HUT35693A - Process for preparing macrolide derivatives modified on carbon 20. and 23. - Google Patents

Process for preparing macrolide derivatives modified on carbon 20. and 23.

Info

Publication number
HUT35693A
HUT35693A HU84770A HU77084A HUT35693A HU T35693 A HUT35693 A HU T35693A HU 84770 A HU84770 A HU 84770A HU 77084 A HU77084 A HU 77084A HU T35693 A HUT35693 A HU T35693A
Authority
HU
Hungary
Prior art keywords
carbon
derivatives modified
macrolide derivatives
preparing macrolide
preparing
Prior art date
Application number
HU84770A
Other languages
English (en)
Inventor
Manuel Debono
Herbert A Kirst
John E Toth
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/470,890 external-priority patent/US4468511A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of HUT35693A publication Critical patent/HUT35693A/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
HU84770A 1983-02-28 1984-02-27 Process for preparing macrolide derivatives modified on carbon 20. and 23. HUT35693A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US47083383A 1983-02-28 1983-02-28
US06/470,890 US4468511A (en) 1983-02-28 1983-02-28 C-20- And C-23-Modified macrolide derivatives

Publications (1)

Publication Number Publication Date
HUT35693A true HUT35693A (en) 1985-07-29

Family

ID=27043239

Family Applications (1)

Application Number Title Priority Date Filing Date
HU84770A HUT35693A (en) 1983-02-28 1984-02-27 Process for preparing macrolide derivatives modified on carbon 20. and 23.

Country Status (14)

Country Link
EP (1) EP0124216B1 (hu)
KR (1) KR860001282B1 (hu)
AU (1) AU561861B2 (hu)
DE (1) DE3474831D1 (hu)
DK (1) DK98184A (hu)
ES (1) ES8602742A1 (hu)
FI (1) FI840780A (hu)
GB (1) GB2135670B (hu)
GR (1) GR79821B (hu)
HU (1) HUT35693A (hu)
IL (1) IL71032A0 (hu)
NZ (1) NZ207259A (hu)
PL (1) PL246417A1 (hu)
PT (1) PT78141A (hu)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4515941A (en) * 1982-04-07 1985-05-07 Toyo Jozo Kabushiki Kaisha 23-Demycinosyldesmycosin derivatives
US4604380A (en) * 1985-01-18 1986-08-05 Eli Lilly And Company C-23-substituted mycaminosyltylonolide compounds, pharmaceutical compositions and methods of use
FR2646081A1 (hu) * 1989-04-20 1990-10-26 Adir
EP0627443B1 (en) * 1992-01-14 1997-03-26 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai 3,4'-dideoxymycaminosyltylonolide derivative and production thereof
TW226373B (hu) * 1992-07-15 1994-07-11 Pfizer
US5677287A (en) * 1993-03-18 1997-10-14 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at C-20
ATE151767T1 (de) * 1993-07-15 1997-05-15 Pfizer Amid-derivate von 16-gliedrige heterocyclen als antibiotische macrolide
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
CA2391834C (en) * 1999-08-30 2008-08-05 Toshiaki Miyake Macrolide antibiotics and treatment of pasteurellosis
CN102875622B (zh) * 2006-07-28 2016-12-07 英特威国际有限公司 大环内酯合成方法
JP5323696B2 (ja) 2006-07-28 2013-10-23 インターベツト・インターナシヨナル・ベー・ベー マクロライド合成方法
NO2999707T3 (hu) 2013-05-23 2018-08-25
CN108299531B (zh) * 2018-01-23 2021-02-05 郑州大学 甲哌泰万菌素可药用盐及其制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
ZA813578B (en) * 1980-06-12 1983-01-26 Lilly Co Eli Macrolide antibiotics
US4321361A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company Demycinosyltylosin and process for its production
US4304856A (en) * 1980-11-10 1981-12-08 Eli Lilly And Company Process for producing 20-dihydro-20-deoxy-23-demycinosyltylosin
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin

Also Published As

Publication number Publication date
FI840780A (fi) 1984-08-29
EP0124216B1 (en) 1988-10-26
DK98184D0 (da) 1984-02-24
ES530081A0 (es) 1985-12-01
GB2135670A (en) 1984-09-05
GB8405086D0 (en) 1984-04-04
AU2503584A (en) 1984-09-06
KR840007733A (ko) 1984-12-10
AU561861B2 (en) 1987-05-21
IL71032A0 (en) 1984-05-31
PT78141A (en) 1984-03-01
FI840780A0 (fi) 1984-02-27
GB2135670B (en) 1987-07-08
DK98184A (da) 1984-08-29
NZ207259A (en) 1987-02-20
PL246417A1 (en) 1985-03-12
EP0124216A1 (en) 1984-11-07
GR79821B (hu) 1984-10-31
ES8602742A1 (es) 1985-12-01
DE3474831D1 (en) 1988-12-01
KR860001282B1 (ko) 1986-09-05

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