AU2010279402B2 - N1-acyl-5-fluoropyrimidinone derivatives - Google Patents

N1-acyl-5-fluoropyrimidinone derivatives Download PDF

Info

Publication number
AU2010279402B2
AU2010279402B2 AU2010279402A AU2010279402A AU2010279402B2 AU 2010279402 B2 AU2010279402 B2 AU 2010279402B2 AU 2010279402 A AU2010279402 A AU 2010279402A AU 2010279402 A AU2010279402 A AU 2010279402A AU 2010279402 B2 AU2010279402 B2 AU 2010279402B2
Authority
AU
Australia
Prior art keywords
optionally substituted
benzyl
phenyl
alkyl
ring system
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2010279402A
Other languages
English (en)
Other versions
AU2010279402A1 (en
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W. Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Adama Makhteshim Ltd
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2010279402(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of AU2010279402A1 publication Critical patent/AU2010279402A1/en
Application granted granted Critical
Publication of AU2010279402B2 publication Critical patent/AU2010279402B2/en
Assigned to ADAMA MAKHTESHIM LTD. reassignment ADAMA MAKHTESHIM LTD. Request for Assignment Assignors: DOW AGROSCIENCES LLC
Ceased legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2010279402A 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives Ceased AU2010279402B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
US61/232,223 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (2)

Publication Number Publication Date
AU2010279402A1 AU2010279402A1 (en) 2012-02-02
AU2010279402B2 true AU2010279402B2 (en) 2015-04-16

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2010279402A Ceased AU2010279402B2 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Country Status (33)

Country Link
US (1) US8470839B2 (enEXAMPLES)
EP (1) EP2519512B1 (enEXAMPLES)
JP (1) JP5748754B2 (enEXAMPLES)
KR (1) KR101792285B1 (enEXAMPLES)
CN (1) CN102548981B (enEXAMPLES)
AU (1) AU2010279402B2 (enEXAMPLES)
BR (1) BR112012002810B1 (enEXAMPLES)
CA (1) CA2768510C (enEXAMPLES)
CL (1) CL2012000316A1 (enEXAMPLES)
CO (1) CO6491117A2 (enEXAMPLES)
CR (1) CR20120030A (enEXAMPLES)
CY (1) CY1122115T1 (enEXAMPLES)
DK (1) DK2519512T3 (enEXAMPLES)
EA (1) EA023411B1 (enEXAMPLES)
EC (1) ECSP12011653A (enEXAMPLES)
ES (1) ES2728966T3 (enEXAMPLES)
HN (1) HN2012000269A (enEXAMPLES)
HR (1) HRP20190919T1 (enEXAMPLES)
HU (1) HUE045290T2 (enEXAMPLES)
IL (1) IL217952A (enEXAMPLES)
IN (1) IN2012DN00539A (enEXAMPLES)
LT (1) LT2519512T (enEXAMPLES)
MX (1) MX2012001620A (enEXAMPLES)
NI (1) NI201200022A (enEXAMPLES)
NZ (1) NZ597570A (enEXAMPLES)
PE (1) PE20120688A1 (enEXAMPLES)
PL (1) PL2519512T3 (enEXAMPLES)
PT (1) PT2519512T (enEXAMPLES)
SI (1) SI2519512T1 (enEXAMPLES)
TR (1) TR201908180T4 (enEXAMPLES)
UA (1) UA106889C2 (enEXAMPLES)
WO (1) WO2011017538A1 (enEXAMPLES)
ZA (1) ZA201200819B (enEXAMPLES)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN2012DN00692A (enEXAMPLES) * 2009-08-07 2015-06-19 Dow Agroscience Llc
UA113062C2 (xx) * 2011-08-17 2016-12-12 Похідні 5-фтор-4-іміно-3-(заміщеного)-3,4-дигідропіримідин-2(1h)ону
HUE047711T2 (hu) 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok
EP2945635A4 (en) * 2012-12-28 2016-05-25 Dow Agrosciences Llc 1- (BENZOYL-SUBSTITUTED) -5-FLUORO-4-IMINO-3-METHYL-3,4-DIHYDROPYRIMIDIN-2 (1H) -ONE DERIVATIVES
KR20150100869A (ko) 2012-12-28 2015-09-02 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복스아미드 유도체
AU2013370494B2 (en) 2012-12-31 2017-08-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
AU2014373850A1 (en) 2013-12-31 2016-08-11 Adama Makhteshim Ltd. Synergistic fungicidal mixtures and compositions for fungal control
MX375727B (es) 2013-12-31 2025-03-06 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparacion.
CN107001397B (zh) 2014-09-26 2020-10-13 科慕埃弗西有限公司 异氰酸酯衍生的有机硅烷
IL309708A (en) 2017-07-17 2024-02-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
US12414559B2 (en) 2018-11-05 2025-09-16 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
WO1997033890A1 (en) * 1996-03-11 1997-09-18 Novartis Ag Pyrimidin-4-one derivatives as pesticide

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enEXAMPLES) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ES2057172T3 (es) 1988-03-09 1994-10-16 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
BR9609613A (pt) 1995-07-05 1999-05-25 Du Pont Composto composição fungicida e método de controle de doenças de plantas
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
US20080269238A1 (en) 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
WO2008005303A2 (en) 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
EP2562161A1 (en) 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
CN102215691B (zh) 2008-08-01 2015-02-04 陶氏益农公司 5-氟胞嘧啶作为杀真菌剂的用途
EP2389375B1 (en) 2009-01-23 2015-05-20 Euro-Celtique S.A. Hydroxamic acid derivatives
IN2012DN00692A (enEXAMPLES) 2009-08-07 2015-06-19 Dow Agroscience Llc

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
WO1997033890A1 (en) * 1996-03-11 1997-09-18 Novartis Ag Pyrimidin-4-one derivatives as pesticide

Also Published As

Publication number Publication date
BR112012002810A2 (pt) 2015-09-15
ES2728966T3 (es) 2019-10-29
PT2519512T (pt) 2019-06-04
WO2011017538A1 (en) 2011-02-10
LT2519512T (lt) 2019-07-25
JP5748754B2 (ja) 2015-07-15
KR101792285B1 (ko) 2017-10-31
HRP20190919T1 (hr) 2019-09-20
UA106889C2 (uk) 2014-10-27
CN102548981A (zh) 2012-07-04
CY1122115T1 (el) 2020-11-25
US20110034490A1 (en) 2011-02-10
CA2768510C (en) 2018-05-15
MX2012001620A (es) 2012-04-11
EP2519512B1 (en) 2019-03-20
US8470839B2 (en) 2013-06-25
EA201270253A1 (ru) 2012-07-30
HN2012000269A (es) 2015-04-27
DK2519512T3 (da) 2019-05-27
CA2768510A1 (en) 2011-02-10
EA023411B1 (ru) 2016-06-30
NZ597570A (en) 2014-04-30
SI2519512T1 (sl) 2019-09-30
AU2010279402A1 (en) 2012-02-02
KR20120041786A (ko) 2012-05-02
PE20120688A1 (es) 2012-06-06
ECSP12011653A (es) 2012-03-30
EP2519512A4 (en) 2013-01-16
TR201908180T4 (tr) 2019-06-21
IL217952A (en) 2017-11-30
CN102548981B (zh) 2015-05-13
CO6491117A2 (es) 2012-07-31
CR20120030A (es) 2012-03-28
EP2519512A1 (en) 2012-11-07
IL217952A0 (en) 2012-03-29
PL2519512T3 (pl) 2019-09-30
BR112012002810B1 (pt) 2018-12-11
JP2013501723A (ja) 2013-01-17
NI201200022A (es) 2012-05-22
ZA201200819B (en) 2013-05-29
CL2012000316A1 (es) 2014-06-27
HUE045290T2 (hu) 2019-12-30
HK1172894A1 (en) 2013-05-03
IN2012DN00539A (enEXAMPLES) 2015-06-12

Similar Documents

Publication Publication Date Title
US9862686B2 (en) N1-sulfonyl-5-fluoropyrimidinone derivatives
AU2010279402B2 (en) N1-acyl-5-fluoropyrimidinone derivatives
AU2010279408B2 (en) 5-fluoro-2-oxopyrimidine- 1(2H)-carboxylate derivatives
EP2461686B1 (en) N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
WO2011017540A1 (en) 5-fluoropyrimidinone derivatives
AU2010339900A1 (en) 2-aldoximino-5-fluoropyrimidine derivatives
AU2010279409B2 (en) N1-substituted-5-fluoro-2-oxopyrimidinone-1(2H)-carboxamide derivatives

Legal Events

Date Code Title Description
FGA Letters patent sealed or granted (standard patent)
PC Assignment registered

Owner name: ADAMA MAKHTESHIM LTD.

Free format text: FORMER OWNER(S): DOW AGROSCIENCES LLC

MK14 Patent ceased section 143(a) (annual fees not paid) or expired