NZ333737A - Parenteral formulations of taxane analogs comprising dimethylacetamide, polyethylene glycol and an aqueous lipid emulsion - Google Patents
Parenteral formulations of taxane analogs comprising dimethylacetamide, polyethylene glycol and an aqueous lipid emulsionInfo
- Publication number
- NZ333737A NZ333737A NZ333737A NZ33373797A NZ333737A NZ 333737 A NZ333737 A NZ 333737A NZ 333737 A NZ333737 A NZ 333737A NZ 33373797 A NZ33373797 A NZ 33373797A NZ 333737 A NZ333737 A NZ 333737A
- Authority
- NZ
- New Zealand
- Prior art keywords
- paclitaxel
- pharmaceutical composition
- dma
- peg
- pachtaxel
- Prior art date
Links
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Dermatology (AREA)
- Organic Chemistry (AREA)
- Dispersion Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/672,594 US5877205A (en) | 1996-06-28 | 1996-06-28 | Parenteral paclitaxel in a stable non-toxic formulation |
| PCT/US1997/011503 WO1998000128A1 (en) | 1996-06-28 | 1997-06-26 | Parenteral paclitaxel in a stable non-toxic formulation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NZ333737A true NZ333737A (en) | 2000-02-28 |
Family
ID=24699210
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NZ333737A NZ333737A (en) | 1996-06-28 | 1997-06-26 | Parenteral formulations of taxane analogs comprising dimethylacetamide, polyethylene glycol and an aqueous lipid emulsion |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US5877205A (enExample) |
| EP (1) | EP0920311A4 (enExample) |
| JP (1) | JP2000515132A (enExample) |
| CN (1) | CN1165300C (enExample) |
| AU (1) | AU722617B2 (enExample) |
| CA (1) | CA2259297C (enExample) |
| NO (1) | NO986165L (enExample) |
| NZ (1) | NZ333737A (enExample) |
| WO (1) | WO1998000128A1 (enExample) |
Families Citing this family (56)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6245805B1 (en) * | 1995-10-26 | 2001-06-12 | Baker Norton Pharmaceuticals, Inc. | Method, compositions and kits for increasing the oral bioavailability of pharmaceutical agents |
| US6964946B1 (en) * | 1995-10-26 | 2005-11-15 | Baker Norton Pharmaceuticals, Inc. | Oral pharmaceutical compositions containing taxanes and methods of treatment employing the same |
| US20030157187A1 (en) * | 1996-12-02 | 2003-08-21 | Angiotech Pharmaceuticals, Inc. | Compositions and methods for treating or preventing inflammatory diseases |
| US20030105156A1 (en) * | 1997-01-07 | 2003-06-05 | Nagesh Palepu | Method for administration of a taxane/tocopherol formulation to enhance taxane therapeutic utility |
| US6458373B1 (en) * | 1997-01-07 | 2002-10-01 | Sonus Pharmaceuticals, Inc. | Emulsion vehicle for poorly soluble drugs |
| US20030087954A1 (en) * | 1997-01-07 | 2003-05-08 | Sonus Pharmaceuticals, Inc. | Method of treating bladder carcinoma using a Taxane/Tocopherol formulation |
| US6727280B2 (en) * | 1997-01-07 | 2004-04-27 | Sonus Pharmaceuticals, Inc. | Method for treating colorectal carcinoma using a taxane/tocopherol formulation |
| US6045815A (en) * | 1997-08-15 | 2000-04-04 | Board Of Regents, The University Of Texas System | Parenteral pimaricin as treatment of systemic infections |
| US6844004B2 (en) | 1997-08-15 | 2005-01-18 | Board Of Regents, The University Of Texas System | Topical formulations of natamycin/pimaricin |
| JP4644364B2 (ja) * | 1998-02-05 | 2011-03-02 | ノバルティス アーゲー | エポシロン組成物 |
| IL131217A0 (en) * | 1998-03-10 | 2001-01-28 | Napro Biotherapeutics Inc | Novel methods and compositions for delivery of taxanes |
| KR19990075621A (ko) * | 1998-03-23 | 1999-10-15 | 임성주 | 경사 평판형 배양조 |
| KR100446959B1 (ko) * | 1998-04-02 | 2004-11-03 | 김종국 | 파클리탁셀주사제조성물 |
| US7030155B2 (en) * | 1998-06-05 | 2006-04-18 | Sonus Pharmaceuticals, Inc. | Emulsion vehicle for poorly soluble drugs |
| US6017948A (en) * | 1998-10-30 | 2000-01-25 | Supergen, Inc. | Water-miscible pharmaceutical compositions |
| JP2002532535A (ja) * | 1998-12-22 | 2002-10-02 | アメリカ合衆国 | 水不溶性薬剤送達システム |
| US6040330A (en) * | 1999-01-08 | 2000-03-21 | Bionumerik Pharmaceuticals, Inc. | Pharmaceutical formulations of taxanes |
| US6121257A (en) * | 1999-03-31 | 2000-09-19 | Abbott Laboratories | Sulfamate containing macrocyclic immunomodulators |
| HK1049787B (en) | 1999-10-01 | 2014-07-25 | Immunogen, Inc. | Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents |
| SE9903831D0 (sv) | 1999-10-22 | 1999-10-22 | Astra Ab | Formulation of substituted benzimidazoles |
| US20040009229A1 (en) * | 2000-01-05 | 2004-01-15 | Unger Evan Charles | Stabilized nanoparticle formulations of camptotheca derivatives |
| CA2367661A1 (en) * | 2000-02-02 | 2001-08-09 | Robert A. Holton | Taxane formulations having improved solubility |
| MXPA02010999A (es) | 2000-05-12 | 2003-03-10 | Samyang Corp | Metodo para la preparacion de micelas polimericas por medio de la separacion de fase de copolimero de bloque. |
| US7217770B2 (en) * | 2000-05-17 | 2007-05-15 | Samyang Corporation | Stable polymeric micelle-type drug composition and method for the preparation thereof |
| CA2417840A1 (en) * | 2000-08-02 | 2002-02-07 | Atossa Healthcare, Inc. | Bimodal emulsions of taxanes and butyrate polyalcohol esters |
| US6919370B2 (en) * | 2000-11-28 | 2005-07-19 | Transform Pharmaceuticals, Inc. | Pharmaceutical formulations comprising paclitaxel, derivatives, and pharmaceutically acceptable salts thereof |
| US20040241094A1 (en) * | 2001-09-13 | 2004-12-02 | Hesson Chung | Oily paclitaxel composition and formulation for chemoembolization and preparation method thereof |
| WO2003045357A1 (en) * | 2001-11-27 | 2003-06-05 | Transform Pharmaceuticals, Inc. | Oral pharmaceutical formulations comprising paclitaxel, derivatives and methods of administration thereof |
| EP1451168A4 (en) * | 2001-11-30 | 2005-08-24 | Bristol Myers Squibb Co | PACLITAXELSOLVATE |
| US20060078618A1 (en) * | 2001-12-11 | 2006-04-13 | Constantinides Panayiotis P | Lipid particles and suspensions and uses thereof |
| US20040213837A1 (en) * | 2002-08-05 | 2004-10-28 | Sankaram Mantripragada | Oil-core compositions for the sustained release of hydrophobic drugs |
| US20050129719A1 (en) * | 2003-12-15 | 2005-06-16 | Yu-Fang Hu | Concentrated emulsion formulation for silatecan |
| US20050220835A1 (en) * | 2004-03-30 | 2005-10-06 | Jayaraman Ramesh B | Agent eluting bioimplantable devices and polymer systems for their preparation |
| DK1792927T3 (da) | 2004-09-22 | 2013-06-10 | Nippon Kayaku Kk | Ny blokcopolymer, micelletilberedning og anticancermiddel indeholdende samme som aktiv ingrediens |
| EP1909771A1 (en) * | 2005-08-02 | 2008-04-16 | Miv Therapeutics Inc. | Microdevices comprising nanocapsules for controlled delivery of drugs and method of manufacturing same |
| WO2007111211A1 (ja) * | 2006-03-28 | 2007-10-04 | Nippon Kayaku Kabushiki Kaisha | タキサン類の高分子結合体 |
| US8940332B2 (en) | 2006-05-18 | 2015-01-27 | Nippon Kayaku Kabushiki Kaisha | High-molecular weight conjugate of podophyllotoxins |
| CA2664852A1 (en) * | 2006-10-03 | 2008-04-10 | Nippon Kayaku Kabushiki Kaisha | High-molecular weight conjugate of resorcinol derivatives |
| US8334364B2 (en) | 2006-11-06 | 2012-12-18 | Nipon Kayaku Kabushiki Kaisha | High-molecular weight derivative of nucleic acid antimetabolite |
| EP2090607B1 (en) | 2006-11-08 | 2015-05-20 | Nippon Kayaku Kabushiki Kaisha | Polymeric derivative of nucleic acid metabolic antagonist |
| WO2009041570A1 (ja) | 2007-09-28 | 2009-04-02 | Nippon Kayaku Kabushiki Kaisha | ステロイド類の高分子結合体 |
| AR063111A1 (es) | 2007-10-03 | 2008-12-30 | Eriochem Sa | Una formulacion farmaceutica de taxano |
| CN101977631A (zh) * | 2008-03-18 | 2011-02-16 | 日本化药株式会社 | 生理活性物质的高分子量偶联物 |
| US9149540B2 (en) | 2008-05-08 | 2015-10-06 | Nippon Kayaku Kabushiki Kaisha | Polymer conjugate of folic acid or folic acid derivative |
| WO2010131675A1 (ja) | 2009-05-15 | 2010-11-18 | 日本化薬株式会社 | 水酸基を有する生理活性物質の高分子結合体 |
| CN102038634B (zh) * | 2009-10-23 | 2014-12-10 | 天士力控股集团有限公司 | 一种含有助溶剂的紫杉烷类药物溶液及其制备方法 |
| CN102038636B (zh) * | 2009-10-23 | 2014-08-13 | 天士力控股集团有限公司 | 一种含有螯合剂的紫杉烷类药物溶液及其制备方法 |
| CN102038635A (zh) * | 2009-10-23 | 2011-05-04 | 天津天士力集团有限公司 | 一种含有pH值调节剂的紫杉烷类药物溶液及其制备方法 |
| TWI438009B (zh) * | 2010-02-19 | 2014-05-21 | Teikoku Pharma Usa Inc | 紫杉烷前－乳劑調配物及其製造與使用之方法 |
| EP2566474B1 (en) | 2010-05-03 | 2017-11-15 | Teikoku Pharma USA, Inc. | Non-aqueous taxane pro-emulsion formulations and methods of making and using the same |
| TWI472340B (zh) * | 2010-11-10 | 2015-02-11 | Tasly Holding Group Co Ltd | Taxanes containing solution and a preparation method of the co-solvent |
| US9018323B2 (en) | 2010-11-17 | 2015-04-28 | Nippon Kayaku Kabushiki Kaisha | Polymer derivative of cytidine metabolic antagonist |
| EP2754682B1 (en) * | 2011-09-11 | 2017-06-07 | Nippon Kayaku Kabushiki Kaisha | Method for manufacturing block copolymer |
| JO3685B1 (ar) | 2012-10-01 | 2020-08-27 | Teikoku Pharma Usa Inc | صيغ التشتيت الجسيمي للتاكسين غير المائي وطرق استخدامها |
| CN109464382B (zh) * | 2019-01-08 | 2020-10-09 | 四川大学 | 一种可注射的高载药量的紫杉醇凝胶及其制备方法和应用 |
| CA3235911A1 (en) * | 2021-10-21 | 2023-04-27 | Kashiv Biosciences, Llc | Stable ready to dilute composition of carfilzomib |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2698543B1 (fr) * | 1992-12-02 | 1994-12-30 | Rhone Poulenc Rorer Sa | Nouvelles compositions à base de taxoides. |
| US5430057A (en) * | 1993-09-30 | 1995-07-04 | Board Of Regents, The University Of Texas System | Parenteral busulfan for treatment of malignant disease |
| US5597829A (en) * | 1994-05-09 | 1997-01-28 | Bionumerik Pharmaceuticals, Inc. | Lactone stable formulation of camptothecin and methods for uses thereof |
| TW372967B (en) * | 1994-12-27 | 1999-11-01 | Kanebo Ltd | 1,4 benzoxazine derivative, pharmaceutical composition containing the same and use thereof |
-
1996
- 1996-06-28 US US08/672,594 patent/US5877205A/en not_active Expired - Fee Related
-
1997
- 1997-06-26 AU AU36478/97A patent/AU722617B2/en not_active Ceased
- 1997-06-26 EP EP97933246A patent/EP0920311A4/en not_active Withdrawn
- 1997-06-26 NZ NZ333737A patent/NZ333737A/en unknown
- 1997-06-26 WO PCT/US1997/011503 patent/WO1998000128A1/en not_active Ceased
- 1997-06-26 JP JP10504432A patent/JP2000515132A/ja not_active Ceased
- 1997-06-26 CN CNB971969345A patent/CN1165300C/zh not_active Expired - Fee Related
- 1997-06-26 CA CA002259297A patent/CA2259297C/en not_active Expired - Fee Related
-
1998
- 1998-12-28 NO NO986165A patent/NO986165L/no unknown
-
1999
- 1999-03-01 US US09/259,533 patent/US6107333A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US5877205A (en) | 1999-03-02 |
| NO986165D0 (no) | 1998-12-28 |
| EP0920311A1 (en) | 1999-06-09 |
| JP2000515132A (ja) | 2000-11-14 |
| AU3647897A (en) | 1998-01-21 |
| CA2259297C (en) | 2003-12-16 |
| NO986165L (no) | 1999-02-25 |
| EP0920311A4 (en) | 2001-10-04 |
| CA2259297A1 (en) | 1998-01-08 |
| US6107333A (en) | 2000-08-22 |
| CN1165300C (zh) | 2004-09-08 |
| WO1998000128A1 (en) | 1998-01-08 |
| AU722617B2 (en) | 2000-08-10 |
| CN1228022A (zh) | 1999-09-08 |
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Legal Events
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| RENW | Renewal (renewal fees accepted) | ||
| ERR | Error or correction |
Free format text: THE OWNER HAS BEEN CORRECTED TO 857962, BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM, 201 WEST 7TH STREET, AUSTIN, TEXAS 78701, US Effective date: 20140808 |