PE20120688A1 - Derivados de n1-acil-5-fluoropirimidinona - Google Patents

Derivados de n1-acil-5-fluoropirimidinona

Info

Publication number
PE20120688A1
PE20120688A1 PE2012000169A PE2012000169A PE20120688A1 PE 20120688 A1 PE20120688 A1 PE 20120688A1 PE 2012000169 A PE2012000169 A PE 2012000169A PE 2012000169 A PE2012000169 A PE 2012000169A PE 20120688 A1 PE20120688 A1 PE 20120688A1
Authority
PE
Peru
Prior art keywords
fluoro
alkyl
optionally substituted
fluoropyrimidinone
acil
Prior art date
Application number
PE2012000169A
Other languages
English (en)
Spanish (es)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20120688(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PE20120688A1 publication Critical patent/PE20120688A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PE2012000169A 2009-08-07 2010-08-05 Derivados de n1-acil-5-fluoropirimidinona PE20120688A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
PE20120688A1 true PE20120688A1 (es) 2012-06-06

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2012000169A PE20120688A1 (es) 2009-08-07 2010-08-05 Derivados de n1-acil-5-fluoropirimidinona

Country Status (33)

Country Link
US (1) US8470839B2 (enEXAMPLES)
EP (1) EP2519512B1 (enEXAMPLES)
JP (1) JP5748754B2 (enEXAMPLES)
KR (1) KR101792285B1 (enEXAMPLES)
CN (1) CN102548981B (enEXAMPLES)
AU (1) AU2010279402B2 (enEXAMPLES)
BR (1) BR112012002810B1 (enEXAMPLES)
CA (1) CA2768510C (enEXAMPLES)
CL (1) CL2012000316A1 (enEXAMPLES)
CO (1) CO6491117A2 (enEXAMPLES)
CR (1) CR20120030A (enEXAMPLES)
CY (1) CY1122115T1 (enEXAMPLES)
DK (1) DK2519512T3 (enEXAMPLES)
EA (1) EA023411B1 (enEXAMPLES)
EC (1) ECSP12011653A (enEXAMPLES)
ES (1) ES2728966T3 (enEXAMPLES)
HN (1) HN2012000269A (enEXAMPLES)
HR (1) HRP20190919T1 (enEXAMPLES)
HU (1) HUE045290T2 (enEXAMPLES)
IL (1) IL217952A (enEXAMPLES)
IN (1) IN2012DN00539A (enEXAMPLES)
LT (1) LT2519512T (enEXAMPLES)
MX (1) MX2012001620A (enEXAMPLES)
NI (1) NI201200022A (enEXAMPLES)
NZ (1) NZ597570A (enEXAMPLES)
PE (1) PE20120688A1 (enEXAMPLES)
PL (1) PL2519512T3 (enEXAMPLES)
PT (1) PT2519512T (enEXAMPLES)
SI (1) SI2519512T1 (enEXAMPLES)
TR (1) TR201908180T4 (enEXAMPLES)
UA (1) UA106889C2 (enEXAMPLES)
WO (1) WO2011017538A1 (enEXAMPLES)
ZA (1) ZA201200819B (enEXAMPLES)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101743791B1 (ko) * 2009-08-07 2017-06-05 다우 아그로사이언시즈 엘엘씨 Ｎ1-술포닐-5-플루오로피리미디논 유도체
CN106977462B (zh) 2011-08-17 2020-04-28 阿达玛马克西姆股份有限公司 5-氟-4-亚氨基-3-(取代的)-3,4-二氢嘧啶-2(1h)酮衍生物
PL2938194T3 (pl) 2012-12-28 2020-09-21 Adama Makhteshim Ltd. Pochodne n-podstawionego 5-fluoro-4-imino-3-metylo-2-okso-3,4-dihydropirymidyno-1(2h)-karboksylanu
RU2656101C2 (ru) * 2012-12-28 2018-05-31 Адама Мактешим Лтд. Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она
UA117743C2 (uk) 2012-12-28 2018-09-25 Адама Махтешім Лтд. N-(заміщені)-5-фтор-4-іміно-3-метил-2-оксо-3,4-дигідропіримідин-1(2h)-карбоксамідні похідні
MX381341B (es) 2012-12-31 2025-03-12 Adama Makhteshim Ltd Derivados de 3-alquil-5-fluoro-4-sustituido-imino-3,4-dihidropirimidin-2(1h)-ona como fungicidas.
JP6608366B2 (ja) 2013-12-31 2019-11-20 アダマ・マクテシム・リミテッド 真菌防除のための相乗的殺真菌性混合物および組成物
WO2015103142A1 (en) 2013-12-31 2015-07-09 Dow Agrosciences Llc 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
WO2016048643A1 (en) 2014-09-26 2016-03-31 The Chemours Company Fc, Llc Isocyanate derived organosilanes
JP2020527563A (ja) 2017-07-17 2020-09-10 アダマ・マクテシム・リミテッド ５−フルオロ−４−イミノ−３−メチル−１−トシル−３，４−ジヒドロピリミジン−２−オンの多形体
CA3118729A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof

Family Cites Families (22)

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Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enEXAMPLES) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
DE58908159D1 (de) 1988-03-09 1994-09-15 Ciba Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
DE69618959T2 (de) * 1995-07-05 2002-08-29 E.I. Du Pont De Nemours And Co., Wilmington Pyrimidone und ihre verwendug als fungizide
EA001148B1 (ru) * 1996-03-11 2000-10-30 Новартис Аг Производные пиримидин-4-она
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
EP1731523A4 (en) * 2004-04-01 2009-08-12 Takeda Pharmaceutical THIAZOLOPYRIMIDINDERIVAT
US20080004253A1 (en) * 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
EP2562163A1 (en) * 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
DK2317851T3 (da) 2008-08-01 2014-04-14 Dow Agrosciences Llc Anvendelse af 5-fluorcytosin som fungicid
WO2010085377A2 (en) 2009-01-23 2010-07-29 Crystal Biopharmaceutical Llc Hydroxamic acid derivatives
KR101743791B1 (ko) * 2009-08-07 2017-06-05 다우 아그로사이언시즈 엘엘씨 Ｎ1-술포닐-5-플루오로피리미디논 유도체

Also Published As

Publication number Publication date
KR20120041786A (ko) 2012-05-02
CR20120030A (es) 2012-03-28
AU2010279402B2 (en) 2015-04-16
CN102548981B (zh) 2015-05-13
ZA201200819B (en) 2013-05-29
UA106889C2 (uk) 2014-10-27
BR112012002810B1 (pt) 2018-12-11
CO6491117A2 (es) 2012-07-31
HN2012000269A (es) 2015-04-27
LT2519512T (lt) 2019-07-25
CY1122115T1 (el) 2020-11-25
US8470839B2 (en) 2013-06-25
IL217952A0 (en) 2012-03-29
HK1172894A1 (en) 2013-05-03
MX2012001620A (es) 2012-04-11
EA201270253A1 (ru) 2012-07-30
EA023411B1 (ru) 2016-06-30
EP2519512A4 (en) 2013-01-16
CN102548981A (zh) 2012-07-04
CA2768510A1 (en) 2011-02-10
JP2013501723A (ja) 2013-01-17
CA2768510C (en) 2018-05-15
BR112012002810A2 (pt) 2015-09-15
EP2519512A1 (en) 2012-11-07
EP2519512B1 (en) 2019-03-20
HRP20190919T1 (hr) 2019-09-20
TR201908180T4 (tr) 2019-06-21
NZ597570A (en) 2014-04-30
NI201200022A (es) 2012-05-22
SI2519512T1 (sl) 2019-09-30
IN2012DN00539A (enEXAMPLES) 2015-06-12
JP5748754B2 (ja) 2015-07-15
ES2728966T3 (es) 2019-10-29
AU2010279402A1 (en) 2012-02-02
PT2519512T (pt) 2019-06-04
KR101792285B1 (ko) 2017-10-31
PL2519512T3 (pl) 2019-09-30
DK2519512T3 (da) 2019-05-27
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
IL217952A (en) 2017-11-30
WO2011017538A1 (en) 2011-02-10
US20110034490A1 (en) 2011-02-10
CL2012000316A1 (es) 2014-06-27

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Legal Events

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FG Grant, registration
FD Application declared void or lapsed