NO20062633L - Pyrazolderivater som proteinkinasemodulatorer - Google Patents

Pyrazolderivater som proteinkinasemodulatorer

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Publication number
NO20062633L
NO20062633L NO20062633A NO20062633A NO20062633L NO 20062633 L NO20062633 L NO 20062633L NO 20062633 A NO20062633 A NO 20062633A NO 20062633 A NO20062633 A NO 20062633A NO 20062633 L NO20062633 L NO 20062633L
Authority
NO
Norway
Prior art keywords
group
atoms
protein kinase
carbon atoms
compounds
Prior art date
Application number
NO20062633A
Other languages
English (en)
Norwegian (no)
Inventor
Valerio Berdini
Gordon Saxty
Marinus Leendert Verdonk
Steven John Woodhead
Paul Graham Wyatt
Robert George Boyle
Hannah Fiona Sore
David Winter Walker
Ian Collins
Robert Downham
Robin Arthur Ellis Carr
Original Assignee
Astex Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0329617A external-priority patent/GB0329617D0/en
Application filed by Astex Therapeutics Ltd filed Critical Astex Therapeutics Ltd
Publication of NO20062633L publication Critical patent/NO20062633L/no

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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WO2005061463A1 (en) 2005-07-07
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US9283226B2 (en) 2016-03-15
EP2228369A1 (de) 2010-09-15
US8247576B2 (en) 2012-08-21
US8691806B2 (en) 2014-04-08
AU2004303602C1 (en) 2009-05-28
EP1706385B1 (de) 2010-10-06
AU2004303602A1 (en) 2005-07-07
AU2004303602B2 (en) 2008-12-18
JP4928949B2 (ja) 2012-05-09
CY1111493T1 (el) 2015-08-05
CA2548374C (en) 2014-05-27
BRPI0418078A8 (pt) 2018-01-02
IL176400A (en) 2011-10-31
US20160250187A1 (en) 2016-09-01
MXPA06007326A (es) 2007-01-26
US20130005702A1 (en) 2013-01-03
KR20060130621A (ko) 2006-12-19
KR101164258B1 (ko) 2012-07-11
HK1097543A1 (en) 2007-06-29
JP2007516272A (ja) 2007-06-21
BRPI0418078A (pt) 2007-04-17
US20140271662A1 (en) 2014-09-18
US20110144080A1 (en) 2011-06-16
NZ547696A (en) 2009-12-24
EP1706385A1 (de) 2006-10-04
HRP20100675T1 (hr) 2011-01-31
IL176400A0 (en) 2006-10-05
PL1706385T3 (pl) 2011-03-31

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