NO20052698D0 - 4(fenylpiperazinyl-metyl)benzamid-derivater og deres anvendelse ved behandling av smerte og gasatrintestinale lidelser. - Google Patents

4(fenylpiperazinyl-metyl)benzamid-derivater og deres anvendelse ved behandling av smerte og gasatrintestinale lidelser.

Info

Publication number
NO20052698D0
NO20052698D0 NO20052698A NO20052698A NO20052698D0 NO 20052698 D0 NO20052698 D0 NO 20052698D0 NO 20052698 A NO20052698 A NO 20052698A NO 20052698 A NO20052698 A NO 20052698A NO 20052698 D0 NO20052698 D0 NO 20052698D0
Authority
NO
Norway
Prior art keywords
phenylpiperazinylmethyl
pain
gaseous
treatment
tract disorders
Prior art date
Application number
NO20052698A
Other languages
English (en)
Norwegian (no)
Other versions
NO20052698L (no
Inventor
William Brown
Christopher Walpole
Andrew Griffin
Niklas Plobeck
Paul Jones
Daniel Page
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20052698L publication Critical patent/NO20052698L/no
Publication of NO20052698D0 publication Critical patent/NO20052698D0/no

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/38—Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
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    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
NO20052698A 2002-11-07 2005-06-06 4(fenylpiperazinyl-metyl)benzamid-derivater og deres anvendelse ved behandling av smerte og gasatrintestinale lidelser. NO20052698D0 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0203303A SE0203303D0 (sv) 2002-11-07 2002-11-07 Novel Compounds
PCT/SE2003/001707 WO2004041802A1 (en) 2002-11-07 2003-11-05 4(phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain or gastrointestinal disorders

Publications (2)

Publication Number Publication Date
NO20052698L NO20052698L (no) 2005-06-06
NO20052698D0 true NO20052698D0 (no) 2005-06-06

Family

ID=20289507

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20052698A NO20052698D0 (no) 2002-11-07 2005-06-06 4(fenylpiperazinyl-metyl)benzamid-derivater og deres anvendelse ved behandling av smerte og gasatrintestinale lidelser.

Country Status (20)

Country Link
US (2) US7253173B2 (sv)
EP (1) EP1562924A1 (sv)
JP (1) JP4528128B2 (sv)
KR (1) KR20050072482A (sv)
CN (1) CN100415729C (sv)
AR (1) AR041895A1 (sv)
AU (1) AU2003278665B2 (sv)
BR (1) BR0315995A (sv)
CA (1) CA2502732A1 (sv)
IS (1) IS7863A (sv)
MX (1) MXPA05004708A (sv)
NO (1) NO20052698D0 (sv)
NZ (1) NZ539484A (sv)
PL (1) PL376894A1 (sv)
RU (1) RU2005111985A (sv)
SE (1) SE0203303D0 (sv)
TW (1) TW200418822A (sv)
UA (1) UA80988C2 (sv)
WO (1) WO2004041802A1 (sv)
ZA (1) ZA200503556B (sv)

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SE0203302D0 (sv) * 2002-11-07 2002-11-07 Astrazeneca Ab Novel Compounds
SE0203301D0 (sv) * 2002-11-07 2002-11-07 Astrazeneca Ab Novel Compounds
SE0203300D0 (sv) 2002-11-07 2002-11-07 Astrazeneca Ab Novel Compounds
SE0203303D0 (sv) * 2002-11-07 2002-11-07 Astrazeneca Ab Novel Compounds
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SE0401968D0 (sv) * 2004-08-02 2004-08-02 Astrazeneca Ab Diarylmethyl piperazine derivatives, preparations thereof and uses thereof
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US7598261B2 (en) 2005-03-31 2009-10-06 Adolor Corporation Spirocyclic heterocyclic derivatives and methods of their use
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WO2019046931A1 (en) * 2017-09-05 2019-03-14 The Royal Institution For The Advancement Of Learning/Mcgill University COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE AS INHIBITORS OF RAN GTPASE

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US7253173B2 (en) 2007-08-07
NZ539484A (en) 2007-05-31
JP4528128B2 (ja) 2010-08-18
AU2003278665A1 (en) 2004-06-07
CN1711252A (zh) 2005-12-21
US7960389B2 (en) 2011-06-14
AR041895A1 (es) 2005-06-01
WO2004041802A1 (en) 2004-05-21
AU2003278665B2 (en) 2008-05-22
EP1562924A1 (en) 2005-08-17
WO2004041802A8 (en) 2005-03-10
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CN100415729C (zh) 2008-09-03
CA2502732A1 (en) 2004-05-21
RU2005111985A (ru) 2006-01-20
BR0315995A (pt) 2005-09-27
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US20070254890A1 (en) 2007-11-01
IS7863A (is) 2005-05-25
NO20052698L (no) 2005-06-06
JP2006514002A (ja) 2006-04-27
UA80988C2 (en) 2007-11-26
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ZA200503556B (en) 2006-08-30

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