NO974405D0 - Fremgangsmåte for fremstilling av 2-substituerte benzo(b)-tiofenforbindelser og mellomprodukter - Google Patents

Fremgangsmåte for fremstilling av 2-substituerte benzo(b)-tiofenforbindelser og mellomprodukter

Info

Publication number
NO974405D0
NO974405D0 NO974405A NO974405A NO974405D0 NO 974405 D0 NO974405 D0 NO 974405D0 NO 974405 A NO974405 A NO 974405A NO 974405 A NO974405 A NO 974405A NO 974405 D0 NO974405 D0 NO 974405D0
Authority
NO
Norway
Prior art keywords
intermediates
preparation
substituted benzo
thiophene compounds
thiophene
Prior art date
Application number
NO974405A
Other languages
English (en)
Norwegian (no)
Other versions
NO974405L (no
Inventor
Kenneth L Hauser
Alan D Palkowitz
Daniel Jon Sall
Kenneth Jeff Thrasher
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of NO974405L publication Critical patent/NO974405L/no
Publication of NO974405D0 publication Critical patent/NO974405D0/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56Radicals substituted by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO974405A 1995-03-31 1997-09-23 Fremgangsmåte for fremstilling av 2-substituerte benzo(b)-tiofenforbindelser og mellomprodukter NO974405D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/415,014 US5614639A (en) 1995-03-31 1995-03-31 Process for preparing 2-substituted benzo[b]thiophene compounds and intermediates thereof
PCT/US1996/004417 WO1996030361A1 (en) 1995-03-31 1996-03-28 PROCESS FOR 2-SUBSTITUTED BENZO[b]THIOPHENE COMPOUNDS AND INTERMEDIATES THEREOF

Publications (2)

Publication Number Publication Date
NO974405L NO974405L (no) 1997-09-23
NO974405D0 true NO974405D0 (no) 1997-09-23

Family

ID=23644002

Family Applications (1)

Application Number Title Priority Date Filing Date
NO974405A NO974405D0 (no) 1995-03-31 1997-09-23 Fremgangsmåte for fremstilling av 2-substituerte benzo(b)-tiofenforbindelser og mellomprodukter

Country Status (17)

Country Link
US (3) US5614639A (de)
EP (1) EP0739890A3 (de)
JP (1) JPH11502855A (de)
KR (1) KR19980703381A (de)
CN (2) CN1073107C (de)
AU (1) AU699368B2 (de)
BR (1) BR9607934A (de)
CA (1) CA2216100C (de)
CZ (1) CZ301697A3 (de)
HU (1) HUP9801253A3 (de)
NO (1) NO974405D0 (de)
NZ (1) NZ305287A (de)
PL (1) PL322495A1 (de)
RU (1) RU2147582C1 (de)
TR (1) TR199701058T1 (de)
UA (1) UA46010C2 (de)
WO (1) WO1996030361A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2000500138A (ja) * 1995-11-07 2000-01-11 イーライ・リリー・アンド・カンパニー 耐性腫瘍の治療方法
EP0919552A4 (de) * 1996-07-24 1999-09-15 Teikoku Hormone Mfg Co Ltd Verfahren zur herstellung von 2,6-disubstituierten benzothiophenverbindungen
ZA9710262B (en) * 1996-11-19 1999-05-13 Lilly Co Eli Process for the synthesis of benzothiophenes
EP1175433B1 (de) 1999-05-04 2005-08-03 Strakan International Limited Androgen glykoside und die androgenische aktivität davon
EP2266590A3 (de) 2002-02-22 2011-04-20 Shire LLC Wirkstoff-Abgabesystem und Verfahren zum Schutz und zur Verabreichung von Wirkstoffen
MX2015016743A (es) * 2013-06-06 2016-03-21 Astellas Pharma Inc Compuesto de benzotiofeno.
CN105753836A (zh) * 2016-02-03 2016-07-13 上海天慈生物谷生物工程有限公司 一种预防骨质疏松症药物的制备方法
CN115073420A (zh) * 2022-04-27 2022-09-20 陕西维世诺新材料有限公司 一种2-苯基苯并噻吩衍生物的制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4133814A (en) * 1975-10-28 1979-01-09 Eli Lilly And Company 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents
US4358593A (en) * 1981-04-03 1982-11-09 Eli Lilly And Company Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes
US4380635A (en) * 1981-04-03 1983-04-19 Eli Lilly And Company Synthesis of acylated benzothiophenes
US4418068A (en) * 1981-04-03 1983-11-29 Eli Lilly And Company Antiestrogenic and antiandrugenic benzothiophenes
US5436259A (en) * 1991-05-10 1995-07-25 Merck & Co., Inc. Substituted 1,2,4-triazolin-3-one compounds bearing acidic functional groups as balanced angiotensin II antagonists
JP3157882B2 (ja) * 1991-11-15 2001-04-16 帝国臓器製薬株式会社 新規なベンゾチオフエン誘導体
ATE198195T1 (de) * 1992-06-09 2001-01-15 Aventis Res & Tech Gmbh & Co 3-fluorpyridine, verfahren zu ihrer herstellung und ihre verwendung in flüssigkristallmischungen
US5254776A (en) * 1992-07-17 1993-10-19 Mallinckrodt Specialty Chemicals Company Synthesis of bromobiphenyls

Also Published As

Publication number Publication date
CA2216100C (en) 2002-01-08
US5710285A (en) 1998-01-20
TR199701058T1 (xx) 1998-02-21
KR19980703381A (ko) 1998-10-15
CA2216100A1 (en) 1996-10-03
EP0739890A2 (de) 1996-10-30
JPH11502855A (ja) 1999-03-09
AU5326196A (en) 1996-10-16
NO974405L (no) 1997-09-23
NZ305287A (en) 1998-04-27
US5712390A (en) 1998-01-27
HUP9801253A2 (hu) 1999-09-28
US5614639A (en) 1997-03-25
CN1335314A (zh) 2002-02-13
AU699368B2 (en) 1998-12-03
RU2147582C1 (ru) 2000-04-20
HUP9801253A3 (en) 2001-02-28
BR9607934A (pt) 1998-06-02
CN1073107C (zh) 2001-10-17
EP0739890A3 (de) 1997-04-09
CN1180353A (zh) 1998-04-29
CZ301697A3 (cs) 1998-01-14
UA46010C2 (uk) 2002-05-15
WO1996030361A1 (en) 1996-10-03
PL322495A1 (en) 1998-02-02

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