NO912750L - Fremgangsmaate for fremstilling av terapeutisk aktive tiokso-heterocykliske forbindelser. - Google Patents

Fremgangsmaate for fremstilling av terapeutisk aktive tiokso-heterocykliske forbindelser.

Info

Publication number
NO912750L
NO912750L NO91912750A NO912750A NO912750L NO 912750 L NO912750 L NO 912750L NO 91912750 A NO91912750 A NO 91912750A NO 912750 A NO912750 A NO 912750A NO 912750 L NO912750 L NO 912750L
Authority
NO
Norway
Prior art keywords
tioxo
procedure
preparation
heterocyclic compounds
therapeutic active
Prior art date
Application number
NO91912750A
Other languages
English (en)
Norwegian (no)
Other versions
NO912750D0 (no
Inventor
Pierre Andre Raymond Bruneau
Original Assignee
Ici Pharma
Ici Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Pharma, Ici Plc filed Critical Ici Pharma
Publication of NO912750D0 publication Critical patent/NO912750D0/no
Publication of NO912750L publication Critical patent/NO912750L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D245/00Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Detergent Compositions (AREA)
NO91912750A 1990-07-13 1991-07-12 Fremgangsmaate for fremstilling av terapeutisk aktive tiokso-heterocykliske forbindelser. NO912750L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP90402034 1990-07-13
EP91400079 1991-01-15

Publications (2)

Publication Number Publication Date
NO912750D0 NO912750D0 (no) 1991-07-12
NO912750L true NO912750L (no) 1992-01-14

Family

ID=26127361

Family Applications (1)

Application Number Title Priority Date Filing Date
NO91912750A NO912750L (no) 1990-07-13 1991-07-12 Fremgangsmaate for fremstilling av terapeutisk aktive tiokso-heterocykliske forbindelser.

Country Status (22)

Country Link
US (1) US5240941A (cs)
EP (1) EP0466452B1 (cs)
JP (1) JPH04243877A (cs)
KR (1) KR920002561A (cs)
AT (1) ATE128133T1 (cs)
AU (1) AU638579B2 (cs)
CA (1) CA2046006A1 (cs)
CS (1) CS214891A3 (cs)
DE (1) DE69113148T2 (cs)
DK (1) DK0466452T3 (cs)
ES (1) ES2076472T3 (cs)
FI (1) FI913369A7 (cs)
GB (1) GB9113137D0 (cs)
GR (1) GR3017453T3 (cs)
HU (1) HUT61999A (cs)
IE (1) IE912138A1 (cs)
IL (1) IL98603A0 (cs)
MX (1) MX174406B (cs)
NO (1) NO912750L (cs)
NZ (1) NZ238703A (cs)
PT (1) PT98292A (cs)
TW (1) TW235918B (cs)

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WO1994029297A1 (en) * 1993-06-07 1994-12-22 Zeneca Limited 2-oxo-1,2,3,4-tetrahydroquinoline derivatives
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US5643933A (en) * 1995-06-02 1997-07-01 G. D. Searle & Co. Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors
US6677364B2 (en) * 1998-04-20 2004-01-13 G.D. Searle & Co. Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors
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US8158362B2 (en) 2005-03-30 2012-04-17 Decode Genetics Ehf. Methods of diagnosing susceptibility to myocardial infarction and screening for an LTA4H haplotype
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US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
WO2009088986A1 (en) 2008-01-04 2009-07-16 Intellikine, Inc. Certain chemical entities, compositions and methods
US8993580B2 (en) 2008-03-14 2015-03-31 Intellikine Llc Benzothiazole kinase inhibitors and methods of use
US8637542B2 (en) 2008-03-14 2014-01-28 Intellikine, Inc. Kinase inhibitors and methods of use
US20110224223A1 (en) 2008-07-08 2011-09-15 The Regents Of The University Of California, A California Corporation MTOR Modulators and Uses Thereof
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EP2751112B1 (en) 2011-09-02 2019-10-09 The Regents of The University of California Substituted pyrazolo[3,4-d]pyrimidines and uses thereof
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US9266892B2 (en) 2012-12-19 2016-02-23 Incyte Holdings Corporation Fused pyrazoles as FGFR inhibitors
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US11466004B2 (en) 2018-05-04 2022-10-11 Incyte Corporation Solid forms of an FGFR inhibitor and processes for preparing the same
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Also Published As

Publication number Publication date
GB9113137D0 (en) 1991-08-07
EP0466452A3 (en) 1992-08-19
NO912750D0 (no) 1991-07-12
IL98603A0 (en) 1992-07-15
NZ238703A (en) 1994-01-26
HUT61999A (en) 1993-03-29
TW235918B (cs) 1994-12-11
FI913369A0 (fi) 1991-07-11
KR920002561A (ko) 1992-02-28
AU7933791A (en) 1992-01-16
EP0466452A2 (en) 1992-01-15
ATE128133T1 (de) 1995-10-15
CS214891A3 (en) 1992-02-19
EP0466452B1 (en) 1995-09-20
MX174406B (es) 1994-05-13
JPH04243877A (ja) 1992-08-31
DK0466452T3 (da) 1996-01-02
US5240941A (en) 1993-08-31
IE912138A1 (en) 1992-01-15
PT98292A (pt) 1992-05-29
GR3017453T3 (en) 1995-12-31
CA2046006A1 (en) 1992-01-14
HU912295D0 (en) 1991-12-30
AU638579B2 (en) 1993-07-01
DE69113148T2 (de) 1996-03-28
ES2076472T3 (es) 1995-11-01
FI913369A7 (fi) 1992-01-14
DE69113148D1 (de) 1995-10-26

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