NO20080083L - Thiomorfolin-forbindelse og framgangsmate for framstilling av samme - Google Patents

Thiomorfolin-forbindelse og framgangsmate for framstilling av samme

Info

Publication number
NO20080083L
NO20080083L NO20080083A NO20080083A NO20080083L NO 20080083 L NO20080083 L NO 20080083L NO 20080083 A NO20080083 A NO 20080083A NO 20080083 A NO20080083 A NO 20080083A NO 20080083 L NO20080083 L NO 20080083L
Authority
NO
Norway
Prior art keywords
optionally substituted
same
group
hydrogen atom
alkyl group
Prior art date
Application number
NO20080083A
Other languages
English (en)
Inventor
Masami Takahashi
Takeshi Yamanaka
Tsutomu Miyake
Original Assignee
Mitsubishi Tanabe Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Tanabe Pharma Corp filed Critical Mitsubishi Tanabe Pharma Corp
Publication of NO20080083L publication Critical patent/NO20080083L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
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    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Virology (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Otolaryngology (AREA)
  • Addiction (AREA)
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Abstract

Thiomorfolinforbindelse representert ved formelen (I), der Ring A representerer en valgfritt substituert benzenring; Ring B representerer en valgfritt substituert benzenring; R1 representerer et hydrogenatom, en valgfritt substituert hydroksylgruppe, en valgfritt substituert amingruppe, en valgfritt substituert alkylgruppe, en substituert karbonylgruppe eller et halogenatom; R2 representerer et hydrogenatom eller en valgfritt substituert alkylgruppe; R3a og R3b kan være like eller forskjellige og representerer hver et hydrogenatom eller en valgfritt substituert alkylgruppe, eller kombinert med hverandre ved begge ender av samme for å danne en alkylengruppe, og n er et heltall lik 1 eller 2, eller et farmasøytisk akseptabelt salt av samme.
NO20080083A 2005-09-01 2008-01-07 Thiomorfolin-forbindelse og framgangsmate for framstilling av samme NO20080083L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2005253105 2005-09-01
PCT/JP2006/317798 WO2007026966A1 (en) 2005-09-01 2006-09-01 Thiomorpholine compound and process for preparing the same

Publications (1)

Publication Number Publication Date
NO20080083L true NO20080083L (no) 2008-05-20

Family

ID=37809039

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20080083A NO20080083L (no) 2005-09-01 2008-01-07 Thiomorfolin-forbindelse og framgangsmate for framstilling av samme

Country Status (17)

Country Link
US (1) US20090281095A1 (no)
EP (1) EP1954677B1 (no)
KR (1) KR20080041733A (no)
CN (1) CN101233106A (no)
AR (1) AR056048A1 (no)
AU (1) AU2006285614B2 (no)
BR (1) BRPI0615045A2 (no)
CA (1) CA2620742A1 (no)
DE (1) DE602006015845D1 (no)
ES (1) ES2347002T3 (no)
IL (1) IL189698A0 (no)
NO (1) NO20080083L (no)
NZ (1) NZ566428A (no)
RU (1) RU2379305C2 (no)
TW (1) TW200740782A (no)
WO (1) WO2007026966A1 (no)
ZA (1) ZA200802814B (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2710293A1 (en) * 2007-12-20 2009-07-02 Teva Women's Health, Inc. Dosage regimens and pharmaceutical compositions and packages for emergency contraception
GB0812849D0 (en) * 2008-07-14 2008-08-20 Glaxo Wellcome Mfg Pte Ltd Novel compounds
CN106397356B (zh) * 2016-08-31 2019-08-13 郑州原理生物科技有限公司 硫代吗啉-1,1-二氧化物盐酸盐的制备方法，硫代吗啉-1,1-二氧化物的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4263433A (en) * 1976-08-12 1981-04-21 Petrolite Corporation Tertiary amino-substituted thiazines
TWI283241B (en) * 2002-05-29 2007-07-01 Tanabe Seiyaku Co Novel piperidine compound
JP4389478B2 (ja) * 2002-05-29 2009-12-24 田辺三菱製薬株式会社 新規ピペリジン誘導体

Also Published As

Publication number Publication date
AU2006285614B2 (en) 2010-02-18
KR20080041733A (ko) 2008-05-13
AU2006285614A1 (en) 2007-03-08
TW200740782A (en) 2007-11-01
ZA200802814B (en) 2009-11-25
EP1954677A1 (en) 2008-08-13
AR056048A1 (es) 2007-09-12
IL189698A0 (en) 2008-06-05
RU2379305C2 (ru) 2010-01-20
RU2008112310A (ru) 2009-10-10
DE602006015845D1 (de) 2010-09-09
BRPI0615045A2 (pt) 2011-04-26
US20090281095A1 (en) 2009-11-12
WO2007026966A1 (en) 2007-03-08
CN101233106A (zh) 2008-07-30
EP1954677A4 (en) 2009-06-17
NZ566428A (en) 2010-04-30
ES2347002T3 (es) 2010-10-22
CA2620742A1 (en) 2007-03-08
EP1954677B1 (en) 2010-07-28

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