OA12081A - Hygromycin derivatives. - Google Patents

Hygromycin derivatives. Download PDF

Info

Publication number
OA12081A
OA12081A OA1200200129A OA1200200129A OA12081A OA 12081 A OA12081 A OA 12081A OA 1200200129 A OA1200200129 A OA 1200200129A OA 1200200129 A OA1200200129 A OA 1200200129A OA 12081 A OA12081 A OA 12081A
Authority
OA
OAPI
Prior art keywords
alkyl
groups
aryl
independently
methyl
Prior art date
Application number
OA1200200129A
Other languages
English (en)
Inventor
Matthew Merrill Hayward
Takushi Kaneko
Linde Robert Gerald Ii
Katherine Elizabeth Brighty
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of OA12081A publication Critical patent/OA12081A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26Acyclic or carbocyclic radicals, substituted by hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
OA1200200129A 1999-10-29 2000-10-09 Hygromycin derivatives. OA12081A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16258199P 1999-10-29 1999-10-29

Publications (1)

Publication Number Publication Date
OA12081A true OA12081A (en) 2006-05-04

Family

ID=22586256

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200200129A OA12081A (en) 1999-10-29 2000-10-09 Hygromycin derivatives.

Country Status (32)

Country Link
US (1) US6562792B1 (es)
EP (1) EP1224197A1 (es)
JP (1) JP2003512473A (es)
KR (1) KR20020063885A (es)
CN (1) CN1382150A (es)
AP (1) AP2002002494A0 (es)
AR (1) AR023282A1 (es)
AU (1) AU7549400A (es)
BG (1) BG106727A (es)
BR (1) BR0015153A (es)
CA (1) CA2389191A1 (es)
CO (1) CO5261498A1 (es)
CZ (1) CZ20021355A3 (es)
EA (1) EA200200292A1 (es)
EE (1) EE200200228A (es)
GT (1) GT200000185A (es)
HK (1) HK1049672A1 (es)
HU (1) HUP0203525A3 (es)
IL (1) IL148577A0 (es)
IS (1) IS6311A (es)
MA (1) MA26838A1 (es)
MX (1) MXPA02004360A (es)
NO (1) NO20021850L (es)
OA (1) OA12081A (es)
PA (1) PA8505801A1 (es)
PE (1) PE20010763A1 (es)
PL (1) PL357083A1 (es)
SK (1) SK5472002A3 (es)
SV (1) SV2002000211A (es)
TN (1) TNSN00211A1 (es)
TR (1) TR200201145T2 (es)
WO (1) WO2001030795A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL152984A0 (en) 2000-06-02 2003-06-24 Pfizer Prod Inc Hygromycin a derivatives for the treatment of bacterial and protozoal infections
US6653481B2 (en) * 2000-12-29 2003-11-25 Synthon Bv Process for making amlodipine
US7923439B2 (en) * 2008-10-15 2011-04-12 Tyco Healthcare Group Lp Hydroxamate compositions
US20210275559A1 (en) * 2018-08-20 2021-09-09 Kim Lewis Hygromycin a compounds and methods of treating spirochete diseases
CR20220316A (es) 2019-12-06 2022-10-07 Vertex Pharma Tetrahidrofuranos sustituidos como moduladores de canales de sodio
CN117794920A (zh) 2021-06-04 2024-03-29 沃泰克斯药物股份有限公司 N-(羟烷基(杂)芳基)四氢呋喃甲酰胺作为钠通道调节剂

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL348063A1 (en) * 1998-12-02 2002-05-06 Pfizer Prod Inc Hygromycin a derivatives as antibacterial agents

Also Published As

Publication number Publication date
JP2003512473A (ja) 2003-04-02
PL357083A1 (en) 2004-07-12
CZ20021355A3 (cs) 2002-11-13
GT200000185A (es) 2002-04-18
HK1049672A1 (zh) 2003-05-23
KR20020063885A (ko) 2002-08-05
NO20021850D0 (no) 2002-04-19
SV2002000211A (es) 2002-07-16
IL148577A0 (en) 2002-09-12
CN1382150A (zh) 2002-11-27
HUP0203525A2 (hu) 2003-02-28
AR023282A1 (es) 2002-09-04
BR0015153A (pt) 2002-07-16
AP2002002494A0 (en) 2002-06-30
CO5261498A1 (es) 2003-03-31
PA8505801A1 (es) 2002-08-26
BG106727A (bg) 2003-01-31
TR200201145T2 (tr) 2002-09-23
SK5472002A3 (en) 2003-02-04
PE20010763A1 (es) 2001-07-25
CA2389191A1 (en) 2001-05-03
US6562792B1 (en) 2003-05-13
WO2001030795A1 (en) 2001-05-03
IS6311A (is) 2002-03-19
AU7549400A (en) 2001-05-08
NO20021850L (no) 2002-04-19
EA200200292A1 (ru) 2002-10-31
EP1224197A1 (en) 2002-07-24
MXPA02004360A (es) 2002-11-07
TNSN00211A1 (fr) 2005-11-10
HUP0203525A3 (en) 2003-08-28
MA26838A1 (fr) 2004-12-20
EE200200228A (et) 2003-06-16

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