OA06504A - Dérivés du benzothiazole, leur procédé de préparation et leurs applications en thérapeutique. - Google Patents
Dérivés du benzothiazole, leur procédé de préparation et leurs applications en thérapeutique.Info
- Publication number
- OA06504A OA06504A OA57074A OA57074A OA06504A OA 06504 A OA06504 A OA 06504A OA 57074 A OA57074 A OA 57074A OA 57074 A OA57074 A OA 57074A OA 06504 A OA06504 A OA 06504A
- Authority
- OA
- OAPI
- Prior art keywords
- preparation process
- therapeutic applications
- benzothiazole derivatives
- benzothiazole
- derivatives
- Prior art date
Links
- IOJUPLGTWVMSFF-UHFFFAOYSA-N benzothiazole Chemical class C1=CC=C2SC=NC2=C1 IOJUPLGTWVMSFF-UHFFFAOYSA-N 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
- C07D277/66—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2 with aromatic rings or ring systems directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Hematology (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7908303A FR2453163A1 (fr) | 1979-04-03 | 1979-04-03 | Derives de benzothiazole, leur procede de preparation et leurs applications en therapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| OA06504A true OA06504A (fr) | 1981-07-31 |
Family
ID=9223868
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| OA57074A OA06504A (fr) | 1979-04-03 | 1980-04-03 | Dérivés du benzothiazole, leur procédé de préparation et leurs applications en thérapeutique. |
Country Status (27)
| Country | Link |
|---|---|
| EP (1) | EP0017543B1 (de) |
| JP (1) | JPS55133367A (de) |
| AR (1) | AR227884A1 (de) |
| AT (1) | ATE4807T1 (de) |
| AU (1) | AU530911B2 (de) |
| BE (1) | BE882270A (de) |
| CA (1) | CA1144556A (de) |
| DD (1) | DD151448A5 (de) |
| DE (1) | DE3065004D1 (de) |
| DK (1) | DK134880A (de) |
| ES (2) | ES490797A0 (de) |
| FI (1) | FI801023A7 (de) |
| FR (1) | FR2453163A1 (de) |
| GR (1) | GR67195B (de) |
| HU (1) | HU178851B (de) |
| IL (1) | IL59655A (de) |
| IT (1) | IT8048308A0 (de) |
| MA (1) | MA18772A1 (de) |
| NO (1) | NO800946L (de) |
| NZ (1) | NZ193337A (de) |
| OA (1) | OA06504A (de) |
| PH (1) | PH15451A (de) |
| PL (1) | PL123701B1 (de) |
| PT (1) | PT71035A (de) |
| SU (1) | SU910120A3 (de) |
| YU (1) | YU80780A (de) |
| ZA (1) | ZA801574B (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60329898D1 (de) | 2002-02-05 | 2009-12-17 | Sumitomo Chemical Co | Verfahren zur herstellung einer biarylverbindung |
| AP2013006707A0 (en) | 2010-07-02 | 2013-02-28 | Gilead Sciences Inc | 2-Quinolinyl-acetic acid derivatives as HIV antiviral compounds |
| TWI453208B (zh) | 2010-07-02 | 2014-09-21 | Gilead Sciences Inc | 治療性化合物類 |
| EP3181555B1 (de) * | 2011-04-21 | 2018-11-28 | Gilead Sciences, Inc. | Benzothiazolverbindungen und deren pharmazeutische verwendung |
| WO2013103724A1 (en) | 2012-01-04 | 2013-07-11 | Gilead Sciences, Inc. | 2- (tert - butoxy) -2- (7 -methylquinolin- 6 - yl) acetic acid derivatives for treating aids |
| WO2013103738A1 (en) | 2012-01-04 | 2013-07-11 | Gilead Sciences, Inc. | Napthalene acetic acid derivatives against hiv infection |
| ES2571479T3 (es) | 2012-04-20 | 2016-05-25 | Gilead Sciences Inc | Derivados del ácido benzotiazol-6-il acético y su uso para tratar una infección por VIH |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2145178C3 (de) * | 1970-09-11 | 1975-12-11 | Tokyo Tanabe Co., Ltd., Tokio | 2-Phenyl-5-oder -6-benzothiazolylessigsäure-Verblndungen |
| US3895028A (en) * | 1972-09-12 | 1975-07-15 | Tokyo Tanabe Co | Alpha-(2-phenylbenzothiazol-5-yl)propionic acid |
-
1979
- 1979-04-03 FR FR7908303A patent/FR2453163A1/fr active Granted
-
1980
- 1980-03-10 MA MA18970A patent/MA18772A1/fr unknown
- 1980-03-17 GR GR61462A patent/GR67195B/el unknown
- 1980-03-17 BE BE0/199830A patent/BE882270A/fr not_active IP Right Cessation
- 1980-03-18 IL IL59655A patent/IL59655A/xx unknown
- 1980-03-18 ZA ZA00801574A patent/ZA801574B/xx unknown
- 1980-03-19 EP EP80400368A patent/EP0017543B1/de not_active Expired
- 1980-03-19 AT AT80400368T patent/ATE4807T1/de not_active IP Right Cessation
- 1980-03-19 DE DE8080400368T patent/DE3065004D1/de not_active Expired
- 1980-03-24 YU YU00807/80A patent/YU80780A/xx unknown
- 1980-03-26 AU AU56864/80A patent/AU530911B2/en not_active Ceased
- 1980-03-28 PT PT71035A patent/PT71035A/pt unknown
- 1980-03-28 DK DK134880A patent/DK134880A/da not_active Application Discontinuation
- 1980-03-31 AR AR280502A patent/AR227884A1/es active
- 1980-04-01 FI FI801023A patent/FI801023A7/fi not_active Application Discontinuation
- 1980-04-01 PH PH23847A patent/PH15451A/en unknown
- 1980-04-01 SU SU802901454A patent/SU910120A3/ru active
- 1980-04-01 CA CA000348939A patent/CA1144556A/en not_active Expired
- 1980-04-01 ES ES490797A patent/ES490797A0/es active Granted
- 1980-04-01 NO NO800946A patent/NO800946L/no unknown
- 1980-04-01 IT IT8048308A patent/IT8048308A0/it unknown
- 1980-04-02 NZ NZ193337A patent/NZ193337A/xx unknown
- 1980-04-02 PL PL1980223191A patent/PL123701B1/pl unknown
- 1980-04-02 HU HU8080789A patent/HU178851B/hu unknown
- 1980-04-02 DD DD80220177A patent/DD151448A5/de unknown
- 1980-04-03 JP JP4402480A patent/JPS55133367A/ja active Pending
- 1980-04-03 OA OA57074A patent/OA06504A/xx unknown
- 1980-12-11 ES ES498313A patent/ES8204989A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| PH15451A (en) | 1983-01-18 |
| DD151448A5 (de) | 1981-10-21 |
| YU80780A (en) | 1983-02-28 |
| SU910120A3 (ru) | 1982-02-28 |
| PL123701B1 (en) | 1982-11-30 |
| MA18772A1 (fr) | 1980-10-01 |
| DK134880A (da) | 1980-10-04 |
| ZA801574B (en) | 1981-03-25 |
| PT71035A (fr) | 1980-04-01 |
| GR67195B (de) | 1981-06-24 |
| ES8200098A1 (es) | 1981-11-01 |
| NZ193337A (en) | 1982-12-07 |
| NO800946L (no) | 1980-10-06 |
| FR2453163B1 (de) | 1982-07-02 |
| AU530911B2 (en) | 1983-08-04 |
| IT8048308A0 (it) | 1980-04-01 |
| AU5686480A (en) | 1980-10-09 |
| PL223191A1 (de) | 1981-01-30 |
| BE882270A (fr) | 1980-09-17 |
| ATE4807T1 (de) | 1983-10-15 |
| CA1144556A (en) | 1983-04-12 |
| ES490797A0 (es) | 1981-11-01 |
| DE3065004D1 (en) | 1983-11-03 |
| EP0017543B1 (de) | 1983-09-28 |
| IL59655A (en) | 1983-05-15 |
| FI801023A7 (fi) | 1981-01-01 |
| AR227884A1 (es) | 1982-12-30 |
| HU178851B (en) | 1982-07-28 |
| JPS55133367A (en) | 1980-10-17 |
| FR2453163A1 (fr) | 1980-10-31 |
| IL59655A0 (en) | 1980-06-30 |
| ES498313A0 (es) | 1982-06-01 |
| ES8204989A1 (es) | 1982-06-01 |
| EP0017543A1 (de) | 1980-10-15 |
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