IL185003A0 - Androgen receptor modulator compounds and methods - Google Patents

Androgen receptor modulator compounds and methods

Info

Publication number
IL185003A0
IL185003A0 IL185003A IL18500307A IL185003A0 IL 185003 A0 IL185003 A0 IL 185003A0 IL 185003 A IL185003 A IL 185003A IL 18500307 A IL18500307 A IL 18500307A IL 185003 A0 IL185003 A0 IL 185003A0
Authority
IL
Israel
Prior art keywords
methods
androgen receptor
receptor modulator
modulator compounds
compounds
Prior art date
Application number
IL185003A
Other versions
IL185003A (en
Original Assignee
Ligand Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ligand Pharm Inc filed Critical Ligand Pharm Inc
Publication of IL185003A0 publication Critical patent/IL185003A0/en
Publication of IL185003A publication Critical patent/IL185003A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Immunology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pregnancy & Childbirth (AREA)
  • Emergency Medicine (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
IL185003A 2005-06-17 2007-08-02 9-chloro-hydropyrrolo[3,2-f]quinolin-7(6h)-one derivatives and pharmaceutical compositions thereof IL185003A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69189105P 2005-06-17 2005-06-17
PCT/US2006/023111 WO2006138347A2 (en) 2005-06-17 2006-06-12 Androgen receptor modulator compounds and methods

Publications (2)

Publication Number Publication Date
IL185003A0 true IL185003A0 (en) 2007-12-03
IL185003A IL185003A (en) 2015-06-30

Family

ID=37546607

Family Applications (1)

Application Number Title Priority Date Filing Date
IL185003A IL185003A (en) 2005-06-17 2007-08-02 9-chloro-hydropyrrolo[3,2-f]quinolin-7(6h)-one derivatives and pharmaceutical compositions thereof

Country Status (14)

Country Link
US (2) US8193357B2 (en)
EP (1) EP1891067B1 (en)
JP (1) JP5199079B2 (en)
KR (1) KR101293935B1 (en)
CN (1) CN101137655A (en)
AR (2) AR054783A1 (en)
AU (1) AU2006259474B2 (en)
BR (1) BRPI0609191B8 (en)
CA (1) CA2598216C (en)
IL (1) IL185003A (en)
MX (1) MX2007009784A (en)
NO (1) NO20074002L (en)
NZ (1) NZ560354A (en)
WO (1) WO2006138347A2 (en)

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KR101293935B1 (en) 2005-06-17 2013-08-08 리간드 파마슈티칼스 인코포레이티드 Androgen receptor modulator compounds and methods
PL2222636T3 (en) 2007-12-21 2014-04-30 Ligand Pharm Inc Selective androgen receptor modulators (sarms) and uses thereof
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CN104856996B (en) * 2015-04-27 2018-01-05 南京舒鹏生物科技有限公司 PQQ, its derivative and/or the new pharmaceutical usage and Pharmaceutical composition of salt
US9649364B2 (en) 2015-09-25 2017-05-16 Xeris Pharmaceuticals, Inc. Methods for producing stable therapeutic formulations in aprotic polar solvents
US11590205B2 (en) 2015-09-25 2023-02-28 Xeris Pharmaceuticals, Inc. Methods for producing stable therapeutic glucagon formulations in aprotic polar solvents
CN110662536B (en) 2017-03-29 2023-06-23 普渡研究基金会 Kinase network inhibitors and uses thereof
AU2018275686B2 (en) 2017-06-02 2024-02-01 Xeris Pharmaceuticals, Inc. Precipitation resistant small molecule drug formulations
US20230312562A1 (en) * 2020-07-02 2023-10-05 Purdue Research Foundation Tetrahydro-3h-pyrazolo quinolone and tetrahydro-3h-pyrrolo[3,2-f]quinoline -containing compounds and uses thereof
WO2022022489A1 (en) * 2020-07-27 2022-02-03 江苏恒瑞医药股份有限公司 Indole fused ring derivative, preparation method therefor and use thereof in medicine

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US20090030027A1 (en) 2009-01-29
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