NO912750L - Fremgangsmaate for fremstilling av terapeutisk aktive tiokso-heterocykliske forbindelser. - Google Patents

Fremgangsmaate for fremstilling av terapeutisk aktive tiokso-heterocykliske forbindelser.

Info

Publication number
NO912750L
NO912750L NO91912750A NO912750A NO912750L NO 912750 L NO912750 L NO 912750L NO 91912750 A NO91912750 A NO 91912750A NO 912750 A NO912750 A NO 912750A NO 912750 L NO912750 L NO 912750L
Authority
NO
Norway
Prior art keywords
tioxo
procedure
preparation
heterocyclic compounds
therapeutic active
Prior art date
Application number
NO91912750A
Other languages
English (en)
Other versions
NO912750D0 (no
Inventor
Pierre Andre Raymond Bruneau
Original Assignee
Ici Pharma
Ici Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Pharma, Ici Plc filed Critical Ici Pharma
Publication of NO912750D0 publication Critical patent/NO912750D0/no
Publication of NO912750L publication Critical patent/NO912750L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D245/00—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Detergent Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Quinoline Compounds (AREA)
NO91912750A 1990-07-13 1991-07-12 Fremgangsmaate for fremstilling av terapeutisk aktive tiokso-heterocykliske forbindelser. NO912750L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP90402034 1990-07-13
EP91400079 1991-01-15

Publications (2)

Publication Number Publication Date
NO912750D0 NO912750D0 (no) 1991-07-12
NO912750L true NO912750L (no) 1992-01-14

Family

ID=26127361

Family Applications (1)

Application Number Title Priority Date Filing Date
NO91912750A NO912750L (no) 1990-07-13 1991-07-12 Fremgangsmaate for fremstilling av terapeutisk aktive tiokso-heterocykliske forbindelser.

Country Status (22)

Country Link
US (1) US5240941A (no)
EP (1) EP0466452B1 (no)
JP (1) JPH04243877A (no)
KR (1) KR920002561A (no)
AT (1) ATE128133T1 (no)
AU (1) AU638579B2 (no)
CA (1) CA2046006A1 (no)
CS (1) CS214891A3 (no)
DE (1) DE69113148T2 (no)
DK (1) DK0466452T3 (no)
ES (1) ES2076472T3 (no)
FI (1) FI913369A (no)
GB (1) GB9113137D0 (no)
GR (1) GR3017453T3 (no)
HU (1) HUT61999A (no)
IE (1) IE912138A1 (no)
IL (1) IL98603A0 (no)
MX (1) MX174406B (no)
NO (1) NO912750L (no)
NZ (1) NZ238703A (no)
PT (1) PT98292A (no)
TW (1) TW235918B (no)

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WO2006068760A2 (en) 2004-11-19 2006-06-29 The Regents Of The University Of California Anti-inflammatory pyrazolopyrimidines
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US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
ES2647163T3 (es) 2008-01-04 2017-12-19 Intellikine, Inc. Derivados de isoquinolinona sustituidos con una purina útiles como inhibidores de la PI3K
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US8993580B2 (en) 2008-03-14 2015-03-31 Intellikine Llc Benzothiazole kinase inhibitors and methods of use
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US9266892B2 (en) 2012-12-19 2016-02-23 Incyte Holdings Corporation Fused pyrazoles as FGFR inhibitors
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US11628162B2 (en) 2019-03-08 2023-04-18 Incyte Corporation Methods of treating cancer with an FGFR inhibitor
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Also Published As

Publication number Publication date
TW235918B (no) 1994-12-11
CS214891A3 (en) 1992-02-19
DK0466452T3 (da) 1996-01-02
ES2076472T3 (es) 1995-11-01
MX174406B (es) 1994-05-13
DE69113148D1 (de) 1995-10-26
IE912138A1 (en) 1992-01-15
NO912750D0 (no) 1991-07-12
GR3017453T3 (en) 1995-12-31
AU638579B2 (en) 1993-07-01
GB9113137D0 (en) 1991-08-07
DE69113148T2 (de) 1996-03-28
AU7933791A (en) 1992-01-16
EP0466452A2 (en) 1992-01-15
CA2046006A1 (en) 1992-01-14
US5240941A (en) 1993-08-31
JPH04243877A (ja) 1992-08-31
FI913369A0 (fi) 1991-07-11
HU912295D0 (en) 1991-12-30
KR920002561A (ko) 1992-02-28
EP0466452B1 (en) 1995-09-20
FI913369A (fi) 1992-01-14
PT98292A (pt) 1992-05-29
ATE128133T1 (de) 1995-10-15
NZ238703A (en) 1994-01-26
HUT61999A (en) 1993-03-29
EP0466452A3 (en) 1992-08-19
IL98603A0 (en) 1992-07-15

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