NO314142B1 - Nye strukturelle analoger av vitamin D - Google Patents

Nye strukturelle analoger av vitamin D Download PDF

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Publication number
NO314142B1
NO314142B1 NO19960099A NO960099A NO314142B1 NO 314142 B1 NO314142 B1 NO 314142B1 NO 19960099 A NO19960099 A NO 19960099A NO 960099 A NO960099 A NO 960099A NO 314142 B1 NO314142 B1 NO 314142B1
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Norway
Prior art keywords
mmol
solution
hexane
synthesis
compound
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NO19960099A
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English (en)
Norwegian (no)
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NO960099L (no
NO960099D0 (no
Inventor
Roger Bouillon
Maurits Vandewalle
Pierre Jean De Clercq
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Theramex
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Publication of NO960099D0 publication Critical patent/NO960099D0/no
Publication of NO960099L publication Critical patent/NO960099L/no
Publication of NO314142B1 publication Critical patent/NO314142B1/no

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    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C47/00Compounds having —CHO groups
    • C07C47/02Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen
    • C07C47/198Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen containing ether groups, groups, groups, or groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • C07C49/00Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/20Unsaturated compounds containing keto groups bound to acyclic carbon atoms
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    • C07C49/385Saturated compounds containing a keto group being part of a ring
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    • C07C49/587Unsaturated compounds containing a keto groups being part of a ring
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    • C07C49/755Unsaturated compounds containing a keto groups being part of a ring containing ether groups, groups, groups, or groups a keto group being part of a condensed ring system with two or three rings, at least one ring being a six-membered aromatic ring
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  • Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Tropical Medicine & Parasitology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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NO19960099A 1993-07-09 1996-01-09 Nye strukturelle analoger av vitamin D NO314142B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP93202037 1993-07-09
PCT/EP1994/002294 WO1995001960A1 (fr) 1993-07-09 1994-07-07 Nouveaux analogues structuraux de la vitamine d

Publications (3)

Publication Number Publication Date
NO960099D0 NO960099D0 (no) 1996-01-09
NO960099L NO960099L (no) 1996-03-08
NO314142B1 true NO314142B1 (no) 2003-02-03

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ID=8213977

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19960099A NO314142B1 (no) 1993-07-09 1996-01-09 Nye strukturelle analoger av vitamin D

Country Status (16)

Country Link
US (2) US6017907A (fr)
EP (2) EP0972762B1 (fr)
JP (2) JP4235256B2 (fr)
CN (1) CN1103755C (fr)
AT (2) ATE191712T1 (fr)
AU (1) AU699200B2 (fr)
CA (1) CA2166898C (fr)
DE (2) DE69423966T2 (fr)
DK (2) DK0972762T3 (fr)
ES (2) ES2147238T3 (fr)
GR (1) GR3033856T3 (fr)
NO (1) NO314142B1 (fr)
NZ (1) NZ271332A (fr)
PT (2) PT972762E (fr)
RU (1) RU2153491C2 (fr)
WO (1) WO1995001960A1 (fr)

Families Citing this family (58)

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US5661140A (en) * 1994-11-21 1997-08-26 Wisconsin Alumni Research Foundation 18-nor-vitamin D compounds
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US5716946A (en) * 1996-02-13 1998-02-10 Wisconsin Alumni Research Foundation Multiple sclerosis treatment
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DE69804606T2 (de) * 1997-05-23 2002-11-07 Basilea Pharmaceutica Ag Binni Cyclohexandiolderivate
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US5962707A (en) * 1998-08-18 1999-10-05 Wisconsin Alumni Research Foundation 19-nor-vitamin D3 compounds with calcemic activity
US6479474B2 (en) 1999-07-08 2002-11-12 Wisconsin Alumni Research Foundation Dietary calcium as a supplement to vitamin D compound treatment of multiple sclerosis
DE19935771A1 (de) * 1999-07-23 2001-02-01 Schering Ag Neue Vitamin D-Derivate mit cyclischen Substrukturen in den Seitenketten, Verfahren und Zwischenprodukte zu ihrer Herstellung und die Verwendung zur Herstellung von Arzneimitteln
US6310262B1 (en) * 1999-10-18 2001-10-30 Basilea Pharmaceutica Ag Process for preparing retiferol derivatives
EP1106618A1 (fr) * 1999-12-08 2001-06-13 Laboratoire Theramex Précurseurs pour le cycle A de la vitamine D, procédé pour les préparer et intermédiaires de ce procédé
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CA2528378A1 (fr) * 2003-06-11 2004-12-23 Novacea, Inc. Traitement des maladies a mediation immunologique au moyen de composes a base de vitamine d active, seuls ou en association avec d'autres agents therapeutiques
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US7713951B2 (en) * 2004-04-09 2010-05-11 Wisconsin Alumni Research Foundation 2-alkylidene-18,19-dinor-vitamin D compounds
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JP6300030B2 (ja) 2011-12-29 2018-03-28 サンド アクツィエンゲゼルシャフト 2−((2s,3s,4r,5r)−5−((s)−3−アミノ−2−ヒドロキシプロプ−1−イル)−4−メトキシ−3−(フェニルスルホニルメチル)テトラヒドロフラン−2−イル)アセトアルデヒド誘導体およびこれらを調製するためのプロセス
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DE69423966T2 (de) 2000-11-16
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DK0972762T3 (da) 2004-02-09
AU7492794A (en) 1995-02-06
CN1130899A (zh) 1996-09-11
EP0972762A2 (fr) 2000-01-19
NO960099L (no) 1996-03-08
CA2166898A1 (fr) 1995-01-19
EP0707566A1 (fr) 1996-04-24
EP0972762B1 (fr) 2003-10-01
ATE251133T1 (de) 2003-10-15
DE69433220D1 (de) 2003-11-06
GR3033856T3 (en) 2000-10-31
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EP0972762A3 (fr) 2000-02-23
PT707566E (pt) 2000-09-29
US6017907A (en) 2000-01-25
AU699200B2 (en) 1998-11-26
US6548715B1 (en) 2003-04-15
CN1103755C (zh) 2003-03-26
ES2209327T3 (es) 2004-06-16
PT972762E (pt) 2004-02-27
JP4235256B2 (ja) 2009-03-11
DE69433220T2 (de) 2004-08-19
DK0707566T3 (da) 2000-09-04
JPH09500117A (ja) 1997-01-07
DE69423966D1 (de) 2000-05-18
RU2153491C2 (ru) 2000-07-27
ATE191712T1 (de) 2000-04-15
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JP4312183B2 (ja) 2009-08-12
CA2166898C (fr) 2004-09-07

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