NO20071967L - Imidazo-benzodiazepinderivater - Google Patents

Imidazo-benzodiazepinderivater

Info

Publication number
NO20071967L
NO20071967L NO20071967A NO20071967A NO20071967L NO 20071967 L NO20071967 L NO 20071967L NO 20071967 A NO20071967 A NO 20071967A NO 20071967 A NO20071967 A NO 20071967A NO 20071967 L NO20071967 L NO 20071967L
Authority
NO
Norway
Prior art keywords
imidazo
benzodiazepine
cognitive
triazolo
gaba
Prior art date
Application number
NO20071967A
Other languages
English (en)
Norwegian (no)
Inventor
Andrew William Thomas
Henner Knust
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO20071967L publication Critical patent/NO20071967L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20071967A 2004-10-20 2007-04-17 Imidazo-benzodiazepinderivater NO20071967L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04105169 2004-10-20
PCT/EP2005/010908 WO2006045430A1 (fr) 2004-10-20 2005-10-11 Derives d'imidazo-benzodiazepine

Publications (1)

Publication Number Publication Date
NO20071967L true NO20071967L (no) 2007-05-14

Family

ID=36035782

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20071967A NO20071967L (no) 2004-10-20 2007-04-17 Imidazo-benzodiazepinderivater

Country Status (18)

Country Link
US (1) US7514426B2 (fr)
EP (1) EP1805184B1 (fr)
JP (1) JP4783375B2 (fr)
KR (1) KR100923399B1 (fr)
CN (1) CN101044145B (fr)
AR (1) AR051395A1 (fr)
AU (1) AU2005299032B2 (fr)
BR (1) BRPI0519991A2 (fr)
CA (1) CA2584259C (fr)
ES (1) ES2399439T3 (fr)
IL (1) IL182585A0 (fr)
MX (1) MX2007004639A (fr)
NO (1) NO20071967L (fr)
NZ (1) NZ554439A (fr)
RU (1) RU2007112940A (fr)
TW (1) TWI303247B (fr)
WO (1) WO2006045430A1 (fr)
ZA (1) ZA200703172B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100923393B1 (ko) * 2004-12-14 2009-10-23 에프. 호프만-라 로슈 아게 Gaba 수용체 조절제로서 테트라사이클릭이미다조-벤조다이아제핀
DE602006016147D1 (en) * 2005-10-11 2010-09-23 Hoffmann La Roche Imidazobenzdiazepinderivate
FR2913886B1 (fr) 2007-03-22 2012-03-02 Guerbet Sa Utilisation de nanoparticules metalliques dans le diagnostique de la maladie d'alzheimer
EP2298296A1 (fr) 2009-08-25 2011-03-23 CNRS Centre National De La Recherche Scientifique Composition et procédé pour le traitement de troubles cognitifs chez des sujets atteints du syndrome de Down
WO2011153377A2 (fr) * 2010-06-03 2011-12-08 The Regents Of The University Of California Procédés et compositions pour le traitement d'un sujet pour une lésion du système nerveux central (snc)
EP2457569A1 (fr) 2010-11-05 2012-05-30 F. Hoffmann-La Roche AG Utilisation de composés pharmaceutiques actifs pour le traitement de conditions du système nerveux central
RU2563167C2 (ru) * 2010-11-05 2015-09-20 Ф. Хоффманн-Ля Рош Аг Применение активных фармацевтических соединений для лечения заболеваний центральной нервной системы
EP2640391B1 (fr) 2010-11-15 2015-11-11 Agenebio, Inc. Dérivés de pyridazine, compositions et méthodes de traitement d'une déficience cognitive
US20150374705A1 (en) 2012-02-14 2015-12-31 Shanghai Institues for Biological Sciences Substances for treatment or relief of pain
EP4032889A1 (fr) * 2013-12-20 2022-07-27 Agenebio, Inc. Dérivés de benzodiazépine, compositions et méthodes de traitement de déficience cognitive
US10815242B2 (en) * 2015-06-19 2020-10-27 Agenebio, Inc. Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
BR112019012821A2 (pt) 2016-12-19 2019-11-26 Agenebio Inc derivados de benzodiazepina, composições e métodos para o tratamento do comprometimento cognitivo
US20180170941A1 (en) * 2016-12-19 2018-06-21 Agenebio, Inc. Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment
EP3810611A4 (fr) 2018-06-19 2022-03-30 Agenebio, Inc. Dérivés de benzodiazépine, compositions, et méthodes de traitement de déficience cognitive

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1143728A (fr) 1979-10-04 1983-03-29 Max Gerecke Derives d'imidazodiazepine
CA1174673A (fr) * 1981-02-27 1984-09-18 Walter Hunkeler Imidazodiazepines
EP0150040B1 (fr) 1984-01-19 1994-08-31 F. Hoffmann-La Roche Ag Dérivés de imidazobenzodiazépine
DK174086D0 (da) * 1986-04-16 1986-04-16 Ferrosan As Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme
ZA881538B (en) * 1987-03-10 1988-09-12 F. Hoffmann-La Roche & Co. Aktiengesellschaft Imidazodiazepine derivatives
US4897392A (en) * 1989-07-03 1990-01-30 Hoechst-Roussel Pharmaceuticals, Inc. 4H-indolo(1,2-d)(1,2,4)triazolo(4,3-A)(1,4)benzodiazepines
TW201311B (fr) * 1991-06-17 1993-03-01 Hoffmann La Roche
TWI239333B (en) 2000-11-16 2005-09-11 Hoffmann La Roche Benzodiazepine derivatives as GABA A receptor modulators
US6686352B2 (en) * 2001-05-18 2004-02-03 Hoffmann-La Roche Inc. Substituted imidazo [1,5-a] pyrimido [5,4-d] [1] benzazepine derivatives

Also Published As

Publication number Publication date
EP1805184B1 (fr) 2013-01-09
US20060084642A1 (en) 2006-04-20
JP4783375B2 (ja) 2011-09-28
AU2005299032B2 (en) 2011-11-17
ES2399439T3 (es) 2013-04-01
NZ554439A (en) 2009-09-25
JP2008517011A (ja) 2008-05-22
AR051395A1 (es) 2007-01-10
AU2005299032A1 (en) 2006-05-04
IL182585A0 (en) 2007-07-24
CA2584259A1 (fr) 2006-05-04
TWI303247B (en) 2008-11-21
BRPI0519991A2 (pt) 2009-04-07
US7514426B2 (en) 2009-04-07
CN101044145A (zh) 2007-09-26
EP1805184A1 (fr) 2007-07-11
RU2007112940A (ru) 2008-11-27
CN101044145B (zh) 2010-06-16
ZA200703172B (en) 2008-08-27
WO2006045430A1 (fr) 2006-05-04
TW200630372A (en) 2006-09-01
KR100923399B1 (ko) 2009-10-23
CA2584259C (fr) 2013-04-02
KR20070054731A (ko) 2007-05-29
MX2007004639A (es) 2007-06-08

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Legal Events

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