NO322752B1 - Polymorfismer av N-metyl-N-(3{3-[2-tienylkarbonyl]pyrazol-[1,5-alfa]-pyrimidin-7-yl}fenyl)acetamid og blandinger og fremgangsmater relatert dertil - Google Patents
Polymorfismer av N-metyl-N-(3{3-[2-tienylkarbonyl]pyrazol-[1,5-alfa]-pyrimidin-7-yl}fenyl)acetamid og blandinger og fremgangsmater relatert dertil Download PDFInfo
- Publication number
- NO322752B1 NO322752B1 NO20021041A NO20021041A NO322752B1 NO 322752 B1 NO322752 B1 NO 322752B1 NO 20021041 A NO20021041 A NO 20021041A NO 20021041 A NO20021041 A NO 20021041A NO 322752 B1 NO322752 B1 NO 322752B1
- Authority
- NO
- Norway
- Prior art keywords
- polymorphic form
- phenyl
- acetamide
- methyl
- pyrimidin
- Prior art date
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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- A—HUMAN NECESSITIES
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- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pain & Pain Management (AREA)
- Physical Education & Sports Medicine (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38952499A | 1999-09-02 | 1999-09-02 | |
| US42162099A | 1999-10-19 | 1999-10-19 | |
| PCT/US2000/024051 WO2001015700A1 (en) | 1999-09-02 | 2000-09-01 | POLYMORPHS OF N-METHYL-N-(3-{3-[2-THIENYLCARBONYL]-PYRAZOL-[1,5-α]-PYRIMIDIN -7-YL }PHENYL )ACETAMIDE AND COMPOSITIONS AND METHODS RELATED THERETO |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20021041D0 NO20021041D0 (no) | 2002-03-01 |
| NO20021041L NO20021041L (no) | 2002-04-03 |
| NO322752B1 true NO322752B1 (no) | 2006-12-04 |
Family
ID=27012737
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20021041A NO322752B1 (no) | 1999-09-02 | 2002-03-01 | Polymorfismer av N-metyl-N-(3{3-[2-tienylkarbonyl]pyrazol-[1,5-alfa]-pyrimidin-7-yl}fenyl)acetamid og blandinger og fremgangsmater relatert dertil |
Country Status (26)
| Country | Link |
|---|---|
| EP (2) | EP1477169A1 (pt) |
| JP (1) | JP4592241B2 (pt) |
| KR (1) | KR20020035585A (pt) |
| CN (2) | CN1198824C (pt) |
| AP (1) | AP1631A (pt) |
| AT (1) | ATE269082T1 (pt) |
| AU (2) | AU769856B2 (pt) |
| BR (1) | BR0014459A (pt) |
| CA (1) | CA2382588C (pt) |
| CZ (1) | CZ2002783A3 (pt) |
| DE (1) | DE60011638T2 (pt) |
| DK (1) | DK1214075T3 (pt) |
| EA (1) | EA004706B1 (pt) |
| ES (1) | ES2222920T3 (pt) |
| HK (1) | HK1047407B (pt) |
| HU (1) | HUP0202698A3 (pt) |
| IL (2) | IL148242A0 (pt) |
| MX (1) | MXPA02002314A (pt) |
| NO (1) | NO322752B1 (pt) |
| NZ (1) | NZ517298A (pt) |
| OA (1) | OA12200A (pt) |
| PL (1) | PL353362A1 (pt) |
| PT (1) | PT1214075E (pt) |
| SK (1) | SK2782002A3 (pt) |
| TR (1) | TR200200534T2 (pt) |
| WO (1) | WO2001015700A1 (pt) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003268212B2 (en) * | 2002-08-26 | 2008-08-14 | Neurocrine Biosciences, Inc. | Novel polymorph of N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1,5-alpha]-pyrimidin-7-YL}phenyl)acetamide and compositions and methods related thereto |
| WO2004110454A1 (ja) * | 2003-06-13 | 2004-12-23 | Ishihara Sangyo Kaisha, Ltd. | アデノシンＡ2ａ受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物 |
| US7371906B2 (en) | 2004-08-24 | 2008-05-13 | Eastman Kodak Company | Process for photo-oxidative stability improvements |
| EP1956021A1 (en) * | 2006-10-11 | 2008-08-13 | Ferrer Internacional, S.A. | Process for the manufacture of a crystalline pyrazolo[1,5-a]pyrimidine compound |
| EP1918290A1 (en) * | 2006-10-11 | 2008-05-07 | Ferrer Internacional, S.A. | Polymorph B of N-{2-Fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo[1,5-a] pyrimidin-7-yl]-phenyl}-N-methyl-acetamide |
| CN101177427B (zh) * | 2006-11-09 | 2011-07-20 | 中国人民解放军军事医学科学院放射与辐射医学研究所 | 一种用于催眠的化合物的多晶型α和溶剂化物,其制备方法及含该物质的组合物 |
| US20120028045A1 (en) * | 2009-03-24 | 2012-02-02 | Glenmark Generics Ltd | Processes for the Preparation of Indiplon and Intermediates Thereof |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4521422A (en) * | 1983-06-23 | 1985-06-04 | American Cyanamid Company | Aryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanones |
| NZ208554A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions |
| US4626538A (en) * | 1983-06-23 | 1986-12-02 | American Cyanamid Company | [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines |
| US4654347A (en) * | 1983-06-23 | 1987-03-31 | American Cyanamid Company | Aryl and heteroaryl[[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]methanones |
| SG30590G (en) * | 1985-05-13 | 1995-09-18 | American Cyanamid Co | D7-(3-disubstituted amino) phenylaepyrazolod 1,5-aaepyrimidines |
| US5421422A (en) * | 1993-11-19 | 1995-06-06 | Boretec Inc | Roller cutter mount for tunneling machine |
-
2000
- 2000-09-01 CN CNB008131589A patent/CN1198824C/zh not_active Expired - Fee Related
- 2000-09-01 CA CA002382588A patent/CA2382588C/en not_active Expired - Fee Related
- 2000-09-01 AP APAP/P/2002/002428A patent/AP1631A/en active
- 2000-09-01 BR BR0014459-2A patent/BR0014459A/pt not_active Application Discontinuation
- 2000-09-01 DE DE60011638T patent/DE60011638T2/de not_active Expired - Lifetime
- 2000-09-01 SK SK278-2002A patent/SK2782002A3/sk unknown
- 2000-09-01 AU AU69491/00A patent/AU769856B2/en not_active Ceased
- 2000-09-01 PT PT00957941T patent/PT1214075E/pt unknown
- 2000-09-01 CZ CZ2002783A patent/CZ2002783A3/cs unknown
- 2000-09-01 EP EP04013998A patent/EP1477169A1/en not_active Withdrawn
- 2000-09-01 DK DK00957941T patent/DK1214075T3/da active
- 2000-09-01 TR TR2002/00534T patent/TR200200534T2/xx unknown
- 2000-09-01 AT AT00957941T patent/ATE269082T1/de active
- 2000-09-01 JP JP2001519914A patent/JP4592241B2/ja not_active Expired - Lifetime
- 2000-09-01 EA EA200200320A patent/EA004706B1/ru not_active IP Right Cessation
- 2000-09-01 CN CNB2005100545485A patent/CN1331865C/zh not_active Expired - Fee Related
- 2000-09-01 NZ NZ517298A patent/NZ517298A/en not_active IP Right Cessation
- 2000-09-01 IL IL14824200A patent/IL148242A0/xx active IP Right Grant
- 2000-09-01 EP EP00957941A patent/EP1214075B1/en not_active Expired - Lifetime
- 2000-09-01 PL PL00353362A patent/PL353362A1/xx not_active Application Discontinuation
- 2000-09-01 MX MXPA02002314A patent/MXPA02002314A/es active IP Right Grant
- 2000-09-01 OA OA1200200057A patent/OA12200A/en unknown
- 2000-09-01 WO PCT/US2000/024051 patent/WO2001015700A1/en active IP Right Grant
- 2000-09-01 ES ES00957941T patent/ES2222920T3/es not_active Expired - Lifetime
- 2000-09-01 KR KR1020027002829A patent/KR20020035585A/ko not_active Application Discontinuation
- 2000-09-01 HU HU0202698A patent/HUP0202698A3/hu unknown
-
2002
- 2002-02-19 IL IL148242A patent/IL148242A/en not_active IP Right Cessation
- 2002-03-01 NO NO20021041A patent/NO322752B1/no not_active IP Right Cessation
- 2002-12-16 HK HK02109094.4A patent/HK1047407B/zh not_active IP Right Cessation
-
2004
- 2004-03-31 AU AU2004201356A patent/AU2004201356A1/en not_active Abandoned
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| Date | Code | Title | Description |
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| MM1K | Lapsed by not paying the annual fees |