NO20052655D0 - Sammensmeltede heterocykliske forbindelser - Google Patents

Sammensmeltede heterocykliske forbindelser

Info

Publication number
NO20052655D0
NO20052655D0 NO20052655A NO20052655A NO20052655D0 NO 20052655 D0 NO20052655 D0 NO 20052655D0 NO 20052655 A NO20052655 A NO 20052655A NO 20052655 A NO20052655 A NO 20052655A NO 20052655 D0 NO20052655 D0 NO 20052655D0
Authority
NO
Norway
Prior art keywords
merged
heterocyclic compounds
heterocyclic
compounds
merged heterocyclic
Prior art date
Application number
NO20052655A
Other languages
English (en)
Other versions
NO20052655L (no
Inventor
Juan C Jaen
Xiaoqi Chen
Pingchen Fan
Leping Li
Xi Chen
Jeffrey T Mihalic
Original Assignee
Tularik Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tularik Inc filed Critical Tularik Inc
Publication of NO20052655D0 publication Critical patent/NO20052655D0/no
Publication of NO20052655L publication Critical patent/NO20052655L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
NO20052655A 2002-11-06 2005-06-02 Sammensmeltede heterocykliske forbindelser NO20052655L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42445602P 2002-11-06 2002-11-06
PCT/US2003/035543 WO2004043958A1 (en) 2002-11-06 2003-11-06 Fused heterocyclic compounds

Publications (2)

Publication Number Publication Date
NO20052655D0 true NO20052655D0 (no) 2005-06-02
NO20052655L NO20052655L (no) 2005-07-26

Family

ID=32312811

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20052655A NO20052655L (no) 2002-11-06 2005-06-02 Sammensmeltede heterocykliske forbindelser

Country Status (16)

Country Link
US (2) US7253179B2 (no)
EP (1) EP1562943A1 (no)
JP (1) JP4547266B2 (no)
KR (1) KR20050103184A (no)
CN (2) CN101134757A (no)
AU (1) AU2003285160B2 (no)
BR (1) BR0316070A (no)
CA (1) CA2505372A1 (no)
EA (1) EA009421B1 (no)
IS (1) IS7833A (no)
MX (1) MXPA05004739A (no)
NO (1) NO20052655L (no)
NZ (1) NZ540328A (no)
PL (1) PL376659A1 (no)
WO (1) WO2004043958A1 (no)
ZA (1) ZA200503654B (no)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6809104B2 (en) * 2001-05-04 2004-10-26 Tularik Inc. Fused heterocyclic compounds
US20070135425A1 (en) * 2001-05-04 2007-06-14 Amgen Inc. Fused heterocyclic compounds
AU2003285160B2 (en) 2002-11-06 2009-06-04 Amgen Inc. Fused heterocyclic compounds
AU2004209505B2 (en) 2003-02-10 2009-07-23 Banyu Pharmaceutical Co., Ltd. Melanin-concentrating hormone receptor antagonists containing piperidine derivatives as the active ingredient
DE102010025663A1 (de) * 2010-06-30 2012-01-05 Karl-Heinz Glüsenkamp Neue beta-Aminoaldehyd-Derivate, Verfahren zu ihrer Herstellung und ihre chemische Verwendung als reaktive Intermediate
CA2807538A1 (en) * 2010-08-10 2012-02-16 Abbvie Inc. Novel trpv3 modulators
WO2012129491A1 (en) 2011-03-24 2012-09-27 Abbott Laboratories Trpv3 modulators
WO2013062964A2 (en) 2011-10-24 2013-05-02 Abbvie Inc. Novel trpv3 modulators
CN106588812B (zh) * 2016-12-07 2019-02-22 烟台大学 一种酰氯制备2,4-二取代噻唑啉类化合物的方法
EA202191968A1 (ru) * 2019-01-14 2021-11-16 Кадила Хелзкэр Лимитед Новые замещенные производные сульфонилмочевины
HUP2200222A1 (hu) 2022-06-17 2023-12-28 Richter Gedeon Nyrt MCHR1 antagonisták a Prader-Willi szindróma kezelésére

Family Cites Families (55)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US23085A (en) * 1859-03-01 chandler
US176694A (en) * 1876-04-25 Improvement in screw-cutting die-stocks
US199549A (en) * 1878-01-22 Improvement in screw-propellers
JPS5825980B2 (ja) * 1976-02-12 1983-05-31 ヤマサ醤油株式会社 サイクリックヌクレオチドの定量法
EP0257701A1 (en) 1986-08-15 1988-03-02 Cedona Pharmaceuticals B.V. A process for preparing hydroxyl derivatives of compounds containing a carbazole, dibenzofurane or dibenzothiophene group
US5049655A (en) * 1989-03-22 1991-09-17 The Salk Institute For Biological Studies Melanin-concentrating hormones
JP2906654B2 (ja) 1989-11-28 1999-06-21 東レ株式会社 免疫抑制剤及びその製造方法
US5401629A (en) * 1990-08-07 1995-03-28 The Salk Institute Biotechnology/Industrial Associates, Inc. Assay methods and compositions useful for measuring the transduction of an intracellular signal
JP3160941B2 (ja) * 1991-06-17 2001-04-25 東レ株式会社 カルバゾール誘導体および免疫抑制剤
US5441956A (en) * 1991-07-05 1995-08-15 Smithkline Beecham Farmaceutici S.P.A. Hydroisoquinoline derivatives
CN1043766C (zh) 1992-09-29 1999-06-23 东丽株式会社 吲哚衍生物及其制法和它们在制备药物中的应用
US5272146A (en) * 1992-10-02 1993-12-21 The United States Of America As Represented By The United States Department Of Health And Human Services 1,2-dihydroellipticines with activity against CNS specific cancer cell lines
US5457208A (en) * 1993-06-21 1995-10-10 Regents Of The University Of Minnesota Kappa opioid receptor antagonists
US5464841A (en) 1993-11-08 1995-11-07 Univ Minnesota Use of delta opioid receptor antagonists to treat immunoregulatory disorders
US5578725A (en) 1995-01-30 1996-11-26 Regents Of The University Of Minnesota Delta opioid receptor antagonists
US5849708A (en) * 1995-06-06 1998-12-15 Joslin Diabetes Center, Inc. Promotion of eating behavior
EP0848060A3 (en) * 1996-12-11 2000-02-02 Smithkline Beecham Corporation Novel human 11CB splice variant
NZ331769A (en) 1997-01-16 2000-05-26 Toray Industries Indolomorphinan derivative and agent for curing and preventing cerebral disorder
US6555339B1 (en) 1997-04-14 2003-04-29 Arena Pharmaceuticals, Inc. Non-endogenous, constitutively activated human protein-coupled receptors
WO1999028492A1 (en) 1997-12-03 1999-06-10 Smithkline Beecham Corporation A method of finding agonist and antagonist to human 11cb splice variant
CA2334551A1 (en) 1998-06-11 1999-12-16 Merck & Co., Inc. Spiropiperidine derivatives as melanocortin receptor agonists
CA2342833A1 (en) 1998-09-17 2000-03-23 Incyte Pharmaceuticals, Inc. Human gpcr proteins
GB9822158D0 (en) 1998-10-09 1998-12-02 Nycomed Imaging As Compositions
US6991908B1 (en) 1998-12-28 2006-01-31 Takeda Chemical Industries, Ltd. Antiobestic agents methods for screening antiobestic agents and kits comprising same
US6221613B1 (en) 1998-12-31 2001-04-24 Synaptic Pharmaceutical Corporation DNA encoding a human melanin concentrating hormone receptor (MCH1) and uses thereof
WO2000049170A1 (en) 1999-02-18 2000-08-24 Smithkline Beecham Corporation MURINE 11cby RECEPTOR
CA2371821A1 (en) 1999-02-19 2000-08-24 Takeda Chemical Industries, Ltd. Novel g protein-coupled receptor protein and dna thereof
AU5260500A (en) 1999-05-19 2000-12-05 Astrazeneca Ab Assays for agonists, agonists and inverse agonists of melanin concentrating hormone (mch) binding to the somatostatin-like receptor (slc-1)
AU5869100A (en) 1999-06-08 2000-12-28 Regents Of The University Of California, The Melanin concentrating hormone receptor
WO2001005947A1 (en) 1999-07-14 2001-01-25 Merck & Co., Inc. Melanin-concentrating hormone receptor
WO2001007611A2 (en) 1999-07-26 2001-02-01 Genentech, Inc. Novel polynucleotides and method for the use thereof
EP1196572A1 (en) 1999-07-27 2002-04-17 Smithkline Beecham Plc Axor21, a g-protein coupled receptor
WO2001021169A1 (fr) 1999-09-20 2001-03-29 Takeda Chemical Industries, Ltd. Antagonistes de l'hormone de concentration de la melanine
AU7315700A (en) 1999-09-20 2001-04-24 Takeda Chemical Industries Ltd. Melanin concentrating hormone antagonist
EP1233981A4 (en) 1999-11-16 2003-02-12 Merck & Co Inc RECEPTOR COUPLED TO A G-PROTEIN
JP2001226269A (ja) 2000-02-18 2001-08-21 Takeda Chem Ind Ltd メラニン凝集ホルモン拮抗剤
JP2003532388A (ja) 2000-03-15 2003-11-05 メルク エンド カムパニー インコーポレーテッド メラニン凝集ホルモン受容体キメラおよび融合タンパク質
JP2005229804A (ja) 2000-03-24 2005-09-02 Astellas Pharma Inc 新規なメラニンコンセントレーティングホルモン受容体
US7229986B2 (en) 2000-05-16 2007-06-12 Takeda Pharmaceutical Company Ltd. Melanin-concentrating hormone antagonist
JP2004502423A (ja) 2000-07-05 2004-01-29 シナプティック・ファーマスーティカル・コーポレーション ヒトメラニン濃縮ホルモン受容体(mch1)をコードするdna及びその使用
EP1299362A4 (en) 2000-07-05 2004-11-03 Synaptic Pharma Corp SELECTIVE RECEPTOR ANTAGONISTS OF MELANINE CONCENTRATING HORMON-1 (MCH1) AND THEIR USE
AU2001269440A1 (en) 2000-07-05 2002-01-14 Takeda Chemical Industries Ltd. Method for screening mch receptor antagonist/agonist
CA2414198A1 (en) * 2000-07-06 2002-01-17 Neurogen Corporation Melanin concentrating hormone receptor ligands
CZ20031012A3 (en) 2000-10-20 2004-04-14 Pfizer Products Inc. Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
US20030022891A1 (en) 2000-12-01 2003-01-30 Anandan Palani MCH antagonists and their use in the treatment of obesity
KR20040011447A (ko) * 2000-12-22 2004-02-05 쉐링 코포레이션 피페리딘 mch 길항제 및 비만 치료에 있어서의 이의 용도
CA2441235C (en) 2001-03-21 2011-05-24 Pharmacopeia, Inc. Aryl and biaryl compounds having mch modulatory activity
US6900329B2 (en) 2001-03-21 2005-05-31 Schering Corporation MCH antagonists and their use in the treatment of obesity
DE60235617D1 (de) * 2001-04-12 2010-04-22 Pharmacopeia Llc Arly und diaryl piperidinderivate verwendbar als mch-hemmer
US6809104B2 (en) 2001-05-04 2004-10-26 Tularik Inc. Fused heterocyclic compounds
JP2004529161A (ja) * 2001-05-04 2004-09-24 トゥラリック インコーポレイテッド 縮合複素環式化合物
BR0209932A (pt) 2001-05-22 2004-10-13 Neurogen Corp Composto ou sal farmaceuticamente aceitável do mesmo, composição farmacêutica, preparação farmacêutica embalada, métodos para modular ligação de mch a um receptor de mch e de mvc, para alterar a atividade de transdução de sinal de um receptor de mch em uma célula, para tratar uma doença ou distúrbio associado com a ativação de receptor de mch patogênico obesidade e para determinar a presença ou ausência de receptor de mch em uma amostra, e, uso de um composto
DE60234116D1 (de) 2001-11-26 2009-12-03 Schering Corp Piperidin mch antagonisten und ihre verwendung in der behandlung von obesität und störungen des zentralnervensystems
CA2473236A1 (en) * 2002-01-10 2003-07-24 Neurogen Corporation Melanin concentrating hormone receptor ligands: substituted 2-(4-benzyl-piperazin-1-ylmethyl)- and 2-(4-benzyl-diazepan-1-ylmethyl)-1h-benzoimidazole analogues
AU2003285160B2 (en) * 2002-11-06 2009-06-04 Amgen Inc. Fused heterocyclic compounds

Also Published As

Publication number Publication date
EA200500770A1 (ru) 2005-12-29
PL376659A1 (pl) 2006-01-09
ZA200503654B (en) 2006-09-27
NO20052655L (no) 2005-07-26
CN1735613A (zh) 2006-02-15
AU2003285160B2 (en) 2009-06-04
IS7833A (is) 2005-05-02
US7253179B2 (en) 2007-08-07
JP4547266B2 (ja) 2010-09-22
AU2003285160A1 (en) 2004-06-03
CN101134757A (zh) 2008-03-05
CN1330651C (zh) 2007-08-08
NZ540328A (en) 2008-02-29
BR0316070A (pt) 2005-09-27
WO2004043958A1 (en) 2004-05-27
EP1562943A1 (en) 2005-08-17
US20040147538A1 (en) 2004-07-29
MXPA05004739A (es) 2005-08-02
KR20050103184A (ko) 2005-10-27
US20080058365A1 (en) 2008-03-06
CA2505372A1 (en) 2004-05-27
JP2006508130A (ja) 2006-03-09
EA009421B1 (ru) 2007-12-28

Similar Documents

Publication Publication Date Title
IS8348A (is) Samrunnin heteróhringasambönd
IS7471A (is) Ný efnasambönd
IS7879A (is) Ný efnasambönd
ATE478870T1 (de) Spiroindolinpiperidinderivate
ATE460418T1 (de) Heterocyclocarboxamidderivate
DE60330372D1 (de) Indol-3-schwefelderivate
ATE467631T1 (de) Chinuclidinamidderivate
ATE368042T1 (de) Cephemverbindungen
IS7720A (is) Píperidín-N-oxíð-afleiður
ATE517888T1 (de) Indolylmaleimid-derivate
ATE438644T1 (de) Chinazolinderivate
DK1474408T3 (da) N-Phenyl-2-pyrimidinaminderivater
NO20052655D0 (no) Sammensmeltede heterocykliske forbindelser
IS7827A (is) Ný efnasambönd
IS7381A (is) Efnasambönd
DE602004019555D1 (de) Heterocyclische 7-aminoalkylidenylchinolone und -naphthyridone
IS7414A (is) Oxó-azabísýklísk efnasambönd
ATE335729T1 (de) 3h-chinazoline -4-on derivaten
NO20045659L (no) Forbindelser
ATE423771T1 (de) Tetrahydrochinolinderivate
ATE496887T1 (de) Substituierte 5-aminomethyl-1h-pyrrol-2-carbons ureamide
DE602004007387D1 (de) 5-substituierte chinazolinonderivate
NO20023047D0 (no) Kompenseringsanordning
DE50306277D1 (de) 4-alkyl-/4-alkenyl-/4-alkinylmethyl/-1-arylcyclohexylamin-derivate
IS7906A (is) Afleiður própargýl-tríflúorómetoxý-amínó-benzóþíazóls

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application