NO20074002L - Androgen reseptor-modulatorforbindelser og fremgangsmater - Google Patents

Androgen reseptor-modulatorforbindelser og fremgangsmater

Info

Publication number
NO20074002L
NO20074002L NO20074002A NO20074002A NO20074002L NO 20074002 L NO20074002 L NO 20074002L NO 20074002 A NO20074002 A NO 20074002A NO 20074002 A NO20074002 A NO 20074002A NO 20074002 L NO20074002 L NO 20074002L
Authority
NO
Norway
Prior art keywords
methods
androgen receptor
receptor modulator
modulator compounds
compounds
Prior art date
Application number
NO20074002A
Other languages
English (en)
Inventor
Lin Zhi
Bijan Pedram
Cornelis A Van Oeveren
Shuo Zhao
Yixing Shen
Original Assignee
Ligand Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ligand Pharm Inc filed Critical Ligand Pharm Inc
Publication of NO20074002L publication Critical patent/NO20074002L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Diabetes (AREA)
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  • Obesity (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
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  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pregnancy & Childbirth (AREA)
  • Emergency Medicine (AREA)
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  • Transplantation (AREA)
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  • Urology & Nephrology (AREA)
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Abstract

Det tilveiebringes forbindelser med generell formel (I) som binder til androgenreseptorer og/eller modulerer aktivitet av androgenreseptorer, og fremgangsmåter for fremstilling og anvendelse av slike forbindelser. Det tilveiebringes også preparater som inkluderer slike forbindelser og fremgangsmåter for fremstilling og anvendelse av slike preparater.
NO20074002A 2005-06-17 2007-08-01 Androgen reseptor-modulatorforbindelser og fremgangsmater NO20074002L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69189105P 2005-06-17 2005-06-17
PCT/US2006/023111 WO2006138347A2 (en) 2005-06-17 2006-06-12 Androgen receptor modulator compounds and methods

Publications (1)

Publication Number Publication Date
NO20074002L true NO20074002L (no) 2008-03-10

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ID=37546607

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Application Number Title Priority Date Filing Date
NO20074002A NO20074002L (no) 2005-06-17 2007-08-01 Androgen reseptor-modulatorforbindelser og fremgangsmater

Country Status (14)

Country Link
US (2) US8193357B2 (no)
EP (1) EP1891067B1 (no)
JP (1) JP5199079B2 (no)
KR (1) KR101293935B1 (no)
CN (1) CN101137655A (no)
AR (2) AR054783A1 (no)
AU (1) AU2006259474B2 (no)
BR (1) BRPI0609191B8 (no)
CA (1) CA2598216C (no)
IL (1) IL185003A (no)
MX (1) MX2007009784A (no)
NO (1) NO20074002L (no)
NZ (1) NZ560354A (no)
WO (1) WO2006138347A2 (no)

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CN101137655A (zh) 2005-06-17 2008-03-05 配体药物公司 雄激素受体调节剂化合物和方法
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BR112013023062B1 (pt) 2011-03-10 2022-01-18 Xeris Pharmaceuticals, Inc Solução estável para a injeção parenteral e método de fabricação da mesma
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EP3871709A1 (en) 2014-08-06 2021-09-01 Xeris Pharmaceuticals, Inc. Syringes, kits, and methods for intracutaneous and/or subcutaneous injection of pastes
CN104856996B (zh) * 2015-04-27 2018-01-05 南京舒鹏生物科技有限公司 吡咯喹啉醌、其衍生物和/或盐新的药用用途以及药用组合物
US9649364B2 (en) 2015-09-25 2017-05-16 Xeris Pharmaceuticals, Inc. Methods for producing stable therapeutic formulations in aprotic polar solvents
US11590205B2 (en) 2015-09-25 2023-02-28 Xeris Pharmaceuticals, Inc. Methods for producing stable therapeutic glucagon formulations in aprotic polar solvents
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AU2018275686B2 (en) 2017-06-02 2024-02-01 Xeris Pharmaceuticals, Inc. Precipitation resistant small molecule drug formulations
EP4175637A2 (en) * 2020-07-02 2023-05-10 Purdue Research Foundation Tetrahydro-3h-pyrazolo quinolone and tetrahydro-3h-pyrrolo[3,2-f]quinoline-containing compounds and uses thereof
TW202214632A (zh) * 2020-07-27 2022-04-16 大陸商江蘇恆瑞醫藥股份有限公司 吲哚稠環類衍生物、其製備方法及其在醫藥上的應用

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AU2006259474B2 (en) 2011-10-27
WO2006138347A3 (en) 2007-03-01
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BRPI0609191B1 (pt) 2020-10-13
US8193357B2 (en) 2012-06-05
US20120165362A1 (en) 2012-06-28
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