PE20130603A1 - Composicion farmaceutica que contiene un inhibidor de esteroide c17,20 liasa - Google Patents

Composicion farmaceutica que contiene un inhibidor de esteroide c17,20 liasa

Info

Publication number
PE20130603A1
PE20130603A1 PE2013000161A PE2013000161A PE20130603A1 PE 20130603 A1 PE20130603 A1 PE 20130603A1 PE 2013000161 A PE2013000161 A PE 2013000161A PE 2013000161 A PE2013000161 A PE 2013000161A PE 20130603 A1 PE20130603 A1 PE 20130603A1
Authority
PE
Peru
Prior art keywords
liasa
pharmaceutical composition
composition containing
steroid inhibitor
steroid
Prior art date
Application number
PE2013000161A
Other languages
English (en)
Inventor
Masuo Yamaoka
Takahito Hara
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40591618&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20130603(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of PE20130603A1 publication Critical patent/PE20130603A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41881,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA QUE COMPRENDE: A) UN INHIBIDOR DE ESTEROIDE C17,20 LIASA TAL COMO (+)-6-(7-HIDROXI-6,7-DIHIDRO-5H-PIRROLO[1,2-c]IMIDAZOL-7-IL)-N-METIL-2-NAFTAMIDA; Y B) UN AGONISTA DEL RECEPTOR DE GnRH, UN ANTAGONISTA DEL RECEPTOR DE GnRH O UN FARMACO DE ADRENOCORTICOHORMONA TAL COMO ACETATO DE LEUPRORELINA O PREDNISOLONA. DICHA COMPOSICION ES UTIL EN EL TRATAMIENTO DE CANCER DE PROSTATA INDEPENDIENTE DE ANDROGENOS
PE2013000161A 2007-10-29 2008-10-28 Composicion farmaceutica que contiene un inhibidor de esteroide c17,20 liasa PE20130603A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2007280813 2007-10-29

Publications (1)

Publication Number Publication Date
PE20130603A1 true PE20130603A1 (es) 2013-05-30

Family

ID=40591618

Family Applications (2)

Application Number Title Priority Date Filing Date
PE2008001841A PE20090931A1 (es) 2007-10-29 2008-10-28 Composicion farmaceutica que contiene un inhibidor de esteroide c17,20 liasa
PE2013000161A PE20130603A1 (es) 2007-10-29 2008-10-28 Composicion farmaceutica que contiene un inhibidor de esteroide c17,20 liasa

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PE2008001841A PE20090931A1 (es) 2007-10-29 2008-10-28 Composicion farmaceutica que contiene un inhibidor de esteroide c17,20 liasa

Country Status (17)

Country Link
US (2) US20100261689A1 (es)
EP (1) EP2205239A2 (es)
JP (1) JP5430576B2 (es)
KR (1) KR20100088144A (es)
CN (1) CN101909622B (es)
AR (1) AR069079A1 (es)
AU (1) AU2008319767B8 (es)
CA (1) CA2703780A1 (es)
CL (1) CL2008003198A1 (es)
IL (1) IL205368A (es)
MX (1) MX2010004405A (es)
NZ (1) NZ585473A (es)
PE (2) PE20090931A1 (es)
RU (1) RU2481107C2 (es)
SG (1) SG185930A1 (es)
TW (1) TWI426901B (es)
WO (1) WO2009057795A2 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY33740A (es) * 2010-11-18 2012-05-31 Takeda Pharmaceutical Método para tratar el cáncer de mama y cáncer de ovarios
EP2709614A4 (en) * 2011-05-17 2015-04-15 Takeda Pharmaceutical PHARMACEUTICAL COMPOSITION AND METHOD FOR THE TREATMENT OF CANCER
US10201549B2 (en) 2013-06-14 2019-02-12 Professional Compounding Centers Of America (Pcca) Testosterone combined with anastrozole injection solutions

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2000505444A (ja) * 1996-02-14 2000-05-09 ヘキスト・マリオン・ルセル・インコーポレイテツド テストステロン5α―レダクターゼおよびC▲下17―20▼リアーゼの活性阻害剤としての17β―シクロプロピル(アミノ/オキシ)4―アザステロイド
PE20010781A1 (es) * 1999-10-22 2001-08-08 Takeda Chemical Industries Ltd Compuestos 1-(1h-imidazol-4-il)-1-(naftil-2-sustituido)etanol, su produccion y utilizacion
MY134929A (en) * 2000-11-17 2008-01-31 Takeda Pharmaceutical Novel imidazole derivatives, production method thereof and use thereof
US7662974B2 (en) * 2002-01-10 2010-02-16 Takeda Pharmaceutical Company Limited Process for producing fused imidazole compound, reformatsky reagent in stable form, and process for producing the same
EP1615944A4 (en) * 2003-04-01 2010-08-11 Harbor Biosciences Inc ANTI-ORANGE PROBLEMS WITH MARGINAL AGONIST EFFECT AND METHOD OF USE
WO2004087190A1 (en) * 2003-04-02 2004-10-14 Genix Therapeutics Inc. Method for the treatment of prostate cancer
GB0312407D0 (en) * 2003-05-29 2003-07-02 Pharma Mar Sau Treatment
CA2610343A1 (en) * 2005-03-03 2006-09-08 Takeda Pharmaceutical Company Limited Release-control composition
EP1861109A2 (en) * 2005-03-09 2007-12-05 Cardax Pharmaceuticals, Inc. Carotenoids, carotenoid analogs, or carotenoid derivatives for the treatment of proliferative disorders
PE20070207A1 (es) * 2005-07-22 2007-03-09 Genentech Inc Tratamiento combinado de los tumores que expresan el her
US20100009949A1 (en) * 2006-03-24 2010-01-14 Bioxell S.P.A. Novel method
CN104306977A (zh) * 2006-08-25 2015-01-28 库伽尔生物科技公司 治疗癌症的方法和组合物
WO2009009132A1 (en) * 2007-07-12 2009-01-15 Cougar Biotechnology, Inc. Use of 17alpha-hydroxylase/c17, 20-lyase inhibitors for the treatment of cancer

Also Published As

Publication number Publication date
WO2009057795A8 (en) 2010-05-14
AU2008319767B8 (en) 2014-01-09
AU2008319767A1 (en) 2009-05-07
CA2703780A1 (en) 2009-05-07
CN101909622A (zh) 2010-12-08
SG185930A1 (en) 2012-12-28
KR20100088144A (ko) 2010-08-06
AU2008319767A8 (en) 2014-01-09
AR069079A1 (es) 2009-12-30
EP2205239A2 (en) 2010-07-14
MX2010004405A (es) 2010-05-03
TWI426901B (zh) 2014-02-21
TW200927097A (en) 2009-07-01
NZ585473A (en) 2012-03-30
US20100261689A1 (en) 2010-10-14
AU2008319767A2 (en) 2010-06-17
JP2011502114A (ja) 2011-01-20
RU2481107C2 (ru) 2013-05-10
PE20090931A1 (es) 2009-08-03
JP5430576B2 (ja) 2014-03-05
US20140256693A1 (en) 2014-09-11
IL205368A (en) 2014-08-31
RU2010121765A (ru) 2011-12-10
CL2008003198A1 (es) 2009-12-18
AU2008319767B2 (en) 2013-12-19
IL205368A0 (en) 2010-12-30
WO2009057795A2 (en) 2009-05-07
WO2009057795A3 (en) 2009-07-09
CN101909622B (zh) 2013-06-19

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