DK350883D0 - Fremgangsmade til fremstilling af mycaminosyltylonolid og beslaegtede macrolidderivater og mellemprodukter herved - Google Patents
Fremgangsmade til fremstilling af mycaminosyltylonolid og beslaegtede macrolidderivater og mellemprodukter hervedInfo
- Publication number
- DK350883D0 DK350883D0 DK3508/83A DK350883A DK350883D0 DK 350883 D0 DK350883 D0 DK 350883D0 DK 3508/83 A DK3508/83 A DK 3508/83A DK 350883 A DK350883 A DK 350883A DK 350883 D0 DK350883 D0 DK 350883D0
- Authority
- DK
- Denmark
- Prior art keywords
- mycaminosyltylonolide
- intermediates
- procedure
- preparation
- macrolide derivatives
- Prior art date
Links
- WGUJDBLMJBJUQU-VKRLOHBMSA-N 5-O-mycaminosyltylonolide Chemical compound O=CC[C@H]1C[C@@H](C)C(=O)\C=C\C(\C)=C\[C@H](CO)[C@@H](CC)OC(=O)C[C@@H](O)[C@H](C)[C@H]1O[C@H]1[C@H](O)[C@@H](N(C)C)[C@H](O)[C@@H](C)O1 WGUJDBLMJBJUQU-VKRLOHBMSA-N 0.000 title 1
- 239000000543 intermediate Substances 0.000 title 1
- 239000003120 macrolide antibiotic agent Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/404,024 US4454314A (en) | 1982-08-02 | 1982-08-02 | Antibacterial mycaminosyl tylonolide and related macrolide derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK350883D0 true DK350883D0 (da) | 1983-08-01 |
| DK350883A DK350883A (da) | 1984-02-03 |
Family
ID=23597822
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK350883A DK350883A (da) | 1982-08-02 | 1983-08-01 | Fremgangsmaade til fremstilling af mycaminosyltylonolid og beslaegtede macrolidderivater og mellemprodukter herved |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US4454314A (da) |
| EP (1) | EP0100645A1 (da) |
| JP (1) | JPS5944398A (da) |
| CA (1) | CA1234108A (da) |
| DK (1) | DK350883A (da) |
| GR (1) | GR79350B (da) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6056995A (ja) * | 1983-09-06 | 1985-04-02 | Microbial Chem Res Found | ２３−デオキシ−２３−オキソ マイカミノシル タイロノライド |
| US4530921A (en) * | 1983-10-03 | 1985-07-23 | Merck & Co., Inc. | Avermectin epoxide derivatives and method of use |
| GB8405087D0 (en) * | 1984-02-27 | 1984-04-04 | Omura S | Antibiotic |
| US4604380A (en) * | 1985-01-18 | 1986-08-05 | Eli Lilly And Company | C-23-substituted mycaminosyltylonolide compounds, pharmaceutical compositions and methods of use |
| US4921947A (en) * | 1986-03-31 | 1990-05-01 | Eli Lilly And Company | Process for preparing macrolide derivatives |
| US4962146A (en) * | 1987-04-29 | 1990-10-09 | Schering Corporation | 3-O-glycosyl 16-membered macrolide antibacterials and related derivatives |
| WO1994021657A1 (en) * | 1993-03-18 | 1994-09-29 | Pfizer Inc. | Antibacterial 16-membered ring macrolides containing olefins at c-20 |
| JP4106104B2 (ja) * | 1997-03-10 | 2008-06-25 | 財団法人微生物化学研究会 | 新規マイカミノシルタイロノライド誘導体 |
| HRP980496B1 (en) * | 1998-09-10 | 2007-03-31 | GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. | New thilozine hydroxy derivatives and a process for the preparation thereof |
| DE122011100013I1 (de) | 1999-08-30 | 2011-09-15 | Zaidan Hojin Biseibutsu | Makrolid-antibiotika und behandlung von pasteurellosis. |
| US6753415B2 (en) | 2002-04-19 | 2004-06-22 | Enanta Pharmaceuticals, Inc. | 23-O-substituted 5-O-mycaminosyltylonide derivatives |
| JP5323696B2 (ja) | 2006-07-28 | 2013-10-23 | インターベツト・インターナシヨナル・ベー・ベー | マクロライド合成方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH630391A5 (en) * | 1975-02-28 | 1982-06-15 | Scherico Ltd | Process for preparing derivatives of rosaramicin |
| JPS5416493A (en) * | 1977-03-03 | 1979-02-07 | Yamanouchi Pharmaceut Co Ltd | Novel josamycin derivatives, their salts, and their preparation |
| JPS5622796A (en) * | 1979-08-03 | 1981-03-03 | Meiji Seika Kaisha Ltd | Novel derivative of demycarosyl-macrolide antibiotic |
| JPS56122397A (en) * | 1980-02-29 | 1981-09-25 | Satoshi Omura | Marcolides |
| US4279896A (en) * | 1980-06-23 | 1981-07-21 | Schering Corporation | Novel 20-imino macrolide antibacterial agents |
| US4438109A (en) * | 1980-07-25 | 1984-03-20 | Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai | Tylosin derivatives |
| JPS5815997A (ja) * | 1981-07-09 | 1983-01-29 | Microbial Chem Res Found | 新規なタイロシン誘導体 |
| AU551142B2 (en) * | 1981-07-09 | 1986-04-17 | Zaidan Hojin Biseibutsu Kagaku Kenkyukai | Tylosin derivatives |
| JPS5855497A (ja) * | 1981-09-29 | 1983-04-01 | Microbial Chem Res Found | 新規タイロシン誘導体 |
-
1982
- 1982-08-02 US US06/404,024 patent/US4454314A/en not_active Expired - Fee Related
-
1983
- 1983-07-27 EP EP83304331A patent/EP0100645A1/en not_active Withdrawn
- 1983-07-29 GR GR72092A patent/GR79350B/el unknown
- 1983-07-29 CA CA000433527A patent/CA1234108A/en not_active Expired
- 1983-08-01 DK DK350883A patent/DK350883A/da not_active Application Discontinuation
- 1983-08-02 JP JP58141820A patent/JPS5944398A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EP0100645A1 (en) | 1984-02-15 |
| CA1234108A (en) | 1988-03-15 |
| US4454314A (en) | 1984-06-12 |
| CA1259307C (da) | 1989-09-12 |
| DK350883A (da) | 1984-02-03 |
| JPS5944398A (ja) | 1984-03-12 |
| GR79350B (da) | 1984-10-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHS | Application shelved for other reasons than non-payment |