IL71032A0 - C-20 and c-23-modified macrolide derivatives - Google Patents

C-20 and c-23-modified macrolide derivatives

Info

Publication number
IL71032A0
IL71032A0 IL71032A IL7103284A IL71032A0 IL 71032 A0 IL71032 A0 IL 71032A0 IL 71032 A IL71032 A IL 71032A IL 7103284 A IL7103284 A IL 7103284A IL 71032 A0 IL71032 A0 IL 71032A0
Authority
IL
Israel
Prior art keywords
macrolide derivatives
modified macrolide
modified
derivatives
macrolide
Prior art date
Application number
IL71032A
Other languages
English (en)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/470,890 external-priority patent/US4468511A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of IL71032A0 publication Critical patent/IL71032A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
IL71032A 1983-02-28 1984-02-21 C-20 and c-23-modified macrolide derivatives IL71032A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US47083383A 1983-02-28 1983-02-28
US06/470,890 US4468511A (en) 1983-02-28 1983-02-28 C-20- And C-23-Modified macrolide derivatives

Publications (1)

Publication Number Publication Date
IL71032A0 true IL71032A0 (en) 1984-05-31

Family

ID=27043239

Family Applications (1)

Application Number Title Priority Date Filing Date
IL71032A IL71032A0 (en) 1983-02-28 1984-02-21 C-20 and c-23-modified macrolide derivatives

Country Status (14)

Country Link
EP (1) EP0124216B1 (hu)
KR (1) KR860001282B1 (hu)
AU (1) AU561861B2 (hu)
DE (1) DE3474831D1 (hu)
DK (1) DK98184A (hu)
ES (1) ES530081A0 (hu)
FI (1) FI840780A (hu)
GB (1) GB2135670B (hu)
GR (1) GR79821B (hu)
HU (1) HUT35693A (hu)
IL (1) IL71032A0 (hu)
NZ (1) NZ207259A (hu)
PL (1) PL246417A1 (hu)
PT (1) PT78141A (hu)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4515941A (en) * 1982-04-07 1985-05-07 Toyo Jozo Kabushiki Kaisha 23-Demycinosyldesmycosin derivatives
US4604380A (en) * 1985-01-18 1986-08-05 Eli Lilly And Company C-23-substituted mycaminosyltylonolide compounds, pharmaceutical compositions and methods of use
FR2646081A1 (hu) * 1989-04-20 1990-10-26 Adir
DE69309259T2 (de) * 1992-01-14 1997-07-17 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai, Tokio/Tokyo 3,4'-didesoxymycaminosyltylonolid-derivate und herstellung davon
TW226373B (hu) * 1992-07-15 1994-07-11 Pfizer
US5677287A (en) * 1993-03-18 1997-10-14 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at C-20
WO1995002594A1 (en) * 1993-07-15 1995-01-26 Pfizer Inc. Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
CA2391834C (en) * 1999-08-30 2008-08-05 Toshiaki Miyake Macrolide antibiotics and treatment of pasteurellosis
CN102875622B (zh) * 2006-07-28 2016-12-07 英特威国际有限公司 大环内酯合成方法
JP5323696B2 (ja) * 2006-07-28 2013-10-23 インターベツト・インターナシヨナル・ベー・ベー マクロライド合成方法
AU2014270353B2 (en) 2013-05-23 2018-09-20 Elanco Animal Health Gmbh Tylosin derivatives and method for preparation thereof
CN108299531B (zh) * 2018-01-23 2021-02-05 郑州大学 甲哌泰万菌素可药用盐及其制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8004922A (nl) * 1979-09-19 1981-03-23 Toyo Jozo Kk Deformyltylosinederivaten.
US4321361A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company Demycinosyltylosin and process for its production
ZA813578B (en) * 1980-06-12 1983-01-26 Lilly Co Eli Macrolide antibiotics
US4304856A (en) * 1980-11-10 1981-12-08 Eli Lilly And Company Process for producing 20-dihydro-20-deoxy-23-demycinosyltylosin
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin

Also Published As

Publication number Publication date
KR860001282B1 (ko) 1986-09-05
EP0124216B1 (en) 1988-10-26
ES8602742A1 (es) 1985-12-01
HUT35693A (en) 1985-07-29
GB8405086D0 (en) 1984-04-04
DK98184D0 (da) 1984-02-24
AU561861B2 (en) 1987-05-21
NZ207259A (en) 1987-02-20
FI840780A (fi) 1984-08-29
GR79821B (hu) 1984-10-31
FI840780A0 (fi) 1984-02-27
GB2135670B (en) 1987-07-08
KR840007733A (ko) 1984-12-10
PT78141A (en) 1984-03-01
EP0124216A1 (en) 1984-11-07
PL246417A1 (en) 1985-03-12
ES530081A0 (es) 1985-12-01
DE3474831D1 (en) 1988-12-01
AU2503584A (en) 1984-09-06
DK98184A (da) 1984-08-29
GB2135670A (en) 1984-09-05

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