NO323374B1 - Steroidforbindelser, anvendelse og farmasoytisk formulering omfattende slike. - Google Patents
Steroidforbindelser, anvendelse og farmasoytisk formulering omfattende slike. Download PDFInfo
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- NO323374B1 NO323374B1 NO20014925A NO20014925A NO323374B1 NO 323374 B1 NO323374 B1 NO 323374B1 NO 20014925 A NO20014925 A NO 20014925A NO 20014925 A NO20014925 A NO 20014925A NO 323374 B1 NO323374 B1 NO 323374B1
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- compound
- acid
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- steroid
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
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- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT1999MI000751A IT1311922B1 (it) | 1999-04-13 | 1999-04-13 | Composti farmaceutici. |
| PCT/EP2000/003238 WO2000061604A2 (en) | 1999-04-13 | 2000-04-11 | Pharmaceutical compounds |
Publications (3)
| Publication Number | Publication Date |
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| NO20014925D0 NO20014925D0 (no) | 2001-10-10 |
| NO20014925L NO20014925L (no) | 2001-12-13 |
| NO323374B1 true NO323374B1 (no) | 2007-04-16 |
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| NO20014925A NO323374B1 (no) | 1999-04-13 | 2001-10-10 | Steroidforbindelser, anvendelse og farmasoytisk formulering omfattende slike. |
| NO20065784A NO20065784L (no) | 1999-04-13 | 2006-12-13 | Steroidforbindelser og anvendelse av slike |
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| NO20065784A NO20065784L (no) | 1999-04-13 | 2006-12-13 | Steroidforbindelser og anvendelse av slike |
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| US (3) | US6909007B1 (de) |
| EP (2) | EP1169337B1 (de) |
| JP (1) | JP2002542162A (de) |
| KR (2) | KR100687821B1 (de) |
| CN (2) | CN1916013A (de) |
| AT (1) | ATE274521T1 (de) |
| AU (2) | AU766798B2 (de) |
| BR (1) | BR0009696A (de) |
| CA (2) | CA2586538C (de) |
| DE (1) | DE60013266T2 (de) |
| DK (1) | DK1169337T3 (de) |
| ES (1) | ES2226805T3 (de) |
| HU (1) | HUP0201872A3 (de) |
| IL (2) | IL145633A0 (de) |
| IT (1) | IT1311922B1 (de) |
| MX (1) | MXPA01010212A (de) |
| NO (2) | NO323374B1 (de) |
| NZ (1) | NZ514572A (de) |
| PL (1) | PL199579B1 (de) |
| PT (1) | PT1169337E (de) |
| RU (1) | RU2240325C2 (de) |
| SI (1) | SI1169337T1 (de) |
| TR (2) | TR200102929T2 (de) |
| WO (1) | WO2000061604A2 (de) |
| ZA (1) | ZA200108124B (de) |
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| EP1246621A4 (de) | 1999-12-23 | 2004-11-24 | Nitromed Inc | Nitrosierte und nitrosylierte cyclooxygenase-2-inhibitoren, zusammensetzungen und methoden für deren verwendung |
| CA2432642A1 (en) | 2000-12-21 | 2002-08-08 | Subhash P. Khanapure | Substituted aryl compounds as novel cyclooxygenase-2 selective inhibitors, compositions and methods of use |
| IT1320176B1 (it) * | 2000-12-22 | 2003-11-26 | Nicox Sa | Dispersioni solide di principi attivi nitrati. |
| EP1219306A1 (de) | 2000-12-29 | 2002-07-03 | Nicox S.A. | Zyklodextrin und NO-abgebende Arzneimittlen enthaltende Zusammensetzungen |
| US6696592B2 (en) | 2001-05-22 | 2004-02-24 | Nicox-S.A. | Methods of making 21-[4′-(nitrooxyalkyl)benzoate] corticosteroid derivatives and intermediates useful in the synthesis thereof |
| ITMI20011307A1 (it) * | 2001-06-21 | 2002-12-21 | Nicox Sa | Farmaci per l'epilessia |
| ITMI20020148A1 (it) | 2002-01-29 | 2003-07-29 | Nicox Sa | Nuovi corticosteroidi |
| ITMI20021025A1 (it) * | 2002-05-14 | 2003-11-14 | Nicox Sa | Farmaci per il trattamento acuto di disfunzioni del circolo venoso epatico e portale |
| US7220749B2 (en) | 2002-06-11 | 2007-05-22 | Nitromed, Inc. | Nitrosated and/or nitrosylated cyclooxygenase-2 selective inhibitors, compositions and methods of use |
| US7163958B2 (en) | 2002-07-03 | 2007-01-16 | Nitromed Inc. | Nitrosated nonsteroidal antiinflammatory compounds, compositions and methods of use |
| AU2003261281A1 (en) | 2002-07-29 | 2004-02-16 | Nicox S.A. | Cyclooxygenase- 2 selective inhibitors, compositions and methods of use |
| CN100513415C (zh) * | 2005-08-03 | 2009-07-15 | 中国人民解放军军事医学科学院毒物药物研究所 | 胆汁酸衍生物及其医药用途 |
| NZ566128A (en) | 2005-09-02 | 2011-03-31 | Nicox Sa | Nitrooxy derivatives of glucocorticoids |
| US8802726B2 (en) | 2006-02-03 | 2014-08-12 | Nicox S.A. | Use of nitrooxyderivative of drug for the treatment of muscular dystrophies |
| US7645749B2 (en) * | 2006-04-03 | 2010-01-12 | Forbes Medi-Tech Inc. | Sterol/stanol nitroderivatives and use thereof |
| US7645748B2 (en) | 2006-04-03 | 2010-01-12 | Forbes Medi-Tech Inc. | Sterol/stanol phosphorylnitroderivatives and use thereof |
| WO2008095806A1 (en) * | 2007-02-05 | 2008-08-14 | Nicox S.A. | Nitric oxide releasing steroids |
| WO2009037584A2 (en) * | 2007-08-10 | 2009-03-26 | Topigen Pharmaceuticals Inc. | Combination of nitroderivatized steroid and bronchodilator for treating respiratory disease |
| WO2009071990A2 (en) * | 2007-08-31 | 2009-06-11 | Topigen Pharmaceuticals Inc. | No-donating cordicosteroid with improved pharmacokinetic, anti-inflammatory and vasodilatory properties |
| AU2008311824A1 (en) * | 2007-10-19 | 2009-04-23 | Burnham Institute For Medical Research | Inhibitors of anti-apoptotic proteins |
| US20110130375A1 (en) | 2008-08-05 | 2011-06-02 | Nicox S.A. | New no-releasing steroids for the treatment of retina and macula lutea diseases |
| EP2560634A1 (de) | 2010-04-23 | 2013-02-27 | Piramal Enterprises Limited | Stickoxidfreisetzende prodrugs aus therapeutika |
| CU20110244A7 (es) | 2011-12-27 | 2013-08-29 | Ct De Investigación Y Desarrollo De Medicamentos Cidem | Sistemas espiroesteroidales con efectos neuroactivos y anti-inflamatorios |
| CA2897571C (en) | 2013-01-21 | 2018-12-18 | Apparao Satyam | Nitric oxide releasing prodrugs of therapeutic agents containing at least one carboxylic acid group |
| KR101711513B1 (ko) * | 2015-06-26 | 2017-03-02 | 주식회사 엘지생활건강 | 피부 개선용 조성물 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| FR2077750B1 (de) | 1970-02-11 | 1973-03-16 | Clin Byla Ets | |
| GB1458372A (en) | 1973-03-05 | 1976-12-15 | Leo Ab | Steroid carbamates and allophanates |
| JPS5845724A (ja) | 1981-09-11 | 1983-03-17 | Oriza Yuka Kk | オリザノ−ル乳化液の製造法 |
| FR2600653B1 (fr) * | 1986-06-24 | 1988-12-16 | Pasteur Strasbourg Universite | Composes de synthese associative d'acides amines soufres ou non soufres avec des derives du d-4 pregnene 3,20-dione ou avec des derives du d-1,4 pregnadiene 3,20-dione aux proprietes glucocorticoides et anti-inflammatoires, procedes d'obtention, compositions pharmaceutiques les contenant. proprietes pharmacologiques et applications |
| IT1204571B (it) * | 1987-05-08 | 1989-03-10 | Chiesi Farma Spa | Esteri di 1,4:3,6-dianidrosorbitolo-2-mononitrato e 5-mononitrato,loro procedimento di preparazione e loro composizioni farmaceutiche |
| EP1229123A3 (de) * | 1987-06-29 | 2004-11-03 | Massachusetts Institute Of Technology | Verfahren zur Herstellung von Polyester-Biopolymeren |
| DE4000397A1 (de) | 1990-01-09 | 1991-07-11 | Hoechst Ag | Lipidselektive antioxidantien sowie deren herstellung und verwendung |
| JPH04273892A (ja) | 1991-02-27 | 1992-09-30 | Kao Corp | 新規な２１−置換ステロイド化合物 |
| JP3108474B2 (ja) | 1991-08-07 | 2000-11-13 | 日清製粉株式会社 | 活性型ビタミンｄ誘導体 |
| DE69214617T2 (de) | 1991-12-26 | 1997-05-28 | Wisconsin Alumni Res Found | 26,27-Dimethylen-1-Alpha, 25-Dihydroxyvitamin-D2 und 26,27-Dihydroxyvitamin-D2 und Verfahren zu ihrer Herstellung |
| EP0562497A1 (de) | 1992-03-27 | 1993-09-29 | Nisshin Flour Milling Co., Ltd. | 1-Alpha-Hydroxy-Vitamine D7 und D4', Verfahren zur ihren Herstellung und pharmazeutische Präparate davon |
| US5194431A (en) | 1992-07-08 | 1993-03-16 | Wisconsin Alumni Research Foundation | 24-cyclopropane vitamin D derivatives |
| US5707984A (en) * | 1995-12-08 | 1998-01-13 | G. D. Searle & Co. | Steroid nitrite/nitrate ester derivatives useful as anti-inflammatory drugs |
| US5985862A (en) * | 1996-05-02 | 1999-11-16 | G.D. Searle & Co. | Pharmaceutical compositions having steroid nitrate ester derivatives useful as anti-inflammatory drugs |
| US5837698A (en) | 1996-05-02 | 1998-11-17 | G. D. Searle & Co. | Steroid nitrite and nitrate ester derivatives useful as anti-inflammatory drugs |
| DE19634793A1 (de) | 1996-08-29 | 1998-03-05 | Sanol Arznei Schwarz Gmbh | S- und O-Nitratoacylverbindungen |
| IT1285770B1 (it) * | 1996-10-04 | 1998-06-18 | Nicox Sa | Composti corticoidei |
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