OA11452A - Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems. - Google Patents

Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems. Download PDF

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Publication number
OA11452A
OA11452A OA1200000225A OA1200000225A OA11452A OA 11452 A OA11452 A OA 11452A OA 1200000225 A OA1200000225 A OA 1200000225A OA 1200000225 A OA1200000225 A OA 1200000225A OA 11452 A OA11452 A OA 11452A
Authority
OA
OAPI
Prior art keywords
formula
phenyl
compound
group
palladium
Prior art date
Application number
OA1200000225A
Other languages
English (en)
Inventor
Megan Elizabeth Hnatow
Timothy Norris
John Francis Lambert
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of OA11452A publication Critical patent/OA11452A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
OA1200000225A 1999-08-31 2000-08-18 Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems. OA11452A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US15161599P 1999-08-31 1999-08-31

Publications (1)

Publication Number Publication Date
OA11452A true OA11452A (en) 2003-12-08

Family

ID=22539529

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200000225A OA11452A (en) 1999-08-31 2000-08-18 Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems.

Country Status (33)

Country Link
US (1) US6346624B1 (pt)
EP (1) EP1081143A1 (pt)
JP (1) JP2001106682A (pt)
KR (1) KR20010050256A (pt)
CN (1) CN1286250A (pt)
AP (1) AP2000001910A0 (pt)
AU (1) AU5360300A (pt)
BG (1) BG104731A (pt)
BR (1) BR0003945A (pt)
CA (1) CA2317097A1 (pt)
CZ (1) CZ20003158A3 (pt)
EA (1) EA200000801A1 (pt)
EE (1) EE200000512A (pt)
GT (1) GT200000142A (pt)
HR (1) HRP20000564A2 (pt)
HU (1) HUP0003439A3 (pt)
ID (1) ID27129A (pt)
IL (1) IL138087A0 (pt)
IS (1) IS5603A (pt)
MA (1) MA26751A1 (pt)
NO (1) NO20004313L (pt)
NZ (1) NZ506632A (pt)
OA (1) OA11452A (pt)
PA (1) PA8499701A1 (pt)
PE (1) PE20010520A1 (pt)
PL (1) PL342281A1 (pt)
SG (1) SG87146A1 (pt)
SK (1) SK12872000A3 (pt)
SV (1) SV2002000159A (pt)
TN (1) TNSN00177A1 (pt)
TR (1) TR200002529A2 (pt)
UY (1) UY26314A1 (pt)
ZA (1) ZA200004435B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6669042B1 (en) * 2002-09-30 2003-12-30 Hewlett-Packard Development Company, L.P. Integrated positioning and locking device
US7674811B2 (en) 2006-03-14 2010-03-09 Ranbaxy Laboratories Limited 5-lipoxygenase inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5883106A (en) * 1994-10-18 1999-03-16 Pfizer Inc. 5-lipoxygenase inhibitors
US6063928A (en) * 1994-10-18 2000-05-16 Pfizer Inc 5-lipoxygenase inhibitors
SK281577B6 (sk) 1994-10-18 2001-05-10 Pfizer Inc. Heterocyklické zlúčeniny a farmaceutický prostriedok na ich báze
US6239285B1 (en) * 1998-02-06 2001-05-29 Pfizer Inc Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems

Also Published As

Publication number Publication date
PE20010520A1 (es) 2001-04-28
NO20004313L (no) 2001-03-01
HUP0003439A2 (hu) 2001-08-28
HUP0003439A3 (en) 2002-08-28
TR200002529A2 (tr) 2001-04-20
EE200000512A (et) 2001-04-16
CA2317097A1 (en) 2001-02-28
NZ506632A (en) 2002-02-01
ZA200004435B (en) 2002-02-28
BG104731A (en) 2001-09-28
IS5603A (is) 2001-03-01
NO20004313D0 (no) 2000-08-30
HRP20000564A2 (en) 2001-12-31
HU0003439D0 (en) 2000-08-30
SG87146A1 (en) 2002-03-19
ID27129A (id) 2001-03-01
JP2001106682A (ja) 2001-04-17
IL138087A0 (en) 2001-10-31
SK12872000A3 (sk) 2001-11-06
UY26314A1 (es) 2001-04-30
GT200000142A (es) 2002-02-19
BR0003945A (pt) 2001-04-03
PL342281A1 (en) 2001-03-12
PA8499701A1 (es) 2001-12-14
EP1081143A1 (en) 2001-03-07
EA200000801A1 (ru) 2001-04-23
US6346624B1 (en) 2002-02-12
KR20010050256A (ko) 2001-06-15
CN1286250A (zh) 2001-03-07
MA26751A1 (fr) 2004-12-20
TNSN00177A1 (fr) 2005-11-10
SV2002000159A (es) 2002-01-23
CZ20003158A3 (cs) 2001-09-12
AU5360300A (en) 2001-03-08
AP2000001910A0 (en) 2000-09-30

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