NO341326B1 - Farmasøytisk sammensetning av CETP-inhibitorer, deres anvendelse ved terapi, og for å øke HDL-kolesterol, samt deres anvendelse ved fremstilling av et medikament for å øke HDL-kolesterolet. - Google Patents
Farmasøytisk sammensetning av CETP-inhibitorer, deres anvendelse ved terapi, og for å øke HDL-kolesterol, samt deres anvendelse ved fremstilling av et medikament for å øke HDL-kolesterolet. Download PDFInfo
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- NO341326B1 NO341326B1 NO20083821A NO20083821A NO341326B1 NO 341326 B1 NO341326 B1 NO 341326B1 NO 20083821 A NO20083821 A NO 20083821A NO 20083821 A NO20083821 A NO 20083821A NO 341326 B1 NO341326 B1 NO 341326B1
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
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- Medicinal Preparation (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US77178206P | 2006-02-09 | 2006-02-09 | |
| PCT/US2007/003799 WO2007092642A2 (en) | 2006-02-09 | 2007-02-09 | Polymer formulations of cetp inhibitors |
Publications (2)
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| NO20083821L NO20083821L (no) | 2008-09-30 |
| NO341326B1 true NO341326B1 (no) | 2017-10-16 |
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| NO20083821A NO341326B1 (no) | 2006-02-09 | 2008-09-08 | Farmasøytisk sammensetning av CETP-inhibitorer, deres anvendelse ved terapi, og for å øke HDL-kolesterol, samt deres anvendelse ved fremstilling av et medikament for å øke HDL-kolesterolet. |
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| EP (1) | EP1983966B1 (https=) |
| JP (2) | JP5773560B2 (https=) |
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| CN (2) | CN103735515A (https=) |
| AU (1) | AU2007212197B2 (https=) |
| BR (1) | BRPI0707584A2 (https=) |
| CA (1) | CA2641451C (https=) |
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| NO (1) | NO341326B1 (https=) |
| NZ (1) | NZ569700A (https=) |
| RU (1) | RU2457841C2 (https=) |
| WO (1) | WO2007092642A2 (https=) |
| ZA (1) | ZA200805854B (https=) |
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| WO2004085996A2 (en) | 2003-03-20 | 2004-10-07 | Albert Einstein College Of Medicine Of Yeshiva University | Biomarkers for longevity and disease and uses thereof |
| US8604055B2 (en) | 2004-12-31 | 2013-12-10 | Dr. Reddy's Laboratories Ltd. | Substituted benzylamino quinolines as cholesterol ester-transfer protein inhibitors |
| WO2006073973A2 (en) * | 2004-12-31 | 2006-07-13 | Reddy Us Therapeutics, Inc. | Novel benzylamine derivatives as cetp inhibitors |
| AU2008313620A1 (en) * | 2007-10-19 | 2009-04-23 | Abbott Gmbh & Co. Kg | Solid dispersion product containing N-aryl urea-based compound |
| JP2011513242A (ja) | 2008-02-25 | 2011-04-28 | アミラ ファーマシューティカルズ，インク． | プロスタグランジンｄ２受容体アンタゴニスト |
| AR071375A1 (es) * | 2008-04-22 | 2010-06-16 | Solvay Pharm Gmbh | Formulaciones para ingredientes farmaceuticos activos de permeabilidad deficiente, proceso de preparacion y producto |
| AU2011332031B2 (en) | 2010-11-24 | 2017-01-12 | Melinta Subsidiary Corp. | Pharmaceutical compositions |
| ES2683350T3 (es) * | 2011-07-08 | 2018-09-26 | Novartis Ag | Método para tratar la aterosclerosis en sujetos con alto nivel de triglicéridos |
| US9199967B2 (en) | 2011-08-18 | 2015-12-01 | Dr. Reddy's Laboratories Ltd. | Substituted heterocyclic amine compounds as cholestryl ester-transfer protein (CETP) inhibitors |
| MX352074B (es) | 2011-09-27 | 2017-11-08 | Dr Reddys Laboratories Ltd | Derivados de 5-bencilaminometil-6-aminopirazolo [3,4-b] piridina como inhibidores de proteina de transferencia de ester de colesterilo (cetp) utiles para el tratamiento de aterosclerosis. |
| MX368859B (es) | 2012-05-31 | 2019-10-18 | Merck Sharp & Dohme | Formulaciones de dosis solida de un antagonista del receptor de orexina. |
| KR102160903B1 (ko) * | 2012-07-17 | 2020-10-05 | 다우 글로벌 테크놀로지스 엘엘씨 | 고도로 치환된 하이드록시알킬 메틸셀룰로즈를 포함하는 고체 분산물 |
| JP6301339B2 (ja) * | 2012-09-27 | 2018-03-28 | ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ | 少なくとも１種の水溶性ビタミンｅ誘導体および少なくとも１種の親水性ポリマーを含む、保存において安定な無塵の均質な粒子製剤 |
| US20170071930A1 (en) | 2012-11-19 | 2017-03-16 | Dr. Reddy's Laboratories Ltd. | Pharmaceutical compositions of cetp inhibitors |
| US20160287568A1 (en) * | 2013-11-22 | 2016-10-06 | Merck Sharp & Dohme Corp. | Composition of a non-nucleoside reverse transcriptase inhibitor |
| US12168004B2 (en) | 2014-02-05 | 2024-12-17 | Merck Sharp & Dohme Llc | Treatment of migraine |
| JP6491669B2 (ja) | 2014-02-05 | 2019-03-27 | メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． | Ｃｇｒｐ活性化合物の錠剤製剤 |
| WO2016084949A1 (ja) * | 2014-11-28 | 2016-06-02 | 興和株式会社 | 医薬 |
| JOP20180092A1 (ar) | 2017-10-13 | 2019-04-13 | Gilead Sciences Inc | مثبطات hiv بروتياز |
| US12383545B1 (en) | 2018-06-08 | 2025-08-12 | Allergan Pharmaceuticals International Limited | Treatment of migraine |
| CN111803632B (zh) * | 2019-04-09 | 2022-04-29 | 北京五和博澳药业股份有限公司 | 黄酮多酚类药物自乳化组合物、其制备方法、药物组合物及用途 |
| BR112021020389A2 (pt) * | 2019-04-12 | 2021-12-07 | Oblita Therapeutics Bvba | Formulações de dosagem em comprimidos de oleil fosfocolina |
| TW202104210A (zh) | 2019-04-17 | 2021-02-01 | 美商基利科學股份有限公司 | Hiv蛋白酶抑制劑 |
| CN116390712A (zh) | 2020-07-29 | 2023-07-04 | 阿勒根制药国际有限公司 | 治疗偏头痛 |
| CA3206184A1 (en) | 2020-12-22 | 2022-06-30 | Allergan Pharmaceuticals International Limited | Treatment of migraine |
| WO2023049920A1 (en) | 2021-09-27 | 2023-03-30 | Allergan Pharmaceuticals International Limited | Combination comprising atogepant for treating migraine |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020103225A1 (en) * | 2000-08-03 | 2002-08-01 | Curatolo William J. | Pharmaceutical compositions of cholesteryl ester transfer protein inhibitors |
| WO2006014357A1 (en) * | 2004-07-02 | 2006-02-09 | Merck & Co., Inc. | Cetp inhibitors |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6627767B2 (en) | 2000-08-29 | 2003-09-30 | Abbott Laboratories | Amino(oxo) acetic acid protein tyrosine phosphatase inhibitors |
| ES2284871T3 (es) | 2001-06-22 | 2007-11-16 | Pfizer Products Inc. | Composiciones farmaceuticas que contienen una dispersion solida de farmaco poco soluble y un polimero potenciador de la solubilidad. |
| EP1269994A3 (en) | 2001-06-22 | 2003-02-12 | Pfizer Products Inc. | Pharmaceutical compositions comprising drug and concentration-enhancing polymers |
| CN100410236C (zh) | 2002-01-29 | 2008-08-13 | 雪兰诺实验室有限公司 | 作为蛋白酪氨酸磷酸酶调节剂的取代亚甲基酰胺衍生物 |
| DE60322665D1 (de) * | 2002-02-01 | 2008-09-18 | Pfizer Prod Inc | Pharmazeutische darreichungsform mit gesteuerter freigabe eines cholesterylester-transferproteininhibitors |
| PL371593A1 (en) | 2002-02-01 | 2005-06-27 | Pfizer Products Inc. | Method for making homogeneous spray-dried solid amorphous drug dispersions using pressure nozzles |
| BR0306208A (pt) | 2002-08-30 | 2004-10-13 | Japan Tobacco Inc | Compostos de dibenzilamina e seu uso farmacêutico |
| MXPA05009848A (es) | 2003-03-17 | 2005-12-06 | Japan Tobacco Inc | Composiciones farmaceuticas de inhibidores de la proteina de transferencia del ester de colesterilo. |
| US20070043079A1 (en) | 2003-04-18 | 2007-02-22 | Hiromu Habashita | Heterocyclic compound containing nitrogen atom and use thereof |
| FR2875409B1 (fr) * | 2004-09-17 | 2010-05-07 | Sanofi Aventis | Composition pharmaceutique comprenant une dispersion solide a matrice polymere comprenant une phase continue de polydextrose et une phase continue d'un polymere autre que du polydextrose |
| CN102757397A (zh) * | 2005-07-01 | 2012-10-31 | 默沙东公司 | 合成cetp抑制剂的方法 |
| EP1965764B1 (en) * | 2005-12-05 | 2011-07-13 | Merck Sharp & Dohme Corp. | Self-emulsifying formulations of cetp inhibitors |
-
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- 2007-02-09 EP EP07763707.2A patent/EP1983966B1/en not_active Not-in-force
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2012
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Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020103225A1 (en) * | 2000-08-03 | 2002-08-01 | Curatolo William J. | Pharmaceutical compositions of cholesteryl ester transfer protein inhibitors |
| WO2006014357A1 (en) * | 2004-07-02 | 2006-02-09 | Merck & Co., Inc. | Cetp inhibitors |
Also Published As
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|---|---|
| CA2641451C (en) | 2012-10-02 |
| WO2007092642A3 (en) | 2007-10-04 |
| EP1983966B1 (en) | 2013-06-26 |
| IL192977A0 (en) | 2009-02-11 |
| JP5648038B2 (ja) | 2015-01-07 |
| BRPI0707584A2 (pt) | 2011-05-10 |
| CA2641451A1 (en) | 2007-08-16 |
| JP2013067635A (ja) | 2013-04-18 |
| AU2007212197B2 (en) | 2012-12-13 |
| KR101418267B1 (ko) | 2014-07-11 |
| KR20080108420A (ko) | 2008-12-15 |
| US8030359B2 (en) | 2011-10-04 |
| US20100227903A1 (en) | 2010-09-09 |
| NO20083821L (no) | 2008-09-30 |
| EP1983966A2 (en) | 2008-10-29 |
| ZA200805854B (en) | 2009-10-28 |
| CN101378731B (zh) | 2014-03-05 |
| WO2007092642A2 (en) | 2007-08-16 |
| RU2457841C2 (ru) | 2012-08-10 |
| RU2008136198A (ru) | 2010-03-20 |
| CN101378731A (zh) | 2009-03-04 |
| JP5773560B2 (ja) | 2015-09-02 |
| IL192977A (en) | 2011-01-31 |
| JP2009526075A (ja) | 2009-07-16 |
| AU2007212197A1 (en) | 2007-08-16 |
| CN103735515A (zh) | 2014-04-23 |
| NZ569700A (en) | 2011-09-30 |
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