NO20074002L - Androgen reseptor-modulatorforbindelser og fremgangsmater - Google Patents

Androgen reseptor-modulatorforbindelser og fremgangsmater

Info

Publication number
NO20074002L
NO20074002L NO20074002A NO20074002A NO20074002L NO 20074002 L NO20074002 L NO 20074002L NO 20074002 A NO20074002 A NO 20074002A NO 20074002 A NO20074002 A NO 20074002A NO 20074002 L NO20074002 L NO 20074002L
Authority
NO
Norway
Prior art keywords
methods
androgen receptor
receptor modulator
modulator compounds
compounds
Prior art date
Application number
NO20074002A
Other languages
English (en)
Norwegian (no)
Inventor
Lin Zhi
Bijan Pedram
Cornelis A Van Oeveren
Shuo Zhao
Yixing Shen
Original Assignee
Ligand Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ligand Pharm Inc filed Critical Ligand Pharm Inc
Publication of NO20074002L publication Critical patent/NO20074002L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Obesity (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Dermatology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pregnancy & Childbirth (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Anesthesiology (AREA)
NO20074002A 2005-06-17 2007-08-01 Androgen reseptor-modulatorforbindelser og fremgangsmater NO20074002L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69189105P 2005-06-17 2005-06-17
PCT/US2006/023111 WO2006138347A2 (en) 2005-06-17 2006-06-12 Androgen receptor modulator compounds and methods

Publications (1)

Publication Number Publication Date
NO20074002L true NO20074002L (no) 2008-03-10

Family

ID=37546607

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20074002A NO20074002L (no) 2005-06-17 2007-08-01 Androgen reseptor-modulatorforbindelser og fremgangsmater

Country Status (14)

Country Link
US (2) US8193357B2 (ja)
EP (1) EP1891067B1 (ja)
JP (1) JP5199079B2 (ja)
KR (1) KR101293935B1 (ja)
CN (1) CN101137655A (ja)
AR (2) AR054783A1 (ja)
AU (1) AU2006259474B2 (ja)
BR (1) BRPI0609191B8 (ja)
CA (1) CA2598216C (ja)
IL (1) IL185003A (ja)
MX (1) MX2007009784A (ja)
NO (1) NO20074002L (ja)
NZ (1) NZ560354A (ja)
WO (1) WO2006138347A2 (ja)

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US7026484B2 (en) * 2001-02-23 2006-04-11 Ligand Pharmaceuticals Incorporated Tricyclic androgen receptor modulator compounds and methods
WO2005090282A1 (en) 2004-03-12 2005-09-29 Ligand Pharmaceuticals Incorporated Androgen receptor modulator compounds and methods
CA2598216C (en) 2005-06-17 2014-04-08 Ligand Pharmaceuticals Incorporated Androgen receptor modulator compounds and methods
CA2709677C (en) 2007-12-21 2017-03-14 Lin Zhi Selective androgen receptor modulators (sarms) and uses thereof
AR072297A1 (es) 2008-06-27 2010-08-18 Novartis Ag Derivados de indol-2-il-piridin-3-ilo, composicion farmaceutica que los comprende y su uso en medicamentos para el tratamiento de enfermedades mediadas por la sintasa aldosterona.
BR112013023062B1 (pt) 2011-03-10 2022-01-18 Xeris Pharmaceuticals, Inc Solução estável para a injeção parenteral e método de fabricação da mesma
US9125805B2 (en) 2012-06-27 2015-09-08 Xeris Pharmaceuticals, Inc. Stable formulations for parenteral injection of small molecule drugs
AU2013315510B2 (en) 2012-09-11 2019-08-22 Visa International Service Association Cloud-based Virtual Wallet NFC Apparatuses, methods and systems
AU2015300944B2 (en) 2014-08-06 2019-07-11 Xeris Pharmaceuticals, Inc. Syringes, kits, and methods for intracutaneous and/or subcutaneous injection of pastes
CN104856996B (zh) * 2015-04-27 2018-01-05 南京舒鹏生物科技有限公司 吡咯喹啉醌、其衍生物和/或盐新的药用用途以及药用组合物
US9649364B2 (en) 2015-09-25 2017-05-16 Xeris Pharmaceuticals, Inc. Methods for producing stable therapeutic formulations in aprotic polar solvents
US11590205B2 (en) 2015-09-25 2023-02-28 Xeris Pharmaceuticals, Inc. Methods for producing stable therapeutic glucagon formulations in aprotic polar solvents
US11040973B2 (en) 2017-03-29 2021-06-22 Purdue Research Foundation Inhibitors of kinase networks and uses thereof
CN110709061B (zh) 2017-06-02 2023-09-08 Xeris药物公司 抗沉淀的小分子药物制剂
EP4175637A4 (en) * 2020-07-02 2024-08-07 Purdue Research Foundation TETRAHYDRO-3H-PYRAZOLOQUINOLONE AND TETRAHYDRO-3H-PYRROLO[3,2-F QUINOLINE-CONTAINING COMPOUNDS AND USES THEREOF
TW202214632A (zh) * 2020-07-27 2022-04-16 大陸商江蘇恆瑞醫藥股份有限公司 吲哚稠環類衍生物、其製備方法及其在醫藥上的應用

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KR20080020592A (ko) 2008-03-05
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EP1891067A2 (en) 2008-02-27
BRPI0609191B8 (pt) 2021-05-25
BRPI0609191A2 (pt) 2010-03-02
US20120165362A1 (en) 2012-06-28
US8193357B2 (en) 2012-06-05
US8580811B2 (en) 2013-11-12
IL185003A (en) 2015-06-30
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