NO952891L - Forbedret fremgangsmåte for fremstilling av 3-(amino-etoksy-benzoyl)benzo[BÅtiofener - Google Patents
Forbedret fremgangsmåte for fremstilling av 3-(amino-etoksy-benzoyl)benzo[BÅtiofenerInfo
- Publication number
- NO952891L NO952891L NO952891A NO952891A NO952891L NO 952891 L NO952891 L NO 952891L NO 952891 A NO952891 A NO 952891A NO 952891 A NO952891 A NO 952891A NO 952891 L NO952891 L NO 952891L
- Authority
- NO
- Norway
- Prior art keywords
- benzo
- thiophenes
- benzoyl
- preparation
- boat
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/56—Radicals substituted by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Photoreceptors In Electrophotography (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27945694A | 1994-07-22 | 1994-07-22 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO952891D0 NO952891D0 (no) | 1995-07-20 |
| NO952891L true NO952891L (no) | 1996-01-23 |
Family
ID=23069049
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO952891A NO952891L (no) | 1994-07-22 | 1995-07-20 | Forbedret fremgangsmåte for fremstilling av 3-(amino-etoksy-benzoyl)benzo[BÅtiofener |
Country Status (27)
| Country | Link |
|---|---|
| US (2) | US5523416A (cs) |
| EP (1) | EP0693488B1 (cs) |
| JP (1) | JPH0853440A (cs) |
| KR (1) | KR960004336A (cs) |
| CN (1) | CN1116624A (cs) |
| AT (1) | ATE205842T1 (cs) |
| AU (1) | AU684181B2 (cs) |
| BR (1) | BR9503408A (cs) |
| CA (1) | CA2154319A1 (cs) |
| CO (1) | CO4410192A1 (cs) |
| CZ (1) | CZ189295A3 (cs) |
| DE (1) | DE69522762T2 (cs) |
| DK (1) | DK0693488T3 (cs) |
| ES (1) | ES2160668T3 (cs) |
| FI (1) | FI953513A7 (cs) |
| HU (1) | HUT71596A (cs) |
| IL (1) | IL114684A (cs) |
| MX (1) | MXPA99010090A (cs) |
| MY (1) | MY131787A (cs) |
| NO (1) | NO952891L (cs) |
| NZ (1) | NZ272609A (cs) |
| PE (1) | PE34396A1 (cs) |
| PL (1) | PL309694A1 (cs) |
| PT (1) | PT693488E (cs) |
| RU (1) | RU95113269A (cs) |
| TW (1) | TW298592B (cs) |
| ZA (1) | ZA956031B (cs) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CO4410190A1 (es) | 1994-09-19 | 1997-01-09 | Lilly Co Eli | 3-[4-(2-AMINOETOXI)-BENZOIL]-2-ARIL-6-HIDROXIBENZO [b] TIOFENO CRISTALINO |
| PE2699A1 (es) * | 1996-09-25 | 1999-02-04 | Lilly Co Eli | Procedimiento para la sintesis de benzotiofenos |
| ZA9710262B (en) * | 1996-11-19 | 1999-05-13 | Lilly Co Eli | Process for the synthesis of benzothiophenes |
| HUP0003187A3 (en) * | 1997-04-30 | 2002-04-29 | Lilly Co Eli | Substituted benzothiophenes and process for preparing them |
| US6921827B2 (en) * | 2000-11-27 | 2005-07-26 | Eli Lilly And Company | Process for preparing 3-aryl-benzo{b} thiophenes |
| EP1826205A1 (en) | 2002-09-30 | 2007-08-29 | A/S GEA Farmaceutisk Fabrik | Novel raloxifene succinic acid addition salts and/or solvates thereof, and pharmaceutical compositions comprising these |
| ITMI20031333A1 (it) * | 2003-06-30 | 2005-01-01 | Erregierre Spa | Processo di preparazione di raloxifene cloridrato. |
| GB2456096B (en) * | 2006-10-17 | 2011-08-17 | Cipla Ltd | Crystalline form of benzothiophene compound and process for preparation thereof |
| CN101812002A (zh) * | 2010-04-16 | 2010-08-25 | 山东新华制药股份有限公司 | 4-甲氧基-α-[(3-甲氧基苯基)硫代]苯乙酮的合成工艺 |
| CN104496963A (zh) * | 2014-12-02 | 2015-04-08 | 千辉药业（安徽）有限责任公司 | 一种盐酸雷洛昔芬的制备方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4133814A (en) * | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
| AU509682B2 (en) * | 1975-10-28 | 1980-05-22 | Eli Lilly And Company | 2-Aroyl-3-Phenylbenzothiophene Derivatives |
| AT364852B (de) * | 1977-11-05 | 1981-11-25 | Thomae Gmbh Dr K | Verfahren zur herstellung von kondensierten isothiazol-3(2h)-on-1,1-dioxiden und von deren salzen |
| US4436748A (en) * | 1980-10-20 | 1984-03-13 | Hoechst-Roussel Pharmaceuticals Inc. | Benzo[b]thiophenes |
| US4380635A (en) * | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
| IL65379A0 (en) * | 1981-04-03 | 1982-05-31 | Lilly Co Eli | Process for preparing acylated benzothiophenes |
| IL65378A (en) * | 1981-04-03 | 1986-02-28 | Lilly Co Eli | Process for preparing 3-(4-aminoethoxybenzoyl)benzo-(b)thiophenes |
| US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
| GB2097788B (en) * | 1981-04-03 | 1985-04-24 | Lilly Co Eli | Benzothiophene compounds and process for preparing them |
| US4436740A (en) * | 1982-07-26 | 1984-03-13 | Merck & Co., Inc. | 3-Cycloalkylamino-2-OR-propoxycyanopyridines |
| DE4204969A1 (de) * | 1992-02-19 | 1993-08-26 | Basf Ag | Verfahren zur herstellung von benzo(b)thiophenen |
| US5298630A (en) * | 1992-06-03 | 1994-03-29 | Sumitomo Seika Chemicals Co., Ltd. | Processes for producing 2-substituted benzo[B]thiophene |
| JP3337728B2 (ja) * | 1992-11-20 | 2002-10-21 | イハラケミカル工業株式会社 | ２‐アセチルベンゾ［ｂ］チオフェンの製造方法 |
| US5426191A (en) * | 1993-12-03 | 1995-06-20 | Warner-Lambert Company | Process for the synthesis of 3-chlorobenzo[b]thiophene-2-carbonyl chlorides |
-
1995
- 1995-04-14 US US08/422,294 patent/US5523416A/en not_active Expired - Lifetime
- 1995-07-19 CO CO95031972A patent/CO4410192A1/es unknown
- 1995-07-19 NZ NZ272609A patent/NZ272609A/en unknown
- 1995-07-19 ZA ZA956031A patent/ZA956031B/xx unknown
- 1995-07-19 HU HU9502176A patent/HUT71596A/hu unknown
- 1995-07-19 AU AU25068/95A patent/AU684181B2/en not_active Expired - Fee Related
- 1995-07-19 MY MYPI95002052A patent/MY131787A/en unknown
- 1995-07-19 PE PE1995274176A patent/PE34396A1/es not_active Application Discontinuation
- 1995-07-19 KR KR1019950021163A patent/KR960004336A/ko not_active Ceased
- 1995-07-19 TW TW084107456A patent/TW298592B/zh active
- 1995-07-19 PL PL95309694A patent/PL309694A1/xx unknown
- 1995-07-20 CA CA002154319A patent/CA2154319A1/en not_active Abandoned
- 1995-07-20 CN CN95109618A patent/CN1116624A/zh active Pending
- 1995-07-20 PT PT95305085T patent/PT693488E/pt unknown
- 1995-07-20 JP JP7183923A patent/JPH0853440A/ja not_active Withdrawn
- 1995-07-20 AT AT95305085T patent/ATE205842T1/de not_active IP Right Cessation
- 1995-07-20 FI FI953513A patent/FI953513A7/fi unknown
- 1995-07-20 DE DE69522762T patent/DE69522762T2/de not_active Expired - Fee Related
- 1995-07-20 IL IL11468495A patent/IL114684A/xx active IP Right Grant
- 1995-07-20 ES ES95305085T patent/ES2160668T3/es not_active Expired - Lifetime
- 1995-07-20 NO NO952891A patent/NO952891L/no unknown
- 1995-07-20 EP EP95305085A patent/EP0693488B1/en not_active Expired - Lifetime
- 1995-07-20 DK DK95305085T patent/DK0693488T3/da active
- 1995-07-20 RU RU95113269/04A patent/RU95113269A/ru unknown
- 1995-07-20 CZ CZ951892A patent/CZ189295A3/cs unknown
- 1995-07-21 BR BR9503408A patent/BR9503408A/pt not_active Application Discontinuation
- 1995-08-08 US US08/512,724 patent/US5512684A/en not_active Expired - Lifetime
-
1999
- 1999-11-03 MX MXPA99010090A patent/MXPA99010090A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| HUT71596A (en) | 1996-01-29 |
| NO952891D0 (no) | 1995-07-20 |
| EP0693488B1 (en) | 2001-09-19 |
| CN1116624A (zh) | 1996-02-14 |
| IL114684A0 (en) | 1995-11-27 |
| RU95113269A (ru) | 1997-06-10 |
| FI953513L (fi) | 1996-01-23 |
| NZ272609A (en) | 1997-05-26 |
| CZ189295A3 (en) | 1996-02-14 |
| PE34396A1 (es) | 1996-09-26 |
| CO4410192A1 (es) | 1997-01-09 |
| MXPA99010090A (es) | 2004-09-01 |
| PL309694A1 (en) | 1996-02-05 |
| ES2160668T3 (es) | 2001-11-16 |
| US5523416A (en) | 1996-06-04 |
| US5512684A (en) | 1996-04-30 |
| CA2154319A1 (en) | 1996-01-23 |
| FI953513A7 (fi) | 1996-01-23 |
| HU9502176D0 (en) | 1995-09-28 |
| EP0693488A1 (en) | 1996-01-24 |
| AU684181B2 (en) | 1997-12-04 |
| FI953513A0 (fi) | 1995-07-20 |
| AU2506895A (en) | 1996-02-01 |
| JPH0853440A (ja) | 1996-02-27 |
| DE69522762D1 (de) | 2001-10-25 |
| DE69522762T2 (de) | 2002-07-04 |
| BR9503408A (pt) | 1996-02-27 |
| KR960004336A (ko) | 1996-02-23 |
| TW298592B (cs) | 1997-02-21 |
| MY131787A (en) | 2007-08-30 |
| DK0693488T3 (da) | 2001-11-12 |
| IL114684A (en) | 1999-06-20 |
| PT693488E (pt) | 2002-02-28 |
| ATE205842T1 (de) | 2001-10-15 |
| ZA956031B (en) | 1997-01-20 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO952891L (no) | Forbedret fremgangsmåte for fremstilling av 3-(amino-etoksy-benzoyl)benzo[BÅtiofener | |
| SE9503213L (sv) | Syntes av 3-4-(2-aminoetoxi)bensoyl -2aryl-4-hydroxi-benso(b)tiofener | |
| Carpenter et al. | The scope and limitations of carboxamide-induced. beta.-directed metalation of 2-substituted furan, thiophene, and 1-methylpyrrole derivatives. Application of the method to syntheses of 2, 3-disubstituted thiophenes and furans | |
| MY112481A (en) | Synthesis of 3-[4-(2-aminoethoxy)-benzoyl] -2-aryl-6-hydroxybenzo [b] thiophenes | |
| IS5300A (is) | Aðferð til framleiðslu á sítalóprami | |
| GR1004074B (el) | Μεθοδος παρασκευης της σιταλοπραμης. | |
| DE69029197D1 (de) | Gamma-retinoinsäure-rezeptor | |
| NO174345C (no) | Analogifremgangsmåte for fremstilling av terapeutisk aktive indol-, benzofuran- og benzotiofenderivater | |
| US4024156A (en) | Thiophene ethanolamines | |
| Kuneš et al. | Synthesis and antifungal activity evaluation of 3-hetaryl-2, 5-dihydrofuran-2-ones. An unusual fragmentation of the oxazole ring via 2, 3-selenoxide shift | |
| DE3768255D1 (de) | Als kompensator wirkender, rohrfoermiger faltenbalg. | |
| Campaigne et al. | Benzo [b] thiophene derivatives. VIII. Benzo [b] thiophene‐3‐earboxaldehyde and derivatives | |
| NO975579D0 (no) | Fremgangsmåte for syntese av benzo£b|tiofener | |
| AU510569B2 (en) | Polymorphic "B" of 4-(2-thenoyl)-2, 3-dichlorophenoxy acetic acid | |
| Goldoni et al. | Synthesis and NMR characterization of 3, 4′‐dibutoxy‐2, 2′‐bithiophene | |
| Kosugi et al. | Cyclisation of polyenic β-keto suiphoxides. A novel route to optically active intermediates for cyclic terpenoid synthesis | |
| Kusuhara et al. | A facile synthesis of β-(4-azuleno [1, 2-b] thienyl) α, β-unsaturated ketones | |
| JPS5353681A (en) | Preparation of debenzazepin derivatives | |
| WO1998052913A3 (de) | Leukotrien-b4-antagonisten, insbesondere 3-oxa-tetrahydronaphthalin -ltb4-antagonisten | |
| Špirková et al. | Preparation and stereochemistry of pentadiene derivatives of furan | |
| JPS51131896A (en) | A process for preparing hexahydro-1h- pyrid(4,3-b)indoles | |
| ES471171A1 (es) | Un procedimiento para la obtencion de la 2-benzo(b)tienil- 1,4-dimetil-1,2,3,6-tetrahidro-2-piridil-cetona | |
| FI851140A7 (fi) | Terapeuttisesti arvokkaiden bentso/b/ tiofeenien valmistuksessa välituotteina käyttökelpoisia 2,3-dihydrobentso/b/tiofeenejä. | |
| ES459895A1 (es) | Un procedimiento para la produccion de acido 6-11-dihidrodi-benzo (b.e) tiepin-11-on-3-acetico. |