NO970079L - Pyrido£3,2,1-i,j|£3,1|benzoksazinderivater - Google Patents
Pyrido£3,2,1-i,j|£3,1|benzoksazinderivaterInfo
- Publication number
- NO970079L NO970079L NO970079A NO970079A NO970079L NO 970079 L NO970079 L NO 970079L NO 970079 A NO970079 A NO 970079A NO 970079 A NO970079 A NO 970079A NO 970079 L NO970079 L NO 970079L
- Authority
- NO
- Norway
- Prior art keywords
- pct
- formula
- compounds
- pyrido
- date jan
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C17/00—Preparation of halogenated hydrocarbons
- C07C17/093—Preparation of halogenated hydrocarbons by replacement by halogens
- C07C17/16—Preparation of halogenated hydrocarbons by replacement by halogens of hydroxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Paper (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
- Seasonings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Det er beskrevet nye pyrldo[3,2,1-1,J][3,Ijbenzoksa- zlnderivater av formel (I) hvori R^ er hytirogen eller Ci-C4-alkyl eventuelt substituert med hydroksy eller halogen; r2 g^ hydrogen eller metyl uavhengig av r1; r3 er hydrogen eller Ci-C4-alkyl; r3 ' er hydrogen eller irietyl ; R'* er hydrogen, alkyl med 1 til 4 karbonatomer, eventuelt substituert med hydroksy, metoksy, amino, metylamino eller dlmetylamino eller (5-metyl-2-okso- 1,3-dloksol-4-yl)-metyl; X^ er hydrogen eller halogen; Z er rester av strukturene ((a), (b), (c)) hvori r'' er hydrogen, hydroksy, -NR^OrII, hydroksymetyl eller -CH2- KrI r11 , karboksyl, metoksykarbonyl eller etoksykar- bonyl , hvor R^O er hydrogen, eventuelt hydroksy substituert C;^-C3-alkyl , alkoksykarbonyl med 1 til 4 karbonatomer i alkoksydelen eller C^-Cs-acyl, og R^l er hydrogen eller metyl; r8 er hydrogen, rettkjedet eller forgrenet C^-Cs-alkyl eller cyklopropyl; R*^ er hydrogen eller metyl; R° er hydrogen eller metyl; R^ er hydrogen, metyl eller rester av strukturene -CH=CH- COaR^', -CH2-CH2CO2R5', -CH2-CO-CH3, -CH2-CH2-CN; rS* er metyl eller etyl, og B er -CH2-, 0 eller en direktebinding. Det er videre beskrevet fremstilling av forbindelsene og deres anvendelse for behandling og forebyggelse av bakterielle infeksjoner.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4424369A DE4424369A1 (de) | 1994-07-11 | 1994-07-11 | Pyrido[3,2,1.i,j][3,1]benzoxazinderivate |
| PCT/EP1995/002510 WO1996001829A1 (de) | 1994-07-11 | 1995-06-28 | PYRIDO[3,2,1-i,j][3,1]BENZOXAZINDERIVATE |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO970079L true NO970079L (no) | 1997-01-09 |
| NO970079D0 NO970079D0 (no) | 1997-01-09 |
Family
ID=6522819
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO970079A NO970079D0 (no) | 1994-07-11 | 1997-01-09 | Pyrido£3,2,1-i,j|£3,1|benzoksazinderivater |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US5854241A (no) |
| EP (1) | EP0770083B1 (no) |
| JP (1) | JPH10502377A (no) |
| KR (1) | KR100372978B1 (no) |
| CN (1) | CN1086706C (no) |
| AT (1) | ATE195941T1 (no) |
| AU (1) | AU684651B2 (no) |
| BR (1) | BR9508384A (no) |
| CA (1) | CA2194694A1 (no) |
| CZ (1) | CZ5697A3 (no) |
| DE (2) | DE4424369A1 (no) |
| DK (1) | DK0770083T3 (no) |
| ES (1) | ES2150576T3 (no) |
| FI (1) | FI970092A (no) |
| HU (1) | HUT77138A (no) |
| IL (1) | IL114499A0 (no) |
| MX (1) | MX9700306A (no) |
| NO (1) | NO970079D0 (no) |
| NZ (1) | NZ289419A (no) |
| PL (1) | PL318097A1 (no) |
| SK (1) | SK2797A3 (no) |
| TW (1) | TW319766B (no) |
| WO (1) | WO1996001829A1 (no) |
| ZA (1) | ZA955707B (no) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6716830B2 (en) | 1998-09-30 | 2004-04-06 | Alcon, Inc. | Ophthalmic antibiotic compositions containing moxifloxacin |
| AR020661A1 (es) * | 1998-09-30 | 2002-05-22 | Alcon Lab Inc | Una composicion farmaceutica topica oftalmica, otica o nasal y el uso de la misma para la manufactura de un medicamento |
| US6395746B1 (en) | 1998-09-30 | 2002-05-28 | Alcon Manufacturing, Ltd. | Methods of treating ophthalmic, otic and nasal infections and attendant inflammation |
| US6509327B1 (en) | 1998-09-30 | 2003-01-21 | Alcon Manufacturing, Ltd. | Compositions and methods for treating otic, ophthalmic and nasal infections |
| CN1332962C (zh) * | 2005-07-12 | 2007-08-22 | 武汉人福药业有限责任公司 | 一种合成甲磺酸帕珠沙星中间体的方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3055894A (en) * | 1960-03-09 | 1962-09-25 | Pfizer & Co C | New heterocyclic amides |
| US3551565A (en) * | 1968-04-26 | 1970-12-29 | Geigy Chem Corp | Pharmaceutical compositions and uses of oxazinoisoquinoline derivatives |
| US3966743A (en) * | 1968-07-23 | 1976-06-29 | Boehringer Mannheim G.M.B.H. | Ortho fused cycloalkano-4-quinolone-3-carboxylic acid derivatives |
| US3984548A (en) * | 1974-02-11 | 1976-10-05 | Riker Laboratories, Inc. | Substituted pyrido[1,2,3,-de]-1,4-benzoxazines as bactericides |
| US3883522A (en) * | 1974-02-11 | 1975-05-13 | Riker Laboratories Inc | Substituted pyrido(1,2,3-de)-1,4-benzoxazines |
| JPS5746986A (en) * | 1980-09-02 | 1982-03-17 | Dai Ichi Seiyaku Co Ltd | Pyrido(1,2,3-de)(1,4)benzoxazine derivative |
| FR2593810B1 (fr) * | 1986-01-24 | 1988-04-22 | Sanofi Sa | Derives de la quinoleine, leur procede de preparation, leur application a titre de medicaments et les compositions les renfermant |
| JPH02157282A (ja) * | 1988-12-12 | 1990-06-18 | Wakunaga Pharmaceut Co Ltd | 新規ピリドベンゾオキサジン誘導体 |
| GB2236751B (en) * | 1989-10-14 | 1993-04-28 | Wyeth John & Brother Ltd | Heterocyclic compounds |
| TW222276B (no) * | 1992-01-27 | 1994-04-11 | Fujisawa Pharmaceutical Co |
-
1994
- 1994-07-11 DE DE4424369A patent/DE4424369A1/de not_active Withdrawn
-
1995
- 1995-06-28 EP EP95924949A patent/EP0770083B1/de not_active Expired - Lifetime
- 1995-06-28 ES ES95924949T patent/ES2150576T3/es not_active Expired - Lifetime
- 1995-06-28 KR KR1019970700058A patent/KR100372978B1/ko not_active IP Right Cessation
- 1995-06-28 AU AU29256/95A patent/AU684651B2/en not_active Ceased
- 1995-06-28 NZ NZ289419A patent/NZ289419A/en unknown
- 1995-06-28 AT AT95924949T patent/ATE195941T1/de not_active IP Right Cessation
- 1995-06-28 HU HU9700075A patent/HUT77138A/hu unknown
- 1995-06-28 BR BR9508384A patent/BR9508384A/pt not_active IP Right Cessation
- 1995-06-28 PL PL95318097A patent/PL318097A1/xx unknown
- 1995-06-28 DE DE59508689T patent/DE59508689D1/de not_active Expired - Fee Related
- 1995-06-28 US US08/765,212 patent/US5854241A/en not_active Expired - Fee Related
- 1995-06-28 MX MX9700306A patent/MX9700306A/es unknown
- 1995-06-28 SK SK27-97A patent/SK2797A3/sk unknown
- 1995-06-28 CZ CZ9756A patent/CZ5697A3/cs unknown
- 1995-06-28 JP JP8504083A patent/JPH10502377A/ja active Pending
- 1995-06-28 CN CN95194072A patent/CN1086706C/zh not_active Expired - Fee Related
- 1995-06-28 DK DK95924949T patent/DK0770083T3/da active
- 1995-06-28 WO PCT/EP1995/002510 patent/WO1996001829A1/de active IP Right Grant
- 1995-06-28 CA CA002194694A patent/CA2194694A1/en not_active Abandoned
- 1995-06-30 TW TW084106729A patent/TW319766B/zh active
- 1995-07-07 IL IL11449995A patent/IL114499A0/xx unknown
- 1995-07-10 ZA ZA955707A patent/ZA955707B/xx unknown
-
1997
- 1997-01-09 NO NO970079A patent/NO970079D0/no unknown
- 1997-01-09 FI FI970092A patent/FI970092A/fi unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI970092A0 (fi) | 1997-01-09 |
| PL318097A1 (en) | 1997-05-12 |
| DE59508689D1 (de) | 2000-10-05 |
| WO1996001829A1 (de) | 1996-01-25 |
| DK0770083T3 (da) | 2000-10-16 |
| US5854241A (en) | 1998-12-29 |
| TW319766B (no) | 1997-11-11 |
| EP0770083B1 (de) | 2000-08-30 |
| MX9700306A (es) | 1997-05-31 |
| ZA955707B (en) | 1996-02-21 |
| HU9700075D0 (en) | 1997-02-28 |
| EP0770083A1 (de) | 1997-05-02 |
| BR9508384A (pt) | 1997-12-23 |
| SK2797A3 (en) | 1997-07-09 |
| JPH10502377A (ja) | 1998-03-03 |
| ES2150576T3 (es) | 2000-12-01 |
| FI970092A (fi) | 1997-01-09 |
| NO970079D0 (no) | 1997-01-09 |
| NZ289419A (en) | 1998-09-24 |
| CN1086706C (zh) | 2002-06-26 |
| KR100372978B1 (ko) | 2003-06-12 |
| CZ5697A3 (en) | 1997-05-14 |
| IL114499A0 (en) | 1995-11-27 |
| CN1152921A (zh) | 1997-06-25 |
| CA2194694A1 (en) | 1996-01-25 |
| DE4424369A1 (de) | 1996-01-18 |
| HUT77138A (hu) | 1998-03-02 |
| AU684651B2 (en) | 1997-12-18 |
| AU2925695A (en) | 1996-02-09 |
| ATE195941T1 (de) | 2000-09-15 |
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