NO20016319D0 - VLA-4 inhibitor-forbindelser - Google Patents
VLA-4 inhibitor-forbindelserInfo
- Publication number
- NO20016319D0 NO20016319D0 NO20016319A NO20016319A NO20016319D0 NO 20016319 D0 NO20016319 D0 NO 20016319D0 NO 20016319 A NO20016319 A NO 20016319A NO 20016319 A NO20016319 A NO 20016319A NO 20016319 D0 NO20016319 D0 NO 20016319D0
- Authority
- NO
- Norway
- Prior art keywords
- vla
- inhibitor compounds
- inhibitor
- compounds
- Prior art date
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- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US14160299P | 1999-06-30 | 1999-06-30 | |
US14169299P | 1999-06-30 | 1999-06-30 | |
US14160199P | 1999-06-30 | 1999-06-30 | |
PCT/US2000/018079 WO2001000206A1 (en) | 1999-06-30 | 2000-06-30 | Vla-4 inhibitor compounds |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20016319D0 true NO20016319D0 (no) | 2001-12-21 |
NO20016319L NO20016319L (no) | 2002-02-28 |
NO324892B1 NO324892B1 (no) | 2007-12-27 |
Family
ID=27385682
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20016319A NO324892B1 (no) | 1999-06-30 | 2001-12-21 | VLA-4 inhibitor-forbindelser, deres anvendelse samt farmasoytisk preparat |
Country Status (13)
Country | Link |
---|---|
EP (1) | EP1189612A4 (no) |
JP (1) | JP2003503350A (no) |
CN (1) | CN1391473A (no) |
AR (1) | AR035011A1 (no) |
AU (1) | AU781438B2 (no) |
BR (1) | BR0012068A (no) |
CA (1) | CA2369308A1 (no) |
HK (1) | HK1043318A1 (no) |
IL (1) | IL146288A0 (no) |
MX (1) | MXPA01013406A (no) |
NO (1) | NO324892B1 (no) |
TW (1) | TWI283240B (no) |
WO (1) | WO2001000206A1 (no) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001053275A2 (de) * | 2000-01-17 | 2001-07-26 | Bayer Aktiengesellschaft | Substituierte arylketone |
DE10006453A1 (de) * | 2000-02-14 | 2001-08-16 | Bayer Ag | Piperidylcarbonsäuren als Integrinantagonisten |
US6638950B2 (en) | 2000-06-21 | 2003-10-28 | Bristol-Myers Squibb Pharma Company | Piperidine amides as modulators of chemokine receptor activity |
ATE524441T1 (de) | 2000-12-28 | 2011-09-15 | Daiichi Seiyaku Co | Vla-4-inhibitoren |
CA2450722A1 (en) | 2001-06-27 | 2003-01-09 | Smithkline Beecham Corporation | Fluoropyrrolidines as dipeptidyl peptidase inhibitors |
GB0123765D0 (en) * | 2001-10-03 | 2001-11-21 | Bayer Ag | Para-amino benzoic acids |
JP2005530772A (ja) * | 2002-05-09 | 2005-10-13 | ミモトープス・プロプライエタリー・リミテッド | アミノ酸類縁体 |
KR101116627B1 (ko) | 2002-06-27 | 2012-10-09 | 노보 노르디스크 에이/에스 | 치료제로서 아릴 카르보닐 유도체 |
RU2340605C2 (ru) | 2002-06-27 | 2008-12-10 | Ново Нордиск А/С | Арилкарбонильные производные в качестве терапевтических средств |
WO2004031118A1 (ja) * | 2002-10-03 | 2004-04-15 | Ono Pharmaceutical Co., Ltd. | Lpa受容体拮抗剤 |
GB0225944D0 (en) * | 2002-11-06 | 2002-12-11 | Glaxo Group Ltd | Novel compounds |
WO2004099136A1 (ja) | 2003-05-09 | 2004-11-18 | Daiichi Pharmaceutical Co., Ltd. | ピロリジン誘導体の製造方法 |
ES2382806T3 (es) | 2003-07-24 | 2012-06-13 | Daiichi Sankyo Company, Limited | Compuesto ácido ciclohexanocarboxílico |
AR046276A1 (es) * | 2003-10-07 | 2005-11-30 | Renovis Inc | Derivados de amida como ligandos de canales ionicos y composiciones farmaceuticas y metodos que los utilizan. |
DK1723128T3 (da) | 2004-01-06 | 2013-02-18 | Novo Nordisk As | Heteroarylurinstoffer og deres anvendelse som glucokinaseaktivatorer |
JP2005350417A (ja) * | 2004-06-11 | 2005-12-22 | Dai Ichi Seiyaku Co Ltd | 還元的エーテル化法を用いたピロリジン誘導体の製造法 |
EP1781686B1 (en) * | 2004-08-16 | 2009-05-06 | Merck & Co., Inc. | Vla-4 antagonists |
JP5107724B2 (ja) | 2005-12-13 | 2012-12-26 | 第一三共株式会社 | Vla−4阻害薬 |
EP2212295A2 (en) | 2007-10-16 | 2010-08-04 | Novartis AG | 4-phenyl-5-oxo-imidazole derivatives, pharmaceutical compositions and uses therof |
WO2009118305A1 (en) * | 2008-03-26 | 2009-10-01 | Novartis Ag | Hydroxamate-based inhibitors of deacetylases b |
PL2513085T3 (pl) * | 2009-11-18 | 2017-09-29 | Suven Life Sciences Limited | Związki dwupierścieniowe jako ligandy receptora nikotynowego alfa4beta2 acetylocholiny |
EP2694472B1 (en) * | 2011-04-05 | 2020-03-11 | Takeda Pharmaceutical Company Limited | Sulfonamide derivative and use thereof |
MX2020008905A (es) | 2018-06-12 | 2020-12-03 | Vtv Therapeutics Llc | Usos terapeuticos de activadores de glucoquinasa en combinacion con insulina o analogos de insulinas. |
CR20210213A (es) | 2018-10-30 | 2021-06-24 | Gilead Sciences Inc | Derivados de quinolina como inhibidores de la integrina alfa4beta7 |
US11174256B2 (en) | 2018-10-30 | 2021-11-16 | Gilead Sciences, Inc. | Imidazopyridine derivatives |
US11179383B2 (en) | 2018-10-30 | 2021-11-23 | Gilead Sciences, Inc. | Compounds for inhibition of α4β7 integrin |
AU2019373242B2 (en) | 2018-10-30 | 2023-07-13 | Gilead Sciences, Inc. | Compounds for inhibition of alpha 4 beta 7 integrin |
AU2020228119A1 (en) | 2019-02-26 | 2021-09-16 | Bayer Aktiengesellschaft | Condensed bicyclic heterocyclic derivatives as pest control agents |
AU2020329207B2 (en) | 2019-08-14 | 2024-02-29 | Gilead Sciences, Inc. | Compounds for inhibition of alpha 4 beta 7 integrin |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6306840B1 (en) * | 1995-01-23 | 2001-10-23 | Biogen, Inc. | Cell adhesion inhibitors |
US6248713B1 (en) * | 1995-07-11 | 2001-06-19 | Biogen, Inc. | Cell adhesion inhibitors |
JP2002512625A (ja) * | 1997-05-29 | 2002-04-23 | メルク エンド カンパニー インコーポレーテッド | 細胞接着阻害薬としての複素環アミド化合物 |
WO1999020272A1 (en) * | 1997-10-21 | 1999-04-29 | Merck & Co., Inc. | Azapeptide acids as cell adhesion inhibitors |
PT1027328E (pt) * | 1997-10-31 | 2006-11-30 | Aventis Pharma Ltd | Anilidas substituídas |
AU3716499A (en) * | 1998-04-21 | 1999-11-08 | Aventis Pharma Limited | Substituted diamines and their use as cell adhesion inhibitors |
HUP0102477A3 (en) * | 1998-06-30 | 2002-08-28 | Pfizer Prod Inc | Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases and pharmaceutical compositions containing the compounds |
-
2000
- 2000-06-30 MX MXPA01013406A patent/MXPA01013406A/es active IP Right Grant
- 2000-06-30 CN CN00809510A patent/CN1391473A/zh active Pending
- 2000-06-30 TW TW089112968A patent/TWI283240B/zh not_active IP Right Cessation
- 2000-06-30 AU AU59031/00A patent/AU781438B2/en not_active Ceased
- 2000-06-30 EP EP00945035A patent/EP1189612A4/en not_active Withdrawn
- 2000-06-30 CA CA002369308A patent/CA2369308A1/en not_active Abandoned
- 2000-06-30 WO PCT/US2000/018079 patent/WO2001000206A1/en active IP Right Grant
- 2000-06-30 IL IL14628800A patent/IL146288A0/xx not_active IP Right Cessation
- 2000-06-30 BR BR0012068-5A patent/BR0012068A/pt not_active Application Discontinuation
- 2000-06-30 AR ARP000103363A patent/AR035011A1/es unknown
- 2000-06-30 JP JP2001505915A patent/JP2003503350A/ja active Pending
-
2001
- 2001-12-21 NO NO20016319A patent/NO324892B1/no unknown
-
2002
- 2002-07-09 HK HK02105102.2A patent/HK1043318A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
EP1189612A1 (en) | 2002-03-27 |
EP1189612A4 (en) | 2005-02-16 |
TWI283240B (en) | 2007-07-01 |
NO324892B1 (no) | 2007-12-27 |
NO20016319L (no) | 2002-02-28 |
MXPA01013406A (es) | 2003-09-04 |
BR0012068A (pt) | 2002-05-14 |
AU781438B2 (en) | 2005-05-26 |
HK1043318A1 (zh) | 2002-09-13 |
AR035011A1 (es) | 2004-04-14 |
CA2369308A1 (en) | 2001-01-04 |
AU5903100A (en) | 2001-01-31 |
IL146288A0 (en) | 2002-07-25 |
WO2001000206A1 (en) | 2001-01-04 |
CN1391473A (zh) | 2003-01-15 |
JP2003503350A (ja) | 2003-01-28 |
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