NO312134B1 - Tiazolderivater, fremgangsmåte for fremstilling og anvendelse av dem, farmasöytisk preparat inneholdende dem og mellomprodukteri fremstillingen - Google Patents
Tiazolderivater, fremgangsmåte for fremstilling og anvendelse av dem, farmasöytisk preparat inneholdende dem og mellomprodukteri fremstillingen Download PDFInfo
- Publication number
- NO312134B1 NO312134B1 NO19986160A NO986160A NO312134B1 NO 312134 B1 NO312134 B1 NO 312134B1 NO 19986160 A NO19986160 A NO 19986160A NO 986160 A NO986160 A NO 986160A NO 312134 B1 NO312134 B1 NO 312134B1
- Authority
- NO
- Norway
- Prior art keywords
- carbonyl
- guanidino
- ylmethoxy
- piperidin
- ethyl
- Prior art date
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Classifications
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Diabetes (AREA)
- Communicable Diseases (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Ophthalmology & Optometry (AREA)
- Nutrition Science (AREA)
- Virology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP98100007 | 1998-01-02 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO986160D0 NO986160D0 (no) | 1998-12-28 |
| NO986160L NO986160L (no) | 1999-07-05 |
| NO312134B1 true NO312134B1 (no) | 2002-03-25 |
Family
ID=8231230
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19986160A NO312134B1 (no) | 1998-01-02 | 1998-12-28 | Tiazolderivater, fremgangsmåte for fremstilling og anvendelse av dem, farmasöytisk preparat inneholdende dem og mellomprodukteri fremstillingen |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US6001855A (fr) |
| JP (1) | JP3154982B2 (fr) |
| KR (1) | KR100312900B1 (fr) |
| CN (1) | CN1098849C (fr) |
| AR (1) | AR014211A1 (fr) |
| AT (1) | ATE217621T1 (fr) |
| AU (1) | AU718659B2 (fr) |
| BR (1) | BR9805750A (fr) |
| CA (1) | CA2257322C (fr) |
| CO (1) | CO4990935A1 (fr) |
| DE (1) | DE69805392T2 (fr) |
| DK (1) | DK0928793T3 (fr) |
| ES (1) | ES2176895T3 (fr) |
| HK (1) | HK1021733A1 (fr) |
| HR (1) | HRP980644B1 (fr) |
| HU (1) | HUP9803041A3 (fr) |
| ID (1) | ID21878A (fr) |
| IL (1) | IL127784A (fr) |
| MA (1) | MA26590A1 (fr) |
| NO (1) | NO312134B1 (fr) |
| PE (1) | PE20000116A1 (fr) |
| PL (1) | PL330620A1 (fr) |
| PT (1) | PT928793E (fr) |
| RU (1) | RU2166503C2 (fr) |
| SG (1) | SG72911A1 (fr) |
| TR (1) | TR199802766A2 (fr) |
| UY (1) | UY25335A1 (fr) |
| YU (1) | YU60998A (fr) |
| ZA (1) | ZA9811923B (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4517454B2 (ja) * | 2000-06-01 | 2010-08-04 | 宇部興産株式会社 | ４−（１−フルオロエチル）チアゾール−５−カルボン酸アミド誘導体及び農園芸用の有害生物防除剤 |
| US6451821B1 (en) * | 2000-06-09 | 2002-09-17 | Aventis Pharma S.A. | Use of 2-aminothiazoline derivatives as inhibitors of inducible no-synthase |
| US6420566B2 (en) * | 2000-06-09 | 2002-07-16 | Aventis Pharma S.A. | Pharmaceutical compositions containing a 4, 5-dihydro-1, 3-thiazol-2-ylamine derivative, novel derivatives and preparation thereof |
| RU2018122461A (ru) * | 2015-12-04 | 2020-01-13 | Янссен Байотек, Инк. | Лечение дегенерации сетчатки с применением клеток-предшественников |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2138803B (en) * | 1983-04-26 | 1986-06-18 | Shionogi & Co | 2-guanidino-4-hydroxymethylthiazole and derivatives thereof |
| IL95548A0 (en) * | 1989-09-15 | 1991-06-30 | Fujisawa Pharmaceutical Co | Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition containing the same |
| TW201303B (fr) * | 1990-07-05 | 1993-03-01 | Hoffmann La Roche | |
| ATE203234T1 (de) * | 1995-08-30 | 2001-08-15 | Searle & Co | Meta-guanidine, harnstoff, thioharnstoff oder azacyklische aminobenzoesäure-derivate als integrin antagonisten |
| EP0880511A4 (fr) * | 1996-01-16 | 1999-06-16 | Merck & Co Inc | Antagonistes du recepteur integrine |
| DE69835430T2 (de) * | 1997-05-30 | 2007-03-08 | Takeda Pharmaceutical Co. Ltd. | Sulfonamidderivate, ihre herstellung und verwendung |
-
1998
- 1998-12-22 US US09/218,200 patent/US6001855A/en not_active Expired - Fee Related
- 1998-12-28 NO NO19986160A patent/NO312134B1/no unknown
- 1998-12-29 YU YU60998A patent/YU60998A/sh unknown
- 1998-12-29 AR ARP980106722A patent/AR014211A1/es not_active Application Discontinuation
- 1998-12-29 PE PE1998001292A patent/PE20000116A1/es not_active Application Discontinuation
- 1998-12-29 ZA ZA9811923A patent/ZA9811923B/xx unknown
- 1998-12-29 IL IL12778498A patent/IL127784A/en not_active IP Right Cessation
- 1998-12-29 HR HR980644A patent/HRP980644B1/xx not_active IP Right Cessation
- 1998-12-30 DK DK98124819T patent/DK0928793T3/da active
- 1998-12-30 AU AU96145/98A patent/AU718659B2/en not_active Ceased
- 1998-12-30 HU HU9803041A patent/HUP9803041A3/hu unknown
- 1998-12-30 PL PL98330620A patent/PL330620A1/xx not_active Application Discontinuation
- 1998-12-30 SG SG1998005979A patent/SG72911A1/en unknown
- 1998-12-30 CA CA002257322A patent/CA2257322C/fr not_active Expired - Fee Related
- 1998-12-30 KR KR1019980061644A patent/KR100312900B1/ko not_active IP Right Cessation
- 1998-12-30 TR TR1998/02766A patent/TR199802766A2/xx unknown
- 1998-12-30 DE DE69805392T patent/DE69805392T2/de not_active Expired - Fee Related
- 1998-12-30 PT PT98124819T patent/PT928793E/pt unknown
- 1998-12-30 MA MA25410A patent/MA26590A1/fr unknown
- 1998-12-30 CO CO98077474A patent/CO4990935A1/es unknown
- 1998-12-30 AT AT98124819T patent/ATE217621T1/de not_active IP Right Cessation
- 1998-12-30 ES ES98124819T patent/ES2176895T3/es not_active Expired - Lifetime
- 1998-12-31 BR BR9805750-2A patent/BR9805750A/pt not_active Application Discontinuation
- 1998-12-31 UY UY25335A patent/UY25335A1/es not_active IP Right Cessation
- 1998-12-31 CN CN98125981A patent/CN1098849C/zh not_active Expired - Fee Related
-
1999
- 1999-01-04 ID IDP990002A patent/ID21878A/id unknown
- 1999-01-04 JP JP00020699A patent/JP3154982B2/ja not_active Expired - Fee Related
- 1999-01-05 RU RU99100205/04A patent/RU2166503C2/ru not_active IP Right Cessation
-
2000
- 2000-01-31 HK HK00100585A patent/HK1021733A1/xx not_active IP Right Cessation
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