NO20091678L - Modulatorer av glucokortikoidreseptoren, AP-1, og/eller NF-kappaB aktivitet og deres anvendelse - Google Patents

Modulatorer av glucokortikoidreseptoren, AP-1, og/eller NF-kappaB aktivitet og deres anvendelse

Info

Publication number
NO20091678L
NO20091678L NO20091678A NO20091678A NO20091678L NO 20091678 L NO20091678 L NO 20091678L NO 20091678 A NO20091678 A NO 20091678A NO 20091678 A NO20091678 A NO 20091678A NO 20091678 L NO20091678 L NO 20091678L
Authority
NO
Norway
Prior art keywords
glucocorticoid receptor
modulators
kappab activity
activity
nr1b
Prior art date
Application number
NO20091678A
Other languages
English (en)
Norwegian (no)
Inventor
T G Murali Dhar
Bingwei Vera Yang
James E Sheppeck
John L Gilmore
Hai-Yun Xiao
Jianmin Wang
Lidia M Doweyko
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20091678L publication Critical patent/NO20091678L/no

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    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
NO20091678A 2006-11-01 2009-04-28 Modulatorer av glucokortikoidreseptoren, AP-1, og/eller NF-kappaB aktivitet og deres anvendelse NO20091678L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US85595306P 2006-11-01 2006-11-01
PCT/US2007/083085 WO2008057857A1 (en) 2006-11-01 2007-10-31 MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-ϰB ACTIVITY AND USE THEREOF

Publications (1)

Publication Number Publication Date
NO20091678L true NO20091678L (no) 2009-05-29

Family

ID=39111670

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20091678A NO20091678L (no) 2006-11-01 2009-04-28 Modulatorer av glucokortikoidreseptoren, AP-1, og/eller NF-kappaB aktivitet og deres anvendelse

Country Status (6)

Country Link
US (1) US8198311B2 (de)
EP (1) EP2099767A1 (de)
JP (1) JP2010508358A (de)
CN (1) CN101573340A (de)
NO (1) NO20091678L (de)
WO (1) WO2008057857A1 (de)

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US10118890B2 (en) 2014-10-10 2018-11-06 The Research Foundation For The State University Of New York Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration
JP6991993B2 (ja) 2015-12-14 2022-01-13 トレベナ・インコーポレイテッド 痛覚過敏を治療する方法
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CN113087696A (zh) * 2019-12-23 2021-07-09 江苏开元药业有限公司 喹啉类化合物及其应用

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US20100075961A1 (en) 2010-03-25
US8198311B2 (en) 2012-06-12

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