DK164455C - 1h-imidazooe4,5-caaquinolin-4-chlorforbindelser - Google Patents

1h-imidazooe4,5-caaquinolin-4-chlorforbindelser

Info

Publication number
DK164455C
DK164455C DK135891A DK135891A DK164455C DK 164455 C DK164455 C DK 164455C DK 135891 A DK135891 A DK 135891A DK 135891 A DK135891 A DK 135891A DK 164455 C DK164455 C DK 164455C
Authority
DK
Denmark
Prior art keywords
carbon atoms
compounds
group
imidazooe4
caaquinolin
Prior art date
Application number
DK135891A
Other languages
English (en)
Other versions
DK135891D0 (da
DK164455B (da
DK135891A (da
Inventor
John F Gerster
Original Assignee
Riker Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Riker Laboratories Inc filed Critical Riker Laboratories Inc
Publication of DK135891D0 publication Critical patent/DK135891D0/da
Publication of DK135891A publication Critical patent/DK135891A/da
Publication of DK164455B publication Critical patent/DK164455B/da
Application granted granted Critical
Publication of DK164455C publication Critical patent/DK164455C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/42Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Physical Water Treatments (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Macromonomer-Based Addition Polymer (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Alarm Systems (AREA)
  • Quinoline Compounds (AREA)
  • Luminescent Compositions (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Lubricants (AREA)
DK135891A 1983-11-18 1991-07-16 1h-imidazooe4,5-caaquinolin-4-chlorforbindelser DK164455C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US55315783A 1983-11-18 1983-11-18
US55315883A 1983-11-18 1983-11-18
US55315783 1983-11-18
US55315883 1983-11-18

Publications (4)

Publication Number Publication Date
DK135891D0 DK135891D0 (da) 1991-07-16
DK135891A DK135891A (da) 1991-07-16
DK164455B DK164455B (da) 1992-06-29
DK164455C true DK164455C (da) 1992-11-16

Family

ID=27070262

Family Applications (6)

Application Number Title Priority Date Filing Date
DK542684A DK164280C (da) 1983-11-18 1984-11-15 1h-imidazooe4,5-caaquinolin eller derivat deraf og farmaceutisk praeparat indeholdende en saadan forbindelse
DK135991A DK165921C (da) 1983-11-18 1991-07-16 1h-imidazooe4,5-caaquinolin-5-oxyforbindelser
DK135791A DK169179B1 (da) 1983-11-18 1991-07-16 1H-imidazo[4,5-c]quinolin-4-amin, farmaceutisk præparat indeholdende en sådan forbindelse og fremga ngsmåde til fremstilling af en sådan forbindelse
DK136091A DK164451C (da) 1983-11-18 1991-07-16 3-aminoquinolinderivat
DK136191A DK164452C (da) 1983-11-18 1991-07-16 3-nitroquinolinderivat
DK135891A DK164455C (da) 1983-11-18 1991-07-16 1h-imidazooe4,5-caaquinolin-4-chlorforbindelser

Family Applications Before (5)

Application Number Title Priority Date Filing Date
DK542684A DK164280C (da) 1983-11-18 1984-11-15 1h-imidazooe4,5-caaquinolin eller derivat deraf og farmaceutisk praeparat indeholdende en saadan forbindelse
DK135991A DK165921C (da) 1983-11-18 1991-07-16 1h-imidazooe4,5-caaquinolin-5-oxyforbindelser
DK135791A DK169179B1 (da) 1983-11-18 1991-07-16 1H-imidazo[4,5-c]quinolin-4-amin, farmaceutisk præparat indeholdende en sådan forbindelse og fremga ngsmåde til fremstilling af en sådan forbindelse
DK136091A DK164451C (da) 1983-11-18 1991-07-16 3-aminoquinolinderivat
DK136191A DK164452C (da) 1983-11-18 1991-07-16 3-nitroquinolinderivat

Country Status (15)

Country Link
EP (2) EP0310950B1 (da)
JP (1) JPS60123488A (da)
KR (1) KR900005657B1 (da)
AT (2) ATE84525T1 (da)
AU (2) AU581190B2 (da)
CA (1) CA1271477A (da)
DE (3) DE19975027I2 (da)
DK (6) DK164280C (da)
ES (1) ES8603477A1 (da)
IE (1) IE57874B1 (da)
IL (2) IL84537A (da)
NL (2) NL980043I1 (da)
NO (7) NO163819C (da)
NZ (1) NZ210228A (da)
PH (1) PH22338A (da)

Families Citing this family (72)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1306260C (en) * 1985-10-18 1992-08-11 Shionogi & Co., Ltd. Condensed imidazopyridine derivatives
US4942168A (en) * 1987-07-13 1990-07-17 Hoechst-Roussel Pharmaceuticals Inc. Hydroxyquinoline amines, and method of enhancing memory in mammals
CA1335996C (en) * 1988-02-16 1995-06-20 Susumu Takada 2-substituted carbonylimidazo¬4,5-c|quinolines
EP0361489A3 (en) * 1988-09-30 1991-06-12 Chugai Seiyaku Kabushiki Kaisha Novel 3,4-diaminoquinoline and pyridine compounds
ES2094141T3 (es) * 1989-02-27 1997-01-16 Riker Laboratories Inc 1h-imidazo(4,5-c)quinolin-4-aminas como antivirales.
US4994468A (en) * 1989-03-07 1991-02-19 Kyowa Hakko Kogyo Co., Ltd. Imidazoquinolone derivatives
US4929624A (en) * 1989-03-23 1990-05-29 Minnesota Mining And Manufacturing Company Olefinic 1H-imidazo(4,5-c)quinolin-4-amines
CA2021338C (en) * 1989-07-18 1996-07-16 Fumio Suzuki Imidazoquinolone derivatives
US4988815A (en) * 1989-10-26 1991-01-29 Riker Laboratories, Inc. 3-Amino or 3-nitro quinoline compounds which are intermediates in preparing 1H-imidazo[4,5-c]quinolines
FR2654021B1 (fr) * 1989-11-07 1992-02-28 Simond Jacques Procede de vitrification de cendres volantes et dispositif pour sa mise en óoeuvre.
GB8928281D0 (en) * 1989-12-14 1990-02-21 Smith Kline French Lab Compounds
EP0459505B1 (en) * 1990-06-01 1996-10-02 Kyowa Hakko Kogyo Co., Ltd. Imidazonaphthyridine derivatives
HU222251B1 (hu) * 1991-03-01 2003-05-28 Minnesota Mining And Manufacturing Company 1-és 2-helyzetben szubsztituált 1H-imidazo[4,5-c]kinolin-4-amin-származékok előállításában alkalmazható 1- és 2-helyzetben szubsztituált 1H-imidazo[4,5-c]kinolin-4-(szubsztituált)-származékok
US5266575A (en) * 1991-11-06 1993-11-30 Minnesota Mining And Manufacturing Company 2-ethyl 1H-imidazo[4,5-ciquinolin-4-amines
IL105325A (en) * 1992-04-16 1996-11-14 Minnesota Mining & Mfg Immunogen/vaccine adjuvant composition
US5395937A (en) * 1993-01-29 1995-03-07 Minnesota Mining And Manufacturing Company Process for preparing quinoline amines
US5693811A (en) * 1996-06-21 1997-12-02 Minnesota Mining And Manufacturing Company Process for preparing tetrahdroimidazoquinolinamines
JP4101302B2 (ja) * 1997-01-09 2008-06-18 テルモ株式会社 新規アミド誘導体および合成中間体
JPH10298181A (ja) * 1997-04-25 1998-11-10 Sumitomo Pharmaceut Co Ltd タイプ2ヘルパーt細胞選択的免疫応答抑制剤
JP2000119271A (ja) 1998-08-12 2000-04-25 Hokuriku Seiyaku Co Ltd 1h―イミダゾピリジン誘導体
JP4602667B2 (ja) * 2001-10-23 2010-12-22 メルク セローノ ソシエテ アノニム アゾール誘導体および該アゾール誘導体を含有する医薬組成物
GB0211649D0 (en) 2002-05-21 2002-07-03 Novartis Ag Organic compounds
EP1543002B1 (en) 2002-07-23 2006-08-30 TEVA Gyógyszergyár Zártkörüen Müködö Részvénytársaság Preparation of 1h-imidazo 4,5-c|quinolin-4-amines via1h-imidazo 4,5-c|quinolin-4-phthalimide intermediates
KR20050030958A (ko) 2002-07-26 2005-03-31 비오갈 기오기스제르갸르 알티. 신규한 1H-이미다조[4,5-c]퀴놀린-4-시아노 및1H-이미다조[4,5-c]퀴놀린-4-카르복스아미드 중간체를통한 1H-이미다조[4,5-c]퀴놀린-4-아민의 제조 방법
MXPA06001674A (es) 2003-08-12 2006-05-12 3M Innovative Properties Co Compuestos que contienen imidazo hidroxilamina-sustituidos.
JP5128815B2 (ja) * 2003-08-27 2013-01-23 スリーエム イノベイティブ プロパティズ カンパニー アリールオキシ置換およびアリールアルキレンオキシ置換イミダゾキノリン
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US7544697B2 (en) 2003-10-03 2009-06-09 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and analogs thereof
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US3700674A (en) * 1969-04-30 1972-10-24 American Cyanamid Co 4-alkylamino-3-nitroquinolines
RO86850B (ro) * 1982-05-03 1985-05-31 Eli Lilly And Company Procedeu pentru prepararea unor 2-fenilimidazo [4,5 c] piridine

Also Published As

Publication number Publication date
NO890825L (no) 1985-05-20
DK135991A (da) 1991-07-16
NO169437B (no) 1992-03-16
DK542684D0 (da) 1984-11-15
NO1999015I1 (no) 1999-07-08
EP0310950B1 (en) 1993-01-13
IE842952L (en) 1985-05-18
EP0145340A2 (en) 1985-06-19
JPS60123488A (ja) 1985-07-02
NO165145C (no) 1991-01-02
DK164452C (da) 1992-11-09
NO169437C (no) 1992-06-24
ATE84525T1 (de) 1993-01-15
ATE49763T1 (de) 1990-02-15
NO168705B (no) 1991-12-16
NO163819C (no) 1990-08-01
NO890824L (no) 1985-05-20
NO165146C (no) 1991-01-02
NO890826D0 (no) 1989-02-27
NO163819B (no) 1990-04-17
NZ210228A (en) 1989-01-27
DE3486043T2 (de) 1993-06-03
KR850003890A (ko) 1985-06-29
DK135891D0 (da) 1991-07-16
KR900005657B1 (ko) 1990-08-03
DK164455B (da) 1992-06-29
DE3486043D1 (de) 1993-02-25
IL84537A0 (en) 1988-04-29
DK542684A (da) 1985-05-19
EP0145340A3 (en) 1986-06-11
NO168705C (no) 1992-03-25
NO844565L (no) 1985-05-20
DK164451C (da) 1992-11-09
NO165147B (no) 1990-09-24
DK165921C (da) 1993-06-28
IL84537A (en) 1990-12-23
NO890823L (no) 1985-05-20
NO165145B (no) 1990-09-24
NO890826L (no) 1985-05-20
IE57874B1 (en) 1993-05-05
DK136191A (da) 1991-07-16
DK136091A (da) 1991-07-16
DK164280B (da) 1992-06-01
DK164452B (da) 1992-06-29
NL980041I2 (nl) 1999-07-01
DK135991D0 (da) 1991-07-16
NO890824D0 (no) 1989-02-27
AU581190B2 (en) 1989-02-16
CA1271477A (en) 1990-07-10
EP0145340B1 (en) 1990-01-24
DE19975027I2 (de) 2000-09-21
DK135791D0 (da) 1991-07-16
DK164280C (da) 1992-11-30
EP0310950A1 (en) 1989-04-12
ES537677A0 (es) 1985-12-16
JPH0586391B2 (da) 1993-12-10
AU3540284A (en) 1985-05-23
DK136091D0 (da) 1991-07-16
PH22338A (en) 1988-08-12
DK135791A (da) 1991-07-16
NO890825D0 (no) 1989-02-27
DK164451B (da) 1992-06-29
DK169179B1 (da) 1994-09-05
NO890822L (no) 1985-05-20
AU611997B2 (en) 1991-06-27
NO890823D0 (no) 1989-02-27
NO165147C (no) 1991-01-02
DK165921B (da) 1993-02-08
NO165146B (no) 1990-09-24
DK135891A (da) 1991-07-16
NL980041I1 (nl) 1999-02-01
NO890822D0 (no) 1989-02-27
DE3481124D1 (de) 1990-03-01
NL980043I1 (nl) 1999-02-01
DK136191D0 (da) 1991-07-16
AU2991189A (en) 1989-06-15
ES8603477A1 (es) 1985-12-16

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