NO20002548L - Nye substituerte dimere forbindelser, en fremgangsmÕte ved deres fremstilling og farmasøytiske sammensetninger som inneholder dem - Google Patents
Nye substituerte dimere forbindelser, en fremgangsmÕte ved deres fremstilling og farmasøytiske sammensetninger som inneholder demInfo
- Publication number
- NO20002548L NO20002548L NO20002548A NO20002548A NO20002548L NO 20002548 L NO20002548 L NO 20002548L NO 20002548 A NO20002548 A NO 20002548A NO 20002548 A NO20002548 A NO 20002548A NO 20002548 L NO20002548 L NO 20002548L
- Authority
- NO
- Norway
- Prior art keywords
- nr1c
- nr2r3
- preparation
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
- C07D339/08—Six-membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrane Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Furan Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9906331A FR2793793B1 (fr) | 1999-05-19 | 1999-05-19 | Nouveaux derives dimeriques substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20002548D0 NO20002548D0 (no) | 2000-05-18 |
NO20002548L true NO20002548L (no) | 2000-11-20 |
Family
ID=9545746
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20002548A NO20002548L (no) | 1999-05-19 | 2000-05-18 | Nye substituerte dimere forbindelser, en fremgangsmÕte ved deres fremstilling og farmasøytiske sammensetninger som inneholder dem |
Country Status (21)
Country | Link |
---|---|
US (1) | US6310074B1 (de) |
EP (1) | EP1057826B1 (de) |
JP (1) | JP3688552B2 (de) |
KR (1) | KR100472520B1 (de) |
CN (1) | CN1128142C (de) |
AT (1) | ATE237610T1 (de) |
AU (1) | AU766322B2 (de) |
BR (1) | BR0003313A (de) |
DE (1) | DE60002126T2 (de) |
DK (1) | DK1057826T3 (de) |
EA (1) | EA003391B1 (de) |
ES (1) | ES2197062T3 (de) |
FR (1) | FR2793793B1 (de) |
HK (1) | HK1030937A1 (de) |
HU (1) | HUP0001961A3 (de) |
NO (1) | NO20002548L (de) |
NZ (1) | NZ504613A (de) |
PL (1) | PL340165A1 (de) |
PT (1) | PT1057826E (de) |
SI (1) | SI1057826T1 (de) |
ZA (1) | ZA200002490B (de) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR0316962A (pt) * | 2002-12-03 | 2005-10-25 | Hoffmann La Roche | Aminoalcoxiindóis como ligantes para o receptor de 5-ht6 para o tratamento de distúrbios do snc |
PL1696920T3 (pl) | 2003-12-19 | 2015-03-31 | Plexxikon Inc | Związki i sposoby opracowywania modulatorów Ret |
US7498342B2 (en) * | 2004-06-17 | 2009-03-03 | Plexxikon, Inc. | Compounds modulating c-kit activity |
BRPI0610066A2 (pt) * | 2005-05-17 | 2010-05-25 | Plexxikon Inc | compostos que modulam atividade de c-kit e c-fms e usos para estes |
BRPI0611863B1 (pt) * | 2005-06-22 | 2021-11-23 | Plexxikon, Inc | Composto, bem como composição e kit compreendendo o mesmo, composto intermediário na preparação do mesmo, método para tratamento e uso do mesmo |
WO2008063888A2 (en) | 2006-11-22 | 2008-05-29 | Plexxikon, Inc. | Compounds modulating c-fms and/or c-kit activity and uses therefor |
PE20121126A1 (es) * | 2006-12-21 | 2012-08-24 | Plexxikon Inc | Compuestos pirrolo [2,3-b] piridinas como moduladores de quinasa |
WO2008079909A1 (en) * | 2006-12-21 | 2008-07-03 | Plexxikon, Inc. | Pyrrolo [2,3-b] pyridines as kinase modulators |
AU2007336811A1 (en) | 2006-12-21 | 2008-07-03 | Plexxikon, Inc. | Compounds and methods for kinase modulation, and indications therefor |
BRPI0814423B1 (pt) | 2007-07-17 | 2022-04-19 | Plexxikon, Inc | Compostos que modulam quinase e composição farmacêutica compreendendo os mesmos |
JP2011529477A (ja) * | 2008-07-30 | 2011-12-08 | フエルレル インターナショナル,ソシエダッド アノニマ | 1,6−ジヒドロ−2h−3−オキサ−6−アザ−as−インダセン化合物 |
AR078033A1 (es) | 2009-04-03 | 2011-10-12 | Plexxikon Inc | Una dispersion solida, que contiene al compuesto {3-[5-(4-(cloro-fenil)-1h-pirrolo[2,3-b]piridina-3-carbonil]-2,4-difluor-fenil}-amida del acido propano-1-sulfonico, composiciones y formulaciones que comprenden a dicha dispersion solida; metodos para fabricar dicha dispersion solida, formas 1 y 2 de |
US8329724B2 (en) | 2009-08-03 | 2012-12-11 | Hoffmann-La Roche Inc. | Process for the manufacture of pharmaceutically active compounds |
ES2633317T3 (es) | 2009-11-06 | 2017-09-20 | Plexxikon, Inc. | Compuestos y métodos para la modulación de quinasas, e indicaciones para ello |
MA34948B1 (fr) | 2011-02-07 | 2014-03-01 | Plexxikon Inc | Composes et procedes de modulation de kinase, et leurs indications |
TWI558702B (zh) | 2011-02-21 | 2016-11-21 | 普雷辛肯公司 | 醫藥活性物質的固態形式 |
US9150570B2 (en) | 2012-05-31 | 2015-10-06 | Plexxikon Inc. | Synthesis of heterocyclic compounds |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SU1639427A3 (ru) * | 1987-07-03 | 1991-03-30 | Глэксо Груп Лимитед (Фирма) | Способ получени производных индола или их фармацевтически приемлемых солей |
FR2658818B1 (fr) * | 1990-02-27 | 1993-12-31 | Adir Cie | Nouveaux derives a structure naphtalenique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
EP0543584B1 (de) * | 1991-11-18 | 1996-05-22 | Lilly Industries Limited | Benzo(b)thiophen-2-carboxamide zur Behandlung von Krankheiten des Zentralnervensystems |
FR2689124A1 (fr) * | 1992-03-27 | 1993-10-01 | Adir | Nouvelles naphtylalkylamines, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent. |
FR2696453B1 (fr) * | 1992-10-02 | 1994-12-23 | Adir | Nouveaux arylalkyl(thio)amides, leur procédé de préparation, et les compositions pharmaceutiques qui les contiennent. |
EP0675109A1 (de) * | 1992-12-21 | 1995-10-04 | Taisho Pharmaceutical Co. Ltd | N-substituiertes indolderivat |
DK0767782T3 (da) * | 1994-06-29 | 2002-02-18 | Pfizer | Aryl- og heteroarylalkoxynaphthalenderivater |
FR2731223A1 (fr) * | 1995-03-02 | 1996-09-06 | Pf Medicament | Nouveaux derives bi-tryptaminiques, leur procede de preparation et leur utilisation a titre de medicaments |
-
1999
- 1999-05-19 FR FR9906331A patent/FR2793793B1/fr not_active Expired - Fee Related
-
2000
- 2000-05-18 PL PL00340165A patent/PL340165A1/xx not_active Application Discontinuation
- 2000-05-18 NO NO20002548A patent/NO20002548L/no not_active Application Discontinuation
- 2000-05-18 HU HU0001961A patent/HUP0001961A3/hu unknown
- 2000-05-18 NZ NZ504613A patent/NZ504613A/en unknown
- 2000-05-18 US US09/573,704 patent/US6310074B1/en not_active Expired - Fee Related
- 2000-05-18 EA EA200000431A patent/EA003391B1/ru not_active IP Right Cessation
- 2000-05-19 ZA ZA200002490A patent/ZA200002490B/xx unknown
- 2000-05-19 KR KR10-2000-0026963A patent/KR100472520B1/ko not_active IP Right Cessation
- 2000-05-19 CN CN00120095A patent/CN1128142C/zh not_active Expired - Fee Related
- 2000-05-19 AU AU35420/00A patent/AU766322B2/en not_active Ceased
- 2000-05-19 BR BR0003313-8A patent/BR0003313A/pt not_active Application Discontinuation
- 2000-05-19 JP JP2000147379A patent/JP3688552B2/ja not_active Expired - Fee Related
- 2000-05-22 SI SI200030081T patent/SI1057826T1/xx unknown
- 2000-05-22 DE DE60002126T patent/DE60002126T2/de not_active Expired - Fee Related
- 2000-05-22 ES ES00610050T patent/ES2197062T3/es not_active Expired - Lifetime
- 2000-05-22 DK DK00610050T patent/DK1057826T3/da active
- 2000-05-22 EP EP00610050A patent/EP1057826B1/de not_active Expired - Lifetime
- 2000-05-22 AT AT00610050T patent/ATE237610T1/de not_active IP Right Cessation
- 2000-05-22 PT PT00610050T patent/PT1057826E/pt unknown
-
2001
- 2001-03-12 HK HK01101746A patent/HK1030937A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CN1128142C (zh) | 2003-11-19 |
CN1277962A (zh) | 2000-12-27 |
AU3542000A (en) | 2000-11-23 |
FR2793793A1 (fr) | 2000-11-24 |
ZA200002490B (en) | 2000-11-20 |
NO20002548D0 (no) | 2000-05-18 |
SI1057826T1 (en) | 2003-08-31 |
EP1057826A1 (de) | 2000-12-06 |
PT1057826E (pt) | 2003-08-29 |
ES2197062T3 (es) | 2004-01-01 |
EA003391B1 (ru) | 2003-04-24 |
EA200000431A2 (ru) | 2000-12-25 |
BR0003313A (pt) | 2001-03-13 |
HUP0001961A3 (en) | 2002-10-28 |
DE60002126D1 (de) | 2003-05-22 |
NZ504613A (en) | 2001-06-29 |
JP3688552B2 (ja) | 2005-08-31 |
FR2793793B1 (fr) | 2004-02-27 |
PL340165A1 (en) | 2000-11-20 |
DE60002126T2 (de) | 2004-03-18 |
HU0001961D0 (en) | 2000-07-28 |
KR20010029729A (ko) | 2001-04-16 |
AU766322B2 (en) | 2003-10-16 |
KR100472520B1 (ko) | 2005-03-07 |
HK1030937A1 (en) | 2001-05-25 |
DK1057826T3 (da) | 2003-07-21 |
EA200000431A3 (ru) | 2001-02-26 |
HUP0001961A2 (hu) | 2001-08-28 |
JP2001011035A (ja) | 2001-01-16 |
US6310074B1 (en) | 2001-10-30 |
EP1057826B1 (de) | 2003-04-16 |
ATE237610T1 (de) | 2003-05-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |