NZ207259A - C-20 and c-23 modified macrolides - Google Patents

C-20 and c-23 modified macrolides

Info

Publication number
NZ207259A
NZ207259A NZ207259A NZ20725984A NZ207259A NZ 207259 A NZ207259 A NZ 207259A NZ 207259 A NZ207259 A NZ 207259A NZ 20725984 A NZ20725984 A NZ 20725984A NZ 207259 A NZ207259 A NZ 207259A
Authority
NZ
New Zealand
Prior art keywords
formula
rnacrolide
optionally substituted
give
hydrogen
Prior art date
Application number
NZ207259A
Other languages
English (en)
Inventor
M Debona
H A Kirst
J E Toth
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/470,890 external-priority patent/US4468511A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of NZ207259A publication Critical patent/NZ207259A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
NZ207259A 1983-02-28 1984-02-23 C-20 and c-23 modified macrolides NZ207259A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US47083383A 1983-02-28 1983-02-28
US06/470,890 US4468511A (en) 1983-02-28 1983-02-28 C-20- And C-23-Modified macrolide derivatives

Publications (1)

Publication Number Publication Date
NZ207259A true NZ207259A (en) 1987-02-20

Family

ID=27043239

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ207259A NZ207259A (en) 1983-02-28 1984-02-23 C-20 and c-23 modified macrolides

Country Status (14)

Country Link
EP (1) EP0124216B1 (forum.php)
KR (1) KR860001282B1 (forum.php)
AU (1) AU561861B2 (forum.php)
DE (1) DE3474831D1 (forum.php)
DK (1) DK98184A (forum.php)
ES (1) ES530081A0 (forum.php)
FI (1) FI840780A7 (forum.php)
GB (1) GB2135670B (forum.php)
GR (1) GR79821B (forum.php)
HU (1) HUT35693A (forum.php)
IL (1) IL71032A0 (forum.php)
NZ (1) NZ207259A (forum.php)
PL (1) PL246417A1 (forum.php)
PT (1) PT78141A (forum.php)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4515941A (en) * 1982-04-07 1985-05-07 Toyo Jozo Kabushiki Kaisha 23-Demycinosyldesmycosin derivatives
US4604380A (en) * 1985-01-18 1986-08-05 Eli Lilly And Company C-23-substituted mycaminosyltylonolide compounds, pharmaceutical compositions and methods of use
FR2646081A1 (forum.php) * 1989-04-20 1990-10-26 Adir
ES2099941T3 (es) * 1992-01-14 1997-06-01 Zaidan Hojin Biseibutsu Derivado de 3,4'-didesoxi-micaminosiltilonolido y su produccion.
TW226373B (forum.php) * 1992-07-15 1994-07-11 Pfizer
WO1994021657A1 (en) * 1993-03-18 1994-09-29 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at c-20
AU6980094A (en) * 1993-07-15 1995-02-13 Pfizer Inc. Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
DK1216256T3 (da) * 1999-08-30 2004-06-21 Zaidan Hojin Biseibutsu Makrolid-antibiotika og behandling af pasteurellosis
CN102875622B (zh) * 2006-07-28 2016-12-07 英特威国际有限公司 大环内酯合成方法
JP5323696B2 (ja) 2006-07-28 2013-10-23 インターベツト・インターナシヨナル・ベー・ベー マクロライド合成方法
CN105408340B (zh) 2013-05-23 2020-06-12 拜耳动物保健有限责任公司 泰乐菌素衍生物及其制备方法
CN108299531B (zh) * 2018-01-23 2021-02-05 郑州大学 甲哌泰万菌素可药用盐及其制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
ZA813578B (en) * 1980-06-12 1983-01-26 Lilly Co Eli Macrolide antibiotics
US4321361A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company Demycinosyltylosin and process for its production
US4304856A (en) * 1980-11-10 1981-12-08 Eli Lilly And Company Process for producing 20-dihydro-20-deoxy-23-demycinosyltylosin
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin

Also Published As

Publication number Publication date
GR79821B (forum.php) 1984-10-31
GB2135670A (en) 1984-09-05
DE3474831D1 (en) 1988-12-01
HUT35693A (en) 1985-07-29
KR840007733A (ko) 1984-12-10
FI840780A0 (fi) 1984-02-27
FI840780A7 (fi) 1984-08-29
IL71032A0 (en) 1984-05-31
DK98184A (da) 1984-08-29
ES8602742A1 (es) 1985-12-01
GB2135670B (en) 1987-07-08
EP0124216A1 (en) 1984-11-07
EP0124216B1 (en) 1988-10-26
DK98184D0 (da) 1984-02-24
AU561861B2 (en) 1987-05-21
AU2503584A (en) 1984-09-06
KR860001282B1 (ko) 1986-09-05
PT78141A (en) 1984-03-01
ES530081A0 (es) 1985-12-01
GB8405086D0 (en) 1984-04-04
PL246417A1 (en) 1985-03-12

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