EA199800026A1 - Способ получения производных винилсульфеновых кислот - Google Patents

Способ получения производных винилсульфеновых кислот

Info

Publication number
EA199800026A1
EA199800026A1 EA199800026A EA199800026A EA199800026A1 EA 199800026 A1 EA199800026 A1 EA 199800026A1 EA 199800026 A EA199800026 A EA 199800026A EA 199800026 A EA199800026 A EA 199800026A EA 199800026 A1 EA199800026 A1 EA 199800026A1
Authority
EA
Eurasian Patent Office
Prior art keywords
acid derivatives
obtaining vinyl
sulphenic acid
obtaining
thiophenes
Prior art date
Application number
EA199800026A
Other languages
English (en)
Other versions
EA000606B1 (ru
Inventor
Дэвид В. Хоард
Уэйн Д. Льюк
Original Assignee
Эли Лилли Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/482,692 external-priority patent/US5512701A/en
Priority claimed from US08/483,607 external-priority patent/US5514826A/en
Application filed by Эли Лилли Энд Компани filed Critical Эли Лилли Энд Компани
Publication of EA199800026A1 publication Critical patent/EA199800026A1/ru
Publication of EA000606B1 publication Critical patent/EA000606B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/10—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C323/11—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/16—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C313/08—Sulfenic acids; Derivatives thereof
    • C07C313/18—Sulfenamides
    • C07C313/20—Sulfenamides having sulfur atoms of sulfenamide groups bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C321/00—Thiols, sulfides, hydropolysulfides or polysulfides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D223/08—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0834—Compounds having one or more O-Si linkage
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Изобретение относится к новым производным винилсульфеновых кислот и новому способу получения новых производных винилсульфеновых кислот. Эти соединения используются для синтеза бензо[b]тиофенов, в частности 2-арилбензо[b]тиофенов.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA199800026A 1995-06-07 1996-06-04 Производные винилсульфеновых кислот и способ их получения EA000606B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/482,692 US5512701A (en) 1995-06-07 1995-06-07 Process for the synthesis of vinyl sulfenic acid derivatives
US08/483,607 US5514826A (en) 1995-06-07 1995-06-07 Vinyl sulfenic acid derivatives
PCT/US1996/009460 WO1996040693A1 (en) 1995-06-07 1996-06-04 Process for the synthesis of vinyl sulfenic acid derivatives

Publications (2)

Publication Number Publication Date
EA199800026A1 true EA199800026A1 (ru) 1998-06-25
EA000606B1 EA000606B1 (ru) 1999-12-29

Family

ID=27047368

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199800026A EA000606B1 (ru) 1995-06-07 1996-06-04 Производные винилсульфеновых кислот и способ их получения

Country Status (16)

Country Link
EP (1) EP0830362A4 (ru)
JP (1) JPH11507346A (ru)
KR (1) KR19990022503A (ru)
CN (2) CN1068883C (ru)
AU (1) AU698076B2 (ru)
BR (1) BR9608847A (ru)
CA (1) CA2224225A1 (ru)
CZ (1) CZ387997A3 (ru)
EA (1) EA000606B1 (ru)
HU (1) HUP9900923A3 (ru)
IL (1) IL122127A (ru)
NO (1) NO975633L (ru)
NZ (1) NZ310241A (ru)
PL (1) PL323907A1 (ru)
TR (1) TR199701511T1 (ru)
WO (1) WO1996040693A1 (ru)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU697352B2 (en) * 1995-06-07 1998-10-01 Eli Lilly And Company Vinyl sulfoxides and a process for their synthesis
SG106558A1 (en) * 1995-06-07 2004-10-29 Lilly Co Eli Vinyl sulfoxides and a process for their synthesis
EP1832583A1 (en) 2002-09-30 2007-09-12 A/S GEA Farmaceutisk Fabrik Novel raloxifene sulphuric acid addition salts and/or solvates thereof, and pharmaceutical compositions comprising these

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4380635A (en) * 1981-04-03 1983-04-19 Eli Lilly And Company Synthesis of acylated benzothiophenes
IL65379A0 (en) * 1981-04-03 1982-05-31 Lilly Co Eli Process for preparing acylated benzothiophenes
DE3543567A1 (de) * 1985-12-10 1987-06-11 Degussa Verfahren zur herstellung von sulfensaeurechloriden und sulfensaeureestern

Also Published As

Publication number Publication date
EP0830362A1 (en) 1998-03-25
CZ387997A3 (cs) 1998-09-16
JPH11507346A (ja) 1999-06-29
AU698076B2 (en) 1998-10-22
NO975633D0 (no) 1997-12-04
AU6100396A (en) 1996-12-30
CA2224225A1 (en) 1996-12-19
EP0830362A4 (en) 1998-09-02
WO1996040693A1 (en) 1996-12-19
HUP9900923A2 (hu) 1999-07-28
PL323907A1 (en) 1998-04-27
IL122127A0 (en) 1998-04-05
TR199701511T1 (xx) 1998-04-21
CN1068883C (zh) 2001-07-25
NO975633L (no) 1998-01-28
BR9608847A (pt) 1999-06-08
CN1192215A (zh) 1998-09-02
HUP9900923A3 (en) 2000-02-28
IL122127A (en) 2001-05-20
MX9709130A (es) 1998-03-31
CN1330071A (zh) 2002-01-09
EA000606B1 (ru) 1999-12-29
NZ310241A (en) 1999-07-29
KR19990022503A (ko) 1999-03-25

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM

MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): RU