NO317251B1 - Nye aminer som farmasoytiske midler - Google Patents

Nye aminer som farmasoytiske midler Download PDF

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Publication number
NO317251B1
NO317251B1 NO20003037A NO20003037A NO317251B1 NO 317251 B1 NO317251 B1 NO 317251B1 NO 20003037 A NO20003037 A NO 20003037A NO 20003037 A NO20003037 A NO 20003037A NO 317251 B1 NO317251 B1 NO 317251B1
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Norway
Prior art keywords
compound according
treatment
preparation
drug
methyl
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NO20003037A
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English (en)
Norwegian (no)
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NO20003037D0 (no
NO20003037L (no
Inventor
David Christopher Horwell
David Juergen Wustrow
Justin Stephen Bryans
Clare Octavia Kneen
Thomas Richard Belliotti
Thomas Capiris
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Warner Lambert Co
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Publication of NO20003037D0 publication Critical patent/NO20003037D0/no
Publication of NO20003037L publication Critical patent/NO20003037L/no
Publication of NO317251B1 publication Critical patent/NO317251B1/no

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    • C07—ORGANIC CHEMISTRY
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    • C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/31—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atoms of the sulfonamide groups bound to acyclic carbon atoms
    • C07C311/32—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atoms of the sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
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    • C07C233/36—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
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    • C07C311/05—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by nitrogen atoms, not being part of nitro or nitroso groups
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    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
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    • C07C311/33—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atoms of the sulfonamide groups bound to acyclic carbon atoms of a saturated carbon skeleton containing rings
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    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
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    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
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    • C07C2601/14—The ring being saturated
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    • C07C2602/00—Systems containing two condensed rings
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    • C07C2602/46—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing nine carbon atoms
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    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/70—Ring systems containing bridged rings containing three rings containing only six-membered rings
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PCT/US1998/023917 WO1999031074A2 (en) 1997-12-16 1998-11-10 ((cyclo)alkyl substituted)-.gamma.-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders

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DE69822214T2 (de) 2005-03-10
NO20003037D0 (no) 2000-06-14
ATE260904T1 (de) 2004-03-15
US6521650B1 (en) 2003-02-18
ES2216338T3 (es) 2004-10-16
NO20040817L (no) 2004-02-24
PL348305A1 (en) 2002-05-20
HUP0100472A2 (hu) 2001-09-28
IS5436A (is) 2000-04-07
KR20010033154A (ko) 2001-04-25
EP1400526A2 (en) 2004-03-24
WO1999031074A3 (en) 1999-11-04
WO1999031074A2 (en) 1999-06-24
US20030229054A1 (en) 2003-12-11
NZ503981A (en) 2002-12-20
CN1279673A (zh) 2001-01-10
AU759619B2 (en) 2003-04-17
HUP0100472A3 (en) 2003-03-28
DE69822214D1 (de) 2004-04-08
JP2002508361A (ja) 2002-03-19
IL135314A0 (en) 2001-05-20
TR200001794T2 (tr) 2000-10-23
NO20003037L (no) 2000-06-14
EP1045839A2 (en) 2000-10-25
CA2304965A1 (en) 1999-06-24
SI1045839T1 (en) 2004-06-30
BR9813656A (pt) 2000-10-10
AU1796299A (en) 1999-07-05
EP1045839B1 (en) 2004-03-03
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