-02
ATE49763T1 (de) 1990-02-15
NO890822D0 (no) 1989-02-27
EP0145340B1 (en) 1990-01-24
NO169437C (no) 1992-06-24
DK164451B (da) 1992-06-29
NO165146C (no) 1991-01-02
ES537677A0 (es) 1985-12-16

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PH22338A (en) 1h-imidazo(4,5-c)quinolines and 1h-imidazo(4,5-c) quinolin-4-amines