IL148242A0 - Polymorphs of n-methyl-n(3-(3-[2 thienylcarbonyl] pyrazol-[1, 5-a]-pyrimidin-7-yl} phenyl) acetamide, pharmaceutical compositions containing the same and processes for the preparation thereof - Google Patents
Polymorphs of n-methyl-n(3-(3-[2 thienylcarbonyl] pyrazol-[1, 5-a]-pyrimidin-7-yl} phenyl) acetamide, pharmaceutical compositions containing the same and processes for the preparation thereofInfo
- Publication number
- IL148242A0 IL148242A0 IL14824200A IL14824200A IL148242A0 IL 148242 A0 IL148242 A0 IL 148242A0 IL 14824200 A IL14824200 A IL 14824200A IL 14824200 A IL14824200 A IL 14824200A IL 148242 A0 IL148242 A0 IL 148242A0
- Authority
- IL
- Israel
- Prior art keywords
- thienylcarbonyl
- polymorphs
- pyrazol
- pyrimidin
- acetamide
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38952499A | 1999-09-02 | 1999-09-02 | |
| US42162099A | 1999-10-19 | 1999-10-19 | |
| PCT/US2000/024051 WO2001015700A1 (en) | 1999-09-02 | 2000-09-01 | POLYMORPHS OF N-METHYL-N-(3-{3-[2-THIENYLCARBONYL]-PYRAZOL-[1,5-α]-PYRIMIDIN -7-YL }PHENYL )ACETAMIDE AND COMPOSITIONS AND METHODS RELATED THERETO |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL148242A0 true IL148242A0 (en) | 2002-09-12 |
Family
ID=27012737
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL14824200A IL148242A0 (en) | 1999-09-02 | 2000-09-01 | Polymorphs of n-methyl-n(3-(3-[2 thienylcarbonyl] pyrazol-[1, 5-a]-pyrimidin-7-yl} phenyl) acetamide, pharmaceutical compositions containing the same and processes for the preparation thereof |
| IL148242A IL148242A (en) | 1999-09-02 | 2002-02-19 | Polymorphs of n-methyl- n |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL148242A IL148242A (en) | 1999-09-02 | 2002-02-19 | Polymorphs of n-methyl- n |
Country Status (26)
| Country | Link |
|---|---|
| EP (2) | EP1477169A1 (pt) |
| JP (1) | JP4592241B2 (pt) |
| KR (1) | KR20020035585A (pt) |
| CN (2) | CN1331865C (pt) |
| AP (1) | AP1631A (pt) |
| AT (1) | ATE269082T1 (pt) |
| AU (2) | AU769856B2 (pt) |
| BR (1) | BR0014459A (pt) |
| CA (1) | CA2382588C (pt) |
| CZ (1) | CZ2002783A3 (pt) |
| DE (1) | DE60011638T2 (pt) |
| DK (1) | DK1214075T3 (pt) |
| EA (1) | EA004706B1 (pt) |
| ES (1) | ES2222920T3 (pt) |
| HK (1) | HK1047407B (pt) |
| HU (1) | HUP0202698A3 (pt) |
| IL (2) | IL148242A0 (pt) |
| MX (1) | MXPA02002314A (pt) |
| NO (1) | NO322752B1 (pt) |
| NZ (1) | NZ517298A (pt) |
| OA (1) | OA12200A (pt) |
| PL (1) | PL353362A1 (pt) |
| PT (1) | PT1214075E (pt) |
| SK (1) | SK2782002A3 (pt) |
| TR (1) | TR200200534T2 (pt) |
| WO (1) | WO2001015700A1 (pt) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003268212B2 (en) * | 2002-08-26 | 2008-08-14 | Neurocrine Biosciences, Inc. | Novel polymorph of N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1,5-alpha]-pyrimidin-7-YL}phenyl)acetamide and compositions and methods related thereto |
| WO2004110454A1 (ja) * | 2003-06-13 | 2004-12-23 | Ishihara Sangyo Kaisha, Ltd. | アデノシンＡ2ａ受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物 |
| US7371906B2 (en) | 2004-08-24 | 2008-05-13 | Eastman Kodak Company | Process for photo-oxidative stability improvements |
| EP1918290A1 (en) | 2006-10-11 | 2008-05-07 | Ferrer Internacional, S.A. | Polymorph B of N-{2-Fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo[1,5-a] pyrimidin-7-yl]-phenyl}-N-methyl-acetamide |
| EP1956021A1 (en) * | 2006-10-11 | 2008-08-13 | Ferrer Internacional, S.A. | Process for the manufacture of a crystalline pyrazolo[1,5-a]pyrimidine compound |
| CN101177427B (zh) * | 2006-11-09 | 2011-07-20 | 中国人民解放军军事医学科学院放射与辐射医学研究所 | 一种用于催眠的化合物的多晶型α和溶剂化物,其制备方法及含该物质的组合物 |
| WO2010109480A2 (en) * | 2009-03-24 | 2010-09-30 | Glenmark Generics Limited | Processes for the preparation of indiplon and intermediates thereof |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ208554A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions |
| US4654347A (en) * | 1983-06-23 | 1987-03-31 | American Cyanamid Company | Aryl and heteroaryl[[7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]methanones |
| US4521422A (en) * | 1983-06-23 | 1985-06-04 | American Cyanamid Company | Aryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanones |
| US4626538A (en) * | 1983-06-23 | 1986-12-02 | American Cyanamid Company | [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines |
| DE19975048I2 (de) * | 1985-05-13 | 2001-06-13 | American Cyanamid Co | 7-(3-Disubstituierte Amino)phenyl pyrazolo 1,5-a -pyrimidine |
| US5421422A (en) * | 1993-11-19 | 1995-06-06 | Boretec Inc | Roller cutter mount for tunneling machine |
-
2000
- 2000-09-01 HU HU0202698A patent/HUP0202698A3/hu unknown
- 2000-09-01 CZ CZ2002783A patent/CZ2002783A3/cs unknown
- 2000-09-01 ES ES00957941T patent/ES2222920T3/es not_active Expired - Lifetime
- 2000-09-01 EP EP04013998A patent/EP1477169A1/en not_active Withdrawn
- 2000-09-01 DK DK00957941T patent/DK1214075T3/da active
- 2000-09-01 AU AU69491/00A patent/AU769856B2/en not_active Ceased
- 2000-09-01 AT AT00957941T patent/ATE269082T1/de active
- 2000-09-01 MX MXPA02002314A patent/MXPA02002314A/es active IP Right Grant
- 2000-09-01 BR BR0014459-2A patent/BR0014459A/pt not_active Application Discontinuation
- 2000-09-01 CN CNB2005100545485A patent/CN1331865C/zh not_active Expired - Fee Related
- 2000-09-01 DE DE60011638T patent/DE60011638T2/de not_active Expired - Lifetime
- 2000-09-01 NZ NZ517298A patent/NZ517298A/en not_active IP Right Cessation
- 2000-09-01 EP EP00957941A patent/EP1214075B1/en not_active Expired - Lifetime
- 2000-09-01 WO PCT/US2000/024051 patent/WO2001015700A1/en active IP Right Grant
- 2000-09-01 PT PT00957941T patent/PT1214075E/pt unknown
- 2000-09-01 JP JP2001519914A patent/JP4592241B2/ja not_active Expired - Lifetime
- 2000-09-01 SK SK278-2002A patent/SK2782002A3/sk unknown
- 2000-09-01 TR TR2002/00534T patent/TR200200534T2/xx unknown
- 2000-09-01 KR KR1020027002829A patent/KR20020035585A/ko not_active Application Discontinuation
- 2000-09-01 CA CA002382588A patent/CA2382588C/en not_active Expired - Fee Related
- 2000-09-01 AP APAP/P/2002/002428A patent/AP1631A/en active
- 2000-09-01 IL IL14824200A patent/IL148242A0/xx active IP Right Grant
- 2000-09-01 OA OA1200200057A patent/OA12200A/en unknown
- 2000-09-01 EA EA200200320A patent/EA004706B1/ru not_active IP Right Cessation
- 2000-09-01 PL PL00353362A patent/PL353362A1/xx not_active Application Discontinuation
- 2000-09-01 CN CNB008131589A patent/CN1198824C/zh not_active Expired - Fee Related
-
2002
- 2002-02-19 IL IL148242A patent/IL148242A/en not_active IP Right Cessation
- 2002-03-01 NO NO20021041A patent/NO322752B1/no not_active IP Right Cessation
- 2002-12-16 HK HK02109094.4A patent/HK1047407B/zh not_active IP Right Cessation
-
2004
- 2004-03-31 AU AU2004201356A patent/AU2004201356A1/en not_active Abandoned
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed |