DK98184A - C-20- og c-23-modificerede derivater af tylosin-lignende makrolider og fremgangsmaade til fremstilling af saadanne derivater - Google Patents

C-20- og c-23-modificerede derivater af tylosin-lignende makrolider og fremgangsmaade til fremstilling af saadanne derivater Download PDF

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Publication number
DK98184A
DK98184A DK98184A DK98184A DK98184A DK 98184 A DK98184 A DK 98184A DK 98184 A DK98184 A DK 98184A DK 98184 A DK98184 A DK 98184A DK 98184 A DK98184 A DK 98184A
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DK
Denmark
Prior art keywords
derivatives
macrolids
tylosin
procedure
preparation
Prior art date
Application number
DK98184A
Other languages
English (en)
Other versions
DK98184D0 (da
Inventor
Manuel Debono
Herbert Andrew Kirst
John Eldon Toth
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/470,890 external-priority patent/US4468511A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DK98184D0 publication Critical patent/DK98184D0/da
Publication of DK98184A publication Critical patent/DK98184A/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK98184A 1983-02-28 1984-02-24 C-20- og c-23-modificerede derivater af tylosin-lignende makrolider og fremgangsmaade til fremstilling af saadanne derivater DK98184A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US47083383A 1983-02-28 1983-02-28
US06/470,890 US4468511A (en) 1983-02-28 1983-02-28 C-20- And C-23-Modified macrolide derivatives

Publications (2)

Publication Number Publication Date
DK98184D0 DK98184D0 (da) 1984-02-24
DK98184A true DK98184A (da) 1984-08-29

Family

ID=27043239

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98184A DK98184A (da) 1983-02-28 1984-02-24 C-20- og c-23-modificerede derivater af tylosin-lignende makrolider og fremgangsmaade til fremstilling af saadanne derivater

Country Status (14)

Country Link
EP (1) EP0124216B1 (da)
KR (1) KR860001282B1 (da)
AU (1) AU561861B2 (da)
DE (1) DE3474831D1 (da)
DK (1) DK98184A (da)
ES (1) ES8602742A1 (da)
FI (1) FI840780A (da)
GB (1) GB2135670B (da)
GR (1) GR79821B (da)
HU (1) HUT35693A (da)
IL (1) IL71032A0 (da)
NZ (1) NZ207259A (da)
PL (1) PL246417A1 (da)
PT (1) PT78141A (da)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4515941A (en) * 1982-04-07 1985-05-07 Toyo Jozo Kabushiki Kaisha 23-Demycinosyldesmycosin derivatives
US4604380A (en) * 1985-01-18 1986-08-05 Eli Lilly And Company C-23-substituted mycaminosyltylonolide compounds, pharmaceutical compositions and methods of use
FR2646081A1 (da) * 1989-04-20 1990-10-26 Adir
WO1993014101A1 (en) * 1992-01-14 1993-07-22 Zaidan Hojin Biseibutsu Kagaku Kenkyukai 3,4'-dideoxymycaminosyltylonolide derivative and production thereof
TW226373B (da) * 1992-07-15 1994-07-11 Pfizer
AU6019794A (en) * 1993-03-18 1994-10-11 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at c-20
US5716939A (en) * 1993-07-15 1998-02-10 Pfizer Inc. Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
EP1216256B1 (en) * 1999-08-30 2004-03-10 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Macrolide antibiotics and treatment of pasteurellosis
NZ574193A (en) * 2006-07-28 2011-09-30 Intervet Int Bv Macrolide synthesis process
KR101538599B1 (ko) 2006-07-28 2015-07-21 인터벳 인터내셔널 비.브이. 마크롤라이드 합성 방법
SI2999707T1 (en) 2013-05-23 2018-07-31 Bayer Animal Health Gmbh Tylosin derivatives and their preparation process
CN108299531B (zh) * 2018-01-23 2021-02-05 郑州大学 甲哌泰万菌素可药用盐及其制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
ZA813578B (en) * 1980-06-12 1983-01-26 Lilly Co Eli Macrolide antibiotics
US4321362A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company De(mycinosyloxy)tylosin and process for its production
US4304856A (en) * 1980-11-10 1981-12-08 Eli Lilly And Company Process for producing 20-dihydro-20-deoxy-23-demycinosyltylosin
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin

Also Published As

Publication number Publication date
GR79821B (da) 1984-10-31
FI840780A (fi) 1984-08-29
KR840007733A (ko) 1984-12-10
NZ207259A (en) 1987-02-20
GB2135670B (en) 1987-07-08
PT78141A (en) 1984-03-01
GB2135670A (en) 1984-09-05
GB8405086D0 (en) 1984-04-04
FI840780A0 (fi) 1984-02-27
EP0124216B1 (en) 1988-10-26
KR860001282B1 (ko) 1986-09-05
PL246417A1 (en) 1985-03-12
ES530081A0 (es) 1985-12-01
IL71032A0 (en) 1984-05-31
DK98184D0 (da) 1984-02-24
DE3474831D1 (en) 1988-12-01
EP0124216A1 (en) 1984-11-07
HUT35693A (en) 1985-07-29
ES8602742A1 (es) 1985-12-01
AU2503584A (en) 1984-09-06
AU561861B2 (en) 1987-05-21

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