NO322394B1 - 2-arylimino-2,3-dihydrotiazoler, fremgangsmate for fremstilling av disse, farmasoytiske preparater inneholdende disse samt deres anvendelse for fremstilling av medikamenter for behandling av tilstander eller sykdommer der somatostatinreseptorene er innvolvert. - Google Patents

2-arylimino-2,3-dihydrotiazoler, fremgangsmate for fremstilling av disse, farmasoytiske preparater inneholdende disse samt deres anvendelse for fremstilling av medikamenter for behandling av tilstander eller sykdommer der somatostatinreseptorene er innvolvert. Download PDF

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Publication number
NO322394B1
NO322394B1 NO20020314A NO20020314A NO322394B1 NO 322394 B1 NO322394 B1 NO 322394B1 NO 20020314 A NO20020314 A NO 20020314A NO 20020314 A NO20020314 A NO 20020314A NO 322394 B1 NO322394 B1 NO 322394B1
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Norway
Prior art keywords
general formula
residue
residues
resin
treatment
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NO20020314A
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English (en)
Norwegian (no)
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NO20020314D0 (no
NO20020314L (no
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Christophe Alain Thurieau
Christophe Philippe Moinet
Carole Sackur
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Sod Conseils Rech Applic
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Publication of NO20020314D0 publication Critical patent/NO20020314D0/no
Publication of NO20020314L publication Critical patent/NO20020314L/no
Publication of NO322394B1 publication Critical patent/NO322394B1/no

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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NO20020314A 1999-07-22 2002-01-21 2-arylimino-2,3-dihydrotiazoler, fremgangsmate for fremstilling av disse, farmasoytiske preparater inneholdende disse samt deres anvendelse for fremstilling av medikamenter for behandling av tilstander eller sykdommer der somatostatinreseptorene er innvolvert. NO322394B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9909496A FR2796643B1 (fr) 1999-07-22 1999-07-22 Derives de 2-arylimino-2, 3-dihydrothiazoles, leurs procedes de preparation et leur utilisation therapeutique
PCT/FR2000/002095 WO2001007424A1 (fr) 1999-07-22 2000-07-21 2-arylimino-2,3-dihydrothiazoles et leur utilisation comme ligands des recepteurs de la somatostatine

Publications (3)

Publication Number Publication Date
NO20020314D0 NO20020314D0 (no) 2002-01-21
NO20020314L NO20020314L (no) 2002-03-06
NO322394B1 true NO322394B1 (no) 2006-10-02

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Family Applications (1)

Application Number Title Priority Date Filing Date
NO20020314A NO322394B1 (no) 1999-07-22 2002-01-21 2-arylimino-2,3-dihydrotiazoler, fremgangsmate for fremstilling av disse, farmasoytiske preparater inneholdende disse samt deres anvendelse for fremstilling av medikamenter for behandling av tilstander eller sykdommer der somatostatinreseptorene er innvolvert.

Country Status (20)

Country Link
US (1) US6727269B1 (fr)
EP (1) EP1202980A1 (fr)
JP (2) JP4063537B2 (fr)
KR (1) KR100692352B1 (fr)
CN (1) CN100443479C (fr)
AR (1) AR035321A1 (fr)
AU (1) AU782187B2 (fr)
BR (1) BR0012647A (fr)
CA (1) CA2382940C (fr)
CZ (1) CZ302073B6 (fr)
FR (1) FR2796643B1 (fr)
HK (1) HK1048314A1 (fr)
HU (1) HUP0202425A3 (fr)
IL (3) IL147582A0 (fr)
MX (1) MXPA02000723A (fr)
NO (1) NO322394B1 (fr)
NZ (1) NZ516599A (fr)
PL (1) PL353831A1 (fr)
RU (1) RU2266287C2 (fr)
WO (1) WO2001007424A1 (fr)

Families Citing this family (30)

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Publication number Priority date Publication date Assignee Title
FR2819508B1 (fr) * 2001-01-12 2005-01-21 Sod Conseils Rech Applic Derives de 2-arylimino-2, 3-dihydorthiazoles, leurs procedes de preparation et leur utilisation therapeutiques
ES2336425T3 (es) 2000-06-30 2010-04-13 Dainippon Sumitomo Pharma Co., Ltd. Derivados de tiazoles utiles como agentes antiinflamatorios.
DE10133665A1 (de) * 2001-07-11 2003-01-30 Boehringer Ingelheim Pharma Carbonsäurederivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Herstellung
AU2002359359A1 (en) 2001-12-28 2003-07-24 Somatocor Pharmaceuticals, Inc. Imidazolidin-2,4-dione derivatives as non-peptide somatostatin receptor ligands
US7067538B2 (en) 2002-08-09 2006-06-27 Warner-Lambert Company, Llc MCP-1 receptor antagonists and methods of use thereof
JP4896387B2 (ja) * 2003-09-30 2012-03-14 武田薬品工業株式会社 チアゾリン誘導体およびその用途
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RU2002104574A (ru) 2004-01-20
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FR2796643B1 (fr) 2005-04-29
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BR0012647A (pt) 2002-04-09
MXPA02000723A (es) 2002-09-17
WO2001007424A1 (fr) 2001-02-01
PL353831A1 (en) 2003-12-01
IL147582A (en) 2009-08-03
FR2796643A1 (fr) 2001-01-26
RU2266287C2 (ru) 2005-12-20
AU7005300A (en) 2001-02-13
KR100692352B1 (ko) 2007-03-12
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JP2006257093A (ja) 2006-09-28
JP4063537B2 (ja) 2008-03-19
CN1362952A (zh) 2002-08-07
CA2382940A1 (fr) 2001-02-01
IL185786A0 (en) 2008-01-06
CZ2002187A3 (cs) 2002-06-12
EP1202980A1 (fr) 2002-05-08
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AU782187B2 (en) 2005-07-07
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