PH21916A - Carboxyalkyl dipeptides and pharmaceutical compositions containing them - Google Patents

Carboxyalkyl dipeptides and pharmaceutical compositions containing them

Info

Publication number
PH21916A
PH21916A PH26366A PH26366A PH21916A PH 21916 A PH21916 A PH 21916A PH 26366 A PH26366 A PH 26366A PH 26366 A PH26366 A PH 26366A PH 21916 A PH21916 A PH 21916A
Authority
PH
Philippines
Prior art keywords
lower alkyl
chem
bridge
hydrogen
alkoxy
Prior art date
Application number
PH26366A
Other languages
English (en)
Inventor
Bernard R Neustadt
Elijah H Gold
Elizabeth M Smith
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26895254&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PH21916(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of PH21916A publication Critical patent/PH21916A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Apparatus For Disinfection Or Sterilisation (AREA)
  • Pyrrole Compounds (AREA)
PH26366A 1980-10-23 1981-10-20 Carboxyalkyl dipeptides and pharmaceutical compositions containing them PH21916A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US19988680A 1980-10-23 1980-10-23
US25848481A 1981-04-28 1981-04-28

Publications (1)

Publication Number Publication Date
PH21916A true PH21916A (en) 1988-04-08

Family

ID=26895254

Family Applications (1)

Application Number Title Priority Date Filing Date
PH26366A PH21916A (en) 1980-10-23 1981-10-20 Carboxyalkyl dipeptides and pharmaceutical compositions containing them

Country Status (28)

Country Link
US (2) US4818749A (de)
EP (1) EP0050800B2 (de)
JP (1) JPH01163197A (de)
KR (1) KR880001843B1 (de)
AT (1) ATE20469T1 (de)
AU (1) AU554362B2 (de)
CA (1) CA1341206C (de)
CY (1) CY1469A (de)
DE (2) DE19575012I2 (de)
DK (1) DK161523C (de)
ES (1) ES8308838A1 (de)
FI (1) FI83222C (de)
GR (1) GR75059B (de)
HK (1) HK36189A (de)
HU (1) HU193146B (de)
IE (1) IE53802B1 (de)
IL (1) IL64085A (de)
KE (1) KE3845A (de)
LU (1) LU88621I2 (de)
MA (1) MA19309A1 (de)
MY (1) MY8700683A (de)
NL (1) NL940001I2 (de)
NO (2) NO164983C (de)
NZ (1) NZ198702A (de)
OA (1) OA06929A (de)
PH (1) PH21916A (de)
PT (1) PT73861B (de)
SG (1) SG78188G (de)

Families Citing this family (144)

* Cited by examiner, † Cited by third party
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DK462581A (da) 1982-04-24
AU7661481A (en) 1982-04-29
ES506414A0 (es) 1983-10-01
DE19575012I2 (de) 2002-01-24
NZ198702A (en) 1985-08-30
IE812475L (en) 1982-04-23
EP0050800B2 (de) 1995-06-07
FI83222B (fi) 1991-02-28
HK36189A (en) 1989-05-12
NO164983C (no) 1990-12-05
JPH01163197A (ja) 1989-06-27
CY1469A (en) 1989-07-21
IE53802B1 (en) 1989-03-01
PT73861B (en) 1985-11-12
GR75059B (de) 1984-07-13
MA19309A1 (fr) 1982-07-01
NO813546L (no) 1982-04-26
AU554362B2 (en) 1986-08-21
DK161523B (da) 1991-07-15
CA1341206C (en) 2001-03-20
NL940001I1 (nl) 1994-03-01
US4831157A (en) 1989-05-16
SG78188G (en) 1989-03-23
EP0050800B1 (de) 1986-06-18
KR830007519A (ko) 1983-10-21
NO164983B (no) 1990-08-27
IL64085A (en) 1986-12-31
FI813283L (fi) 1982-04-24
DE3174844D1 (en) 1986-07-24
HU193146B (en) 1987-08-28
FI83222C (sv) 1991-06-10
MY8700683A (en) 1987-12-31
KE3845A (en) 1989-04-07
US4818749A (en) 1989-04-04
ES8308838A1 (es) 1983-10-01
LU88621I2 (fr) 1995-09-01
PT73861A (en) 1981-11-01
NL940001I2 (nl) 1998-03-02
DK161523C (da) 1991-12-23
NO1995008I1 (no) 1995-09-22
ATE20469T1 (de) 1986-07-15
KR880001843B1 (ko) 1988-09-21
EP0050800A1 (de) 1982-05-05
OA06929A (fr) 1983-05-31

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