NO20092049L - Nye fenylsulfamoylbenzamidderivater som bradykininantagonister - Google Patents

Nye fenylsulfamoylbenzamidderivater som bradykininantagonister

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Publication number
NO20092049L
NO20092049L NO20092049A NO20092049A NO20092049L NO 20092049 L NO20092049 L NO 20092049L NO 20092049 A NO20092049 A NO 20092049A NO 20092049 A NO20092049 A NO 20092049A NO 20092049 L NO20092049 L NO 20092049L
Authority
NO
Norway
Prior art keywords
novel
derivatives
phenylsulfamoylbenzamide
bradykinin antagonists
bradykinin
Prior art date
Application number
NO20092049A
Other languages
English (en)
Norwegian (no)
Inventor
Sandor Farkas
Eva Schmidt
Istvan Vago
Gyorgy Keseru
Eva Bozo
Gyula Beke
Katalin Hornok
Eva Szentirmay
Monika Vastag
Original Assignee
Richter Gedeon Nyrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Nyrt filed Critical Richter Gedeon Nyrt
Publication of NO20092049L publication Critical patent/NO20092049L/no

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    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/21—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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    • A61K31/18—Sulfonamides
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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NO20092049A 2006-10-27 2009-05-26 Nye fenylsulfamoylbenzamidderivater som bradykininantagonister NO20092049L (no)

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HU0600809A HUP0600809A3 (en) 2006-10-27 2006-10-27 New phenylsulfamoyl-benzamide derivatives as bradykinin antagonists, process and intermediates for their preparation and pharmaceutical compositions containing them
PCT/HU2007/000103 WO2008050167A1 (fr) 2006-10-27 2007-10-27 Nouveaux dérivés de phénylsulfamoyl-benzamide utilisés come antagonistes de la bradyquinine

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HUP0600808A3 (en) * 2006-10-27 2008-09-29 Richter Gedeon Nyrt New benzamide derivatives as bradykinin antagonists, process for their preparation and pharmaceutical compositions containing them
HUP0600810A3 (en) * 2006-10-27 2008-09-29 Richter Gedeon Nyrt New sulfonamide derivatives as bradykinin antagonists, process and intermediates for their preparation and pharmaceutical compositions containing them
WO2009027450A1 (fr) 2007-08-29 2009-03-05 Boehringer Ingelheim International Gmbh Nouveaux antagonistes de la bradykinine b1
US20100298299A1 (en) * 2007-10-27 2010-11-25 Istvan Vago non-peptide derivatives as bradykinin b1 antagonists
EP2330899A1 (fr) * 2008-08-21 2011-06-15 Richter Gedeon Nyrt. Procédé de traitement de douleur neuropathique
US20100048630A1 (en) * 2008-08-21 2010-02-25 Pradeep Banerjee Methods for treating cns disorders
HU230067B1 (hu) * 2008-12-17 2015-06-29 Richter Gedeon Nyrt Új piperazin só és eljárás előállítására
CN102414177B (zh) * 2009-02-26 2014-07-02 贝林格尔.英格海姆国际有限公司 作为缓激肽b1拮抗剂的化合物
CA2790952C (fr) * 2010-02-23 2017-07-04 Boehringer Ingelheim International Gmbh Composes en tant qu'antagonistes de la bradykinine b1
US8937073B2 (en) 2010-08-20 2015-01-20 Boehringer Ingelheim International Gmbh Disubstituted tetrahydrofuranyl compounds and their use as B1-receptor antagonists
CN104151248B (zh) * 2014-07-17 2016-02-17 陕西师范大学 双咪唑丹磺酰衍生物阳离子型荧光探针及其合成方法和应用
CN104693075B (zh) * 2015-02-13 2016-05-11 程涛 p18小分子抑制剂及在人造血干细胞体外扩增中的用途
CN106601606B (zh) * 2015-10-19 2019-09-20 中芯国际集成电路制造(上海)有限公司 Nmos器件、半导体装置及其制造方法
TW202202495A (zh) 2020-03-26 2022-01-16 匈牙利商羅特格登公司 作為ｇａｍｍａ－胺基丁酸Ａ受體次單元ａｌｐｈａ ５受體調節劑之㖠啶及吡啶并〔３，４－ｃ〕嗒𠯤衍生物
KR20210150011A (ko) * 2020-06-03 2021-12-10 주식회사 삼오파마켐 프로베네시드 및 아르기닌의 아미드 유도체, 이를 포함하는 약제학적 조성물 및 이의 제조 방법
HUP2100338A1 (hu) 2021-09-29 2023-04-28 Richter Gedeon Nyrt GABAA ALFA5 receptor modulátor hatású biciklusos aminszármazékok

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BR9814645A (pt) * 1997-11-18 2001-07-31 Teijin Ltd Derivados de amina cìclica e seu uso como medicamentos
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FR2822827B1 (fr) * 2001-03-28 2003-05-16 Sanofi Synthelabo Nouveaux derives de n-(arylsulfonyl) beta-aminoacides comportant un groupe aminomethyle substitue, leur procede de preparation et les compositions pharmaceutiques en contenant
SI1409477T1 (sl) * 2001-07-24 2009-02-28 Richter Gedeon Nyrt Derivati piperidina kot antagonisti nmda-receptorjev
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HU230518B1 (hu) * 2005-12-20 2016-10-28 Richter Gedeon Nyrt. Bradykinin B1 receptor szelektív antagonista hatással rendelkező új fenatridin származékok, eljárás előállításukra, és az ezeket tartalmazó gyógyszerkészítmények
HUP0600810A3 (en) * 2006-10-27 2008-09-29 Richter Gedeon Nyrt New sulfonamide derivatives as bradykinin antagonists, process and intermediates for their preparation and pharmaceutical compositions containing them
HUP0600808A3 (en) * 2006-10-27 2008-09-29 Richter Gedeon Nyrt New benzamide derivatives as bradykinin antagonists, process for their preparation and pharmaceutical compositions containing them
US20100298299A1 (en) * 2007-10-27 2010-11-25 Istvan Vago non-peptide derivatives as bradykinin b1 antagonists
EP2330899A1 (fr) * 2008-08-21 2011-06-15 Richter Gedeon Nyrt. Procédé de traitement de douleur neuropathique
US20100048630A1 (en) * 2008-08-21 2010-02-25 Pradeep Banerjee Methods for treating cns disorders

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KR20090076926A (ko) 2009-07-13
MX2009004528A (es) 2009-07-02
EA018032B1 (ru) 2013-05-30
EA200900605A1 (ru) 2009-08-28
HU0600809D0 (en) 2006-12-28
HUP0600809A3 (en) 2008-09-29
EP2057116A1 (fr) 2009-05-13
MA30912B1 (fr) 2009-11-02
US20100105686A1 (en) 2010-04-29
CN101528680A (zh) 2009-09-09
HUP0600809A2 (en) 2008-08-28
JP2010507643A (ja) 2010-03-11
GEP20125393B (en) 2012-02-10
NZ575765A (en) 2011-12-22
BRPI0718494A2 (pt) 2014-01-21
AU2007310587A1 (en) 2008-05-02
CA2667481C (fr) 2012-09-25
EP2057116B1 (fr) 2013-02-13
CA2667481A1 (fr) 2008-05-02
WO2008050167A1 (fr) 2008-05-02
US20130029991A1 (en) 2013-01-31
MY155039A (en) 2015-08-28
IL197586A0 (en) 2009-12-24
TN2009000108A1 (en) 2010-08-19

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