NO20083630L - Nye pyridinderivater - Google Patents
Nye pyridinderivaterInfo
- Publication number
- NO20083630L NO20083630L NO20083630A NO20083630A NO20083630L NO 20083630 L NO20083630 L NO 20083630L NO 20083630 A NO20083630 A NO 20083630A NO 20083630 A NO20083630 A NO 20083630A NO 20083630 L NO20083630 L NO 20083630L
- Authority
- NO
- Norway
- Prior art keywords
- pyridine derivatives
- new pyridine
- new
- compounds
- preparation
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4436—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A—HUMAN NECESSITIES
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- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P11/02—Nasal agents, e.g. decongestants
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- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pulmonology (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Dermatology (AREA)
- Neurology (AREA)
- Urology & Nephrology (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Oncology (AREA)
- Ophthalmology & Optometry (AREA)
- Endocrinology (AREA)
- Biomedical Technology (AREA)
- Cardiology (AREA)
- Reproductive Health (AREA)
- Obesity (AREA)
- Communicable Diseases (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychology (AREA)
- Pregnancy & Childbirth (AREA)
- Vascular Medicine (AREA)
- Emergency Medicine (AREA)
- Transplantation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IB2006050260 | 2006-01-24 | ||
| PCT/IB2007/050225 WO2007086001A2 (en) | 2006-01-24 | 2007-01-23 | Novel pyridine derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20083630L true NO20083630L (no) | 2008-10-10 |
Family
ID=38068825
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20083630A NO20083630L (no) | 2006-01-24 | 2008-08-22 | Nye pyridinderivater |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US8178562B2 (pl) |
| EP (1) | EP1979345B1 (pl) |
| JP (1) | JP5063615B2 (pl) |
| KR (1) | KR20080092385A (pl) |
| CN (1) | CN101370805B (pl) |
| AT (1) | ATE447568T1 (pl) |
| AU (1) | AU2007209051A1 (pl) |
| BR (1) | BRPI0706725A2 (pl) |
| CA (1) | CA2635124C (pl) |
| DE (1) | DE602007003074D1 (pl) |
| ES (1) | ES2335242T3 (pl) |
| IL (1) | IL192948A0 (pl) |
| NO (1) | NO20083630L (pl) |
| PL (1) | PL1979345T3 (pl) |
| RU (1) | RU2008134423A (pl) |
| WO (1) | WO2007086001A2 (pl) |
| ZA (1) | ZA200807274B (pl) |
Families Citing this family (38)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2533587A1 (en) | 2002-07-30 | 2004-02-05 | University Of Virginia Patent Foundation | Compounds active in sphingosine 1-phosphate signaling |
| WO2005041899A2 (en) | 2003-11-03 | 2005-05-12 | University Of Virginia Patent Foundation | Orally available sphingosine 1-phosphate receptor agonists and antagonists |
| JP4678139B2 (ja) * | 2004-05-10 | 2011-04-27 | トヨタ自動車株式会社 | 自動車の暖房制御システム |
| MX2007009848A (es) | 2005-02-14 | 2008-03-10 | Univ Virginia | Agonistas de esfingosina 1-fosfato comprendiendo cicloalcanos y heterociclos de 5 miembros substituidos por grupos amino y fenilo. |
| KR101382733B1 (ko) | 2005-03-23 | 2014-04-14 | 액테리온 파마슈티칼 리미티드 | 면역조절물질로서의 수첨 벤조(ｃ) 티오펜 유도체 |
| AU2006226022A1 (en) | 2005-03-23 | 2006-09-28 | Actelion Pharmaceuticals Ltd. | Novel thiophene derivatives as sphingosine-1-phosphate-1 receptor agonists |
| WO2006100633A1 (en) * | 2005-03-23 | 2006-09-28 | Actelion Pharmaceuticals Ltd | NOVEL THIOPHENE DERIVATIVES AS SPHINGOSINE-l-PHOSPHATE-1 RECEPTOR AGONISTS |
| KR20080024533A (ko) * | 2005-06-24 | 2008-03-18 | 액테리온 파마슈티칼 리미티드 | 신규한 티오펜 유도체 |
| AR057894A1 (es) * | 2005-11-23 | 2007-12-26 | Actelion Pharmaceuticals Ltd | Derivados de tiofeno |
| AU2007209961A1 (en) | 2006-01-27 | 2007-08-09 | University Of Virginia Patent Foundation | Method for treatment of neuropathic pain |
| JP2009526073A (ja) | 2006-02-09 | 2009-07-16 | ユニバーシティ オブ バージニア パテント ファンデーション | 二環式スフィンゴシン−１−リン酸受容体アナログ |
| AR061841A1 (es) * | 2006-09-07 | 2008-09-24 | Actelion Pharmaceuticals Ltd | Derivados de tiofen-oxadiazoles, agonistas del receptor s1p1/edg1, composiciones farmaceuticas que los contienen y usos como agentes inmunomoduladores. |
| ES2400533T3 (es) * | 2006-09-07 | 2013-04-10 | Actelion Pharmaceuticals Ltd. | Derivados de piridin 4-ilo como agentes inmunomoduladores |
| MY150661A (en) * | 2006-09-08 | 2014-02-14 | Actelion Pharmaceuticals Ltd | Pyridin-3-yl derivatives as immunomodulating agents |
| WO2008064320A2 (en) | 2006-11-21 | 2008-05-29 | University Of Virginia Patent Foundation | Hydrindane analogs having sphingosine 1-phosphate receptor agonist activity |
| CA2669102A1 (en) | 2006-11-21 | 2008-05-29 | University Of Virginia Patent Foundation | Tetralin analogs having sphingosine 1-phosphate agonist activity |
| WO2008064337A2 (en) | 2006-11-21 | 2008-05-29 | University Of Virginia Patent Foundation | Benzocycloheptyl analogs having sphingosine 1-phosphate receptor activity |
| ES2450750T3 (es) * | 2007-03-16 | 2014-03-25 | Actelion Pharmaceuticals Ltd. | Derivados de amino-piridina como agonistas del receptor S1P1/EDG1 |
| NZ583957A (en) * | 2007-08-17 | 2011-09-30 | Actelion Pharmaceuticals Ltd | Pyridine derivatives as s1p1/edg1 receptor modulators |
| TW200930363A (en) * | 2007-12-10 | 2009-07-16 | Actelion Pharmaceuticals Ltd | Novel thiophene derivatives |
| WO2009109906A1 (en) * | 2008-03-06 | 2009-09-11 | Actelion Pharmaceuticals Ltd | Pyridine compounds |
| NZ588438A (en) * | 2008-03-07 | 2012-05-25 | Actelion Pharmaceuticals Ltd | Pyridin-2-yl oxadiazole derivatives as immunomodulating agents |
| MY177360A (en) | 2008-03-17 | 2020-09-14 | Actelion Pharmaceuticals Ltd | Dosing regimen for aselective s1p1 receptor agonist |
| SI2326621T1 (sl) | 2008-07-23 | 2016-10-28 | Arena Pharmaceuticals, Inc. | Substituirani derivati 1,2,3,4-tetrahidrociklopenta(b)indol-3-il)ocetne kisline, uporabni pri zdravljenju avtoimunskih in vnetnih motenj |
| SI2342205T1 (sl) | 2008-08-27 | 2016-09-30 | Arena Pharmaceuticals, Inc. | Substituirani triciklični kislinski derivati kot agonisti S1P1 receptorja, uporabni v zdravljenju avtoimunskih in vnetnih obolenj |
| ES2441845T3 (es) | 2009-07-16 | 2014-02-06 | Actelion Pharmaceuticals Ltd. | Derivados de piridin-4-ilo como agonistas de S1P1/EDG1 |
| JP5856980B2 (ja) | 2010-01-27 | 2016-02-10 | アリーナ ファーマシューティカルズ， インコーポレイテッド | （Ｒ）−２−（７−（４−シクロペンチル−３−（トリフルオロメチル）ベンジルオキシ）−１，２，３，４−テトラヒドロシクロペンタ［ｂ］インドール−３−イル）酢酸およびその塩の調製のためのプロセス |
| SG10201501575VA (en) | 2010-03-03 | 2015-04-29 | Arena Pharm Inc | Processes for the preparation of s1p1 receptor modulators and crystalline forms thereof |
| ES2544086T3 (es) | 2011-01-19 | 2015-08-27 | Actelion Pharmaceuticals Ltd. | Derivados de 2-metoxi-piridin-4-ilo |
| LT2885266T (lt) | 2012-08-17 | 2020-07-10 | Actelion Pharmaceuticals Ltd | (2z,5z)-5-(3-chlor-4-((r)-2,3-dihidroksipropoksi)benziliden)-2-(propilimino)-3-(o-tolil)tiazolidin-4-ono gamybos būdas ir šiame procese naudojamas tarpinis junginys |
| WO2014029722A1 (en) | 2012-08-21 | 2014-02-27 | F. Hoffmann-La Roche Ag | Novel pyridine derivatives |
| CN107405332A (zh) | 2015-01-06 | 2017-11-28 | 艾尼纳制药公司 | 治疗与s1p1受体有关的病症的方法 |
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2007
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- 2007-01-23 DE DE602007003074T patent/DE602007003074D1/de active Active
- 2007-01-23 CN CN2007800028024A patent/CN101370805B/zh not_active Expired - Fee Related
- 2007-01-23 AU AU2007209051A patent/AU2007209051A1/en not_active Abandoned
- 2007-01-23 KR KR1020087018084A patent/KR20080092385A/ko not_active Application Discontinuation
- 2007-01-23 WO PCT/IB2007/050225 patent/WO2007086001A2/en active Application Filing
- 2007-01-23 PL PL07700666T patent/PL1979345T3/pl unknown
- 2007-01-23 RU RU2008134423/04A patent/RU2008134423A/ru not_active Application Discontinuation
- 2007-01-23 BR BRPI0706725-9A patent/BRPI0706725A2/pt not_active IP Right Cessation
- 2007-01-23 EP EP07700666A patent/EP1979345B1/en active Active
- 2007-01-23 ES ES07700666T patent/ES2335242T3/es active Active
- 2007-01-23 CA CA2635124A patent/CA2635124C/en not_active Expired - Fee Related
- 2007-01-23 AT AT07700666T patent/ATE447568T1/de active
- 2007-01-23 JP JP2008550900A patent/JP5063615B2/ja not_active Expired - Fee Related
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2008
- 2008-07-22 IL IL192948A patent/IL192948A0/en unknown
- 2008-08-22 NO NO20083630A patent/NO20083630L/no not_active Application Discontinuation
- 2008-08-22 ZA ZA200807274A patent/ZA200807274B/xx unknown
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Also Published As
| Publication number | Publication date |
|---|---|
| ATE447568T1 (de) | 2009-11-15 |
| EP1979345B1 (en) | 2009-11-04 |
| ZA200807274B (en) | 2009-11-25 |
| US8178562B2 (en) | 2012-05-15 |
| JP5063615B2 (ja) | 2012-10-31 |
| WO2007086001A2 (en) | 2007-08-02 |
| WO2007086001A3 (en) | 2008-04-03 |
| DE602007003074D1 (de) | 2009-12-17 |
| BRPI0706725A2 (pt) | 2011-04-05 |
| CN101370805A (zh) | 2009-02-18 |
| CA2635124A1 (en) | 2007-08-02 |
| KR20080092385A (ko) | 2008-10-15 |
| IL192948A0 (en) | 2009-08-03 |
| AU2007209051A1 (en) | 2007-08-02 |
| JP2009524603A (ja) | 2009-07-02 |
| CA2635124C (en) | 2014-04-29 |
| PL1979345T3 (pl) | 2010-04-30 |
| EP1979345A2 (en) | 2008-10-15 |
| US20120195930A1 (en) | 2012-08-02 |
| US20090005421A1 (en) | 2009-01-01 |
| ES2335242T3 (es) | 2010-03-23 |
| RU2008134423A (ru) | 2010-02-27 |
| US8697732B2 (en) | 2014-04-15 |
| CN101370805B (zh) | 2011-04-27 |
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