NO20071343L - Substituerte fenylaminotiazoler og anvendelse derav - Google Patents

Substituerte fenylaminotiazoler og anvendelse derav

Info

Publication number
NO20071343L
NO20071343L NO20071343A NO20071343A NO20071343L NO 20071343 L NO20071343 L NO 20071343L NO 20071343 A NO20071343 A NO 20071343A NO 20071343 A NO20071343 A NO 20071343A NO 20071343 L NO20071343 L NO 20071343L
Authority
NO
Norway
Prior art keywords
phenylaminothiazoles
substituted
diseases
prevention
preparation
Prior art date
Application number
NO20071343A
Other languages
English (en)
Inventor
Andreas Knorr
Joachim Huetter
Walter Huebsch
Kerstin Henninger
Karl-Heinz Schlemmer
Ulrich Rosentreter
Barbara Albrecht
Peter Nell
Dirk Brohm
Nicole Diedrichs
Jens-Kerim Ergueden
Gunter Karig
Sabine Arndt
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of NO20071343L publication Critical patent/NO20071343L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Foreliggende oppfinnelse angår nye fenylaminotiazol derivater, fremgangsmåter for fremstilling derav, anvendelse derav for behandling og/eller hindring av sykdommer og anvendelse derav for fremstilling av medikamenter anvendt for behandling og/eller hindring av sykdommer, foretrukket hypertensjon og andre kardiovaskulære sykdommer.
NO20071343A 2004-09-03 2007-03-13 Substituerte fenylaminotiazoler og anvendelse derav NO20071343L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004042607A DE102004042607A1 (de) 2004-09-03 2004-09-03 Substituierte Phenylaminothiazole und ihre Verwendung
PCT/EP2005/009316 WO2006027142A1 (de) 2004-09-03 2005-08-30 Substituierte phenylaminothiazole und ihre verwendung

Publications (1)

Publication Number Publication Date
NO20071343L true NO20071343L (no) 2007-05-30

Family

ID=35852458

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20071343A NO20071343L (no) 2004-09-03 2007-03-13 Substituerte fenylaminotiazoler og anvendelse derav

Country Status (24)

Country Link
US (1) US8691850B2 (no)
EP (1) EP1812430B1 (no)
JP (1) JP4999691B2 (no)
KR (1) KR20070057235A (no)
CN (1) CN101056875A (no)
AR (1) AR050551A1 (no)
AT (1) ATE428710T1 (no)
AU (1) AU2005281941A1 (no)
BR (1) BRPI0514833A (no)
CA (1) CA2578596C (no)
DE (2) DE102004042607A1 (no)
EC (1) ECSP077296A (no)
ES (1) ES2324049T3 (no)
GT (1) GT200500238A (no)
IL (1) IL181670A0 (no)
MA (1) MA28869B1 (no)
MX (1) MX2007002470A (no)
NO (1) NO20071343L (no)
PE (1) PE20060589A1 (no)
SV (1) SV2006002218A (no)
TW (1) TW200621765A (no)
UY (1) UY29099A1 (no)
WO (1) WO2006027142A1 (no)
ZA (1) ZA200701820B (no)

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DE102006056740A1 (de) 2006-12-01 2008-06-05 Bayer Healthcare Ag Cyclisch substituierte 3,5-Dicyano-2-thiopyridine und ihre Verwendung
DE102006056739A1 (de) * 2006-12-01 2008-06-05 Bayer Healthcare Ag Substituierte 4-Amino-3,5-dicyano-2-thiopyridine und ihre Verwendung
DE102007035367A1 (de) * 2007-07-27 2009-01-29 Bayer Healthcare Ag Substituierte Aryloxazole und ihre Verwendung
DE102007036076A1 (de) 2007-08-01 2009-02-05 Bayer Healthcare Aktiengesellschaft Dipeptoid-Produgs und ihre Verwendung
DE102007061763A1 (de) * 2007-12-20 2009-06-25 Bayer Healthcare Ag Substituierte azabicyclische Verbindungen und ihre Verwendung
DE102007061764A1 (de) 2007-12-20 2009-06-25 Bayer Healthcare Ag Anellierte Cyanopyridine und ihre Verwendung
DE102008008838A1 (de) 2008-02-13 2009-08-20 Bayer Healthcare Ag Cycloalkoxy-substituierte 4-Phenyl-3,5-dicyanopyridine und ihre Verwendung
DE102008013587A1 (de) * 2008-03-11 2009-09-17 Bayer Schering Pharma Aktiengesellschaft Heteroaryl-substituierte Dicyanopyridine und ihre Verwendung
JP2011520997A (ja) * 2008-05-29 2011-07-21 バイエル・シェーリング・ファルマ・アクチェンゲゼルシャフト ２−アルコキシ置換ジシアノピリジン類およびそれらの使用
DE102008062567A1 (de) 2008-12-16 2010-06-17 Bayer Schering Pharma Aktiengesellschaft Dipeptoid-Prodrugs und ihre Verwendung
DE102009006602A1 (de) * 2009-01-29 2010-08-05 Bayer Schering Pharma Aktiengesellschaft Alkylamino-substituierte Dicyanopyridine und deren Aminosäureester-Prodrugs
DE102009022894A1 (de) * 2009-05-27 2010-12-02 Bayer Schering Pharma Aktiengesellschaft Substituierte Piperidine
DE102010030688A1 (de) 2010-06-30 2012-01-05 Bayer Schering Pharma Aktiengesellschaft Substituierte Dicyanopyridine und ihre Verwendung
KR20220147691A (ko) 2013-08-09 2022-11-03 알데릭스, 인코포레이티드 인산염 수송을 억제하기 위한 화합물 및 방법
WO2018153895A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit einem inhibitor der neutralen endopeptidase und/oder einem angiotensin ii rezeptor-antagonisten
WO2018153898A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit mineralocorticoid-rezeptor-antagonisten
WO2018153900A1 (de) 2017-02-22 2018-08-30 Bayer Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit sglt-2-hemmern
WO2018153899A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit stimulatoren und/oder aktivatoren der löslichen guanylatcyclase (sgc)
WO2018153897A1 (de) 2017-02-22 2018-08-30 Bayer Pharma Aktiengesellschaft Selektive partielle adenosin a1 rezeptor-agonisten in kombination mit hcn-kanal-hemmern
JP7323913B2 (ja) * 2019-04-12 2023-08-09 国立大学法人 筑波大学 睡眠誘導剤である複素環化合物

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Also Published As

Publication number Publication date
UY29099A1 (es) 2006-04-28
PE20060589A1 (es) 2006-08-12
ECSP077296A (es) 2007-04-26
ZA200701820B (en) 2008-08-27
JP4999691B2 (ja) 2012-08-15
SV2006002218A (es) 2006-10-04
CN101056875A (zh) 2007-10-17
EP1812430B1 (de) 2009-04-15
US8691850B2 (en) 2014-04-08
IL181670A0 (en) 2007-07-04
JP2008511614A (ja) 2008-04-17
MA28869B1 (fr) 2007-09-03
US20080269300A1 (en) 2008-10-30
GT200500238A (es) 2006-04-10
BRPI0514833A (pt) 2008-06-24
DE502005007106D1 (de) 2009-05-28
EP1812430A1 (de) 2007-08-01
MX2007002470A (es) 2009-02-12
ES2324049T3 (es) 2009-07-29
AR050551A1 (es) 2006-11-01
DE102004042607A1 (de) 2006-03-09
CA2578596A1 (en) 2006-03-16
CA2578596C (en) 2012-10-23
AU2005281941A1 (en) 2006-03-16
ATE428710T1 (de) 2009-05-15
WO2006027142A1 (de) 2006-03-16
KR20070057235A (ko) 2007-06-04
TW200621765A (en) 2006-07-01

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