ES530081A0 - Un procedimiento para la preparacion de una macrolida - Google Patents

Un procedimiento para la preparacion de una macrolida

Info

Publication number
ES530081A0
ES530081A0 ES530081A ES530081A ES530081A0 ES 530081 A0 ES530081 A0 ES 530081A0 ES 530081 A ES530081 A ES 530081A ES 530081 A ES530081 A ES 530081A ES 530081 A0 ES530081 A0 ES 530081A0
Authority
ES
Spain
Prior art keywords
macrolide
procedure
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES530081A
Other languages
English (en)
Other versions
ES8602742A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/470,890 external-priority patent/US4468511A/en
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES8602742A1 publication Critical patent/ES8602742A1/es
Publication of ES530081A0 publication Critical patent/ES530081A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
ES530081A 1983-02-28 1984-02-27 Un procedimiento para la preparacion de una macrolida Granted ES530081A0 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US47083383A 1983-02-28 1983-02-28
US06/470,890 US4468511A (en) 1983-02-28 1983-02-28 C-20- And C-23-Modified macrolide derivatives

Publications (2)

Publication Number Publication Date
ES8602742A1 ES8602742A1 (es) 1985-12-01
ES530081A0 true ES530081A0 (es) 1985-12-01

Family

ID=27043239

Family Applications (1)

Application Number Title Priority Date Filing Date
ES530081A Granted ES530081A0 (es) 1983-02-28 1984-02-27 Un procedimiento para la preparacion de una macrolida

Country Status (14)

Country Link
EP (1) EP0124216B1 (es)
KR (1) KR860001282B1 (es)
AU (1) AU561861B2 (es)
DE (1) DE3474831D1 (es)
DK (1) DK98184A (es)
ES (1) ES530081A0 (es)
FI (1) FI840780A (es)
GB (1) GB2135670B (es)
GR (1) GR79821B (es)
HU (1) HUT35693A (es)
IL (1) IL71032A0 (es)
NZ (1) NZ207259A (es)
PL (1) PL246417A1 (es)
PT (1) PT78141A (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4515941A (en) * 1982-04-07 1985-05-07 Toyo Jozo Kabushiki Kaisha 23-Demycinosyldesmycosin derivatives
US4604380A (en) * 1985-01-18 1986-08-05 Eli Lilly And Company C-23-substituted mycaminosyltylonolide compounds, pharmaceutical compositions and methods of use
FR2646081A1 (es) * 1989-04-20 1990-10-26 Adir
ES2099941T3 (es) * 1992-01-14 1997-06-01 Zaidan Hojin Biseibutsu Derivado de 3,4'-didesoxi-micaminosiltilonolido y su produccion.
TW226373B (es) * 1992-07-15 1994-07-11 Pfizer
WO1994021657A1 (en) * 1993-03-18 1994-09-29 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at c-20
EP0708770B1 (en) * 1993-07-15 1997-04-16 Pfizer Inc. Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
PT1216256E (pt) * 1999-08-30 2004-07-30 Zaidan Hojin Biseibutsu Antibioticos macrolidos e tratamento de pasteurelose
MX2009001072A (es) * 2006-07-28 2009-06-26 Intervet Int Bv Proceso de sintesis de macrolido.
ES2374950T3 (es) * 2006-07-28 2012-02-23 Intervet International B.V. Procedimiento de síntesis de macrolidos.
KR102307218B1 (ko) 2013-05-23 2021-10-05 바이엘 애니멀 헬스 게엠베하 틸로신 유도체 및 그의 제조 방법
CN108299531B (zh) * 2018-01-23 2021-02-05 郑州大学 甲哌泰万菌素可药用盐及其制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
US4321362A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company De(mycinosyloxy)tylosin and process for its production
ZA813578B (en) * 1980-06-12 1983-01-26 Lilly Co Eli Macrolide antibiotics
US4304856A (en) * 1980-11-10 1981-12-08 Eli Lilly And Company Process for producing 20-dihydro-20-deoxy-23-demycinosyltylosin
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin

Also Published As

Publication number Publication date
GR79821B (es) 1984-10-31
DE3474831D1 (en) 1988-12-01
EP0124216B1 (en) 1988-10-26
GB2135670B (en) 1987-07-08
PL246417A1 (en) 1985-03-12
HUT35693A (en) 1985-07-29
FI840780A0 (fi) 1984-02-27
ES8602742A1 (es) 1985-12-01
AU2503584A (en) 1984-09-06
DK98184D0 (da) 1984-02-24
PT78141A (en) 1984-03-01
AU561861B2 (en) 1987-05-21
GB2135670A (en) 1984-09-05
EP0124216A1 (en) 1984-11-07
NZ207259A (en) 1987-02-20
FI840780A (fi) 1984-08-29
IL71032A0 (en) 1984-05-31
DK98184A (da) 1984-08-29
KR840007733A (ko) 1984-12-10
KR860001282B1 (ko) 1986-09-05
GB8405086D0 (en) 1984-04-04

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19960603