NO20060719L - Substituerte cykloalkylaminderivater som modulatorer av kemokin reseptor aktivitet - Google Patents
Substituerte cykloalkylaminderivater som modulatorer av kemokin reseptor aktivitetInfo
- Publication number
- NO20060719L NO20060719L NO20060719A NO20060719A NO20060719L NO 20060719 L NO20060719 L NO 20060719L NO 20060719 A NO20060719 A NO 20060719A NO 20060719 A NO20060719 A NO 20060719A NO 20060719 L NO20060719 L NO 20060719L
- Authority
- NO
- Norway
- Prior art keywords
- modulators
- chemokine receptor
- receptor activity
- substituted cycloalkylamine
- cycloalkylamine derivatives
- Prior art date
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- C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
- C07C237/22—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
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- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/205—Radicals derived from carbonic acid
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- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
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- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/66—Nitrogen atoms
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- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- C07C2601/14—The ring being saturated
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US49697403P | 2003-08-21 | 2003-08-21 | |
US10/923,538 US7378409B2 (en) | 2003-08-21 | 2004-08-19 | Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity |
PCT/US2004/027195 WO2005020899A2 (en) | 2003-08-21 | 2004-08-20 | Substituted cycloalkyamine derivatives as modulators of chemokine receptor activity |
Publications (1)
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NO20060719L true NO20060719L (no) | 2006-04-27 |
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NO20060719A NO20060719L (no) | 2003-08-21 | 2006-02-14 | Substituerte cykloalkylaminderivater som modulatorer av kemokin reseptor aktivitet |
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US (1) | US7378409B2 (de) |
EP (1) | EP1656138A4 (de) |
JP (1) | JP2007502842A (de) |
IS (1) | IS8312A (de) |
NO (1) | NO20060719L (de) |
WO (1) | WO2005020899A2 (de) |
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WO2005020899A2 (en) | 2005-03-10 |
US20050054626A1 (en) | 2005-03-10 |
EP1656138A4 (de) | 2007-04-18 |
JP2007502842A (ja) | 2007-02-15 |
WO2005020899A3 (en) | 2005-06-30 |
EP1656138A2 (de) | 2006-05-17 |
US7378409B2 (en) | 2008-05-27 |
IS8312A (is) | 2006-02-20 |
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