PE20220580A1 - Carboxamidas de tiofeno sustituidas y derivados de estas - Google Patents

Carboxamidas de tiofeno sustituidas y derivados de estas

Info

Publication number
PE20220580A1
PE20220580A1 PE2021002260A PE2021002260A PE20220580A1 PE 20220580 A1 PE20220580 A1 PE 20220580A1 PE 2021002260 A PE2021002260 A PE 2021002260A PE 2021002260 A PE2021002260 A PE 2021002260A PE 20220580 A1 PE20220580 A1 PE 20220580A1
Authority
PE
Peru
Prior art keywords
substituted thiophene
derivatives
atoms
group
thiophene carboxamides
Prior art date
Application number
PE2021002260A
Other languages
English (en)
Inventor
Jeremy Dufour
Lionel Nicolas
Tomoki Tsuchiya
David Bernier
Thomas Knobloch
Stephane Brunet
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of PE20220580A1 publication Critical patent/PE20220580A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/06—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings
    • A01N43/10—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings with sulfur as the ring hetero atom
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N53/00—Biocides, pest repellants or attractants, or plant growth regulators containing cyclopropane carboxylic acids or derivatives thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P1/00—Disinfectants; Antimicrobial compounds or mixtures thereof

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invencion se refiere a compuestos derivados de carboxamida de tiofeno sustituidos de formula (I); en donde R1 son atomos de Br o Cl; R2 se selecciona del grupo que consiste en Br, Cl, I y F; R3 se selecciona del grupo que consiste en H, alquilo C1-C6, haloalquilo C1-C6, cianoalquilo C1-C6, alquenilo C2-C6, entre otros; siempre que R2 no sea un atomo de Cl cuando R1 son atomos de Cl. Un compuesto seleccionado es 1-{[(3-bromo-4,5-dicloro-2- tienil)carbonil]amino}ciclopropanocarboxilato de etilo. Tambien refiere una composicion que los comprende y un metodo de preparacion de los mismos siendo utiles para controlar microorganismos fitopatogenos.
PE2021002260A 2019-07-03 2020-06-30 Carboxamidas de tiofeno sustituidas y derivados de estas PE20220580A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP19184093 2019-07-03
PCT/EP2020/068324 WO2021001331A1 (en) 2019-07-03 2020-06-30 Substituted thiophene carboxamides and derivatives thereof as microbicides

Publications (1)

Publication Number Publication Date
PE20220580A1 true PE20220580A1 (es) 2022-04-20

Family

ID=67145689

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2021002260A PE20220580A1 (es) 2019-07-03 2020-06-30 Carboxamidas de tiofeno sustituidas y derivados de estas

Country Status (18)

Country Link
US (1) US20220274945A1 (es)
EP (1) EP3994130A1 (es)
JP (1) JP2022538262A (es)
KR (1) KR20220029697A (es)
CN (1) CN114364663A (es)
AR (1) AR119344A1 (es)
AU (1) AU2020298744A1 (es)
BR (1) BR112021026696A2 (es)
CA (1) CA3145592A1 (es)
CL (1) CL2021003501A1 (es)
CO (1) CO2021017743A2 (es)
CR (1) CR20210678A (es)
EC (1) ECSP21093925A (es)
MA (1) MA56441A (es)
MX (1) MX2022000122A (es)
PE (1) PE20220580A1 (es)
TW (1) TW202116747A (es)
WO (1) WO2021001331A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2019297401B2 (en) * 2018-07-05 2024-04-18 Bayer Aktiengesellschaft Substituted thiophenecarboxamides and analogues as antibacterials agents

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Also Published As

Publication number Publication date
AR119344A1 (es) 2021-12-09
CR20210678A (es) 2022-02-15
CO2021017743A2 (es) 2022-01-17
MX2022000122A (es) 2022-02-16
MA56441A (fr) 2022-05-11
AU2020298744A1 (en) 2022-01-27
KR20220029697A (ko) 2022-03-08
BR112021026696A2 (pt) 2022-02-15
EP3994130A1 (en) 2022-05-11
TW202116747A (zh) 2021-05-01
CA3145592A1 (en) 2021-01-07
WO2021001331A1 (en) 2021-01-07
CL2021003501A1 (es) 2022-08-12
CN114364663A (zh) 2022-04-15
JP2022538262A (ja) 2022-09-01
US20220274945A1 (en) 2022-09-01
ECSP21093925A (es) 2022-01-31

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